UBP 301CAS: 569371-10-4
MF: C15H14IN3O6
MW: 459.2
A kainate potent receptor antagonist.

UBP 301 (CAS 569371-10-4)

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Synonym: (αS)-α-Amino-3-[(4-carboxyphenyl)methyl]-3,4-dihydro-5-iodo-2,4-dioxo-1(2H)-pyrimidinepropanoic acid
Application: A kainate potent receptor antagonist
CAS Number: 569371-10-4
Purity: ≥99%
Molecular Weight: 459.2
Molecular Formula: C15H14IN3O6
* Refer to Certificate of Analysis for lot specific data (including water content).
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UBP 301 is a kainate potent receptor (GluR and KA) antagonist (apparent Kd = 5.94 mM). Displays ~ 30-fold selectivity over GluR (AMPA) receptors.


References

1. More, J.C., et al. 2003. Br. J. Pharmacol. 138: 1093-1100.

Physical State :
Solid
Solubility :
Soluble in DMSO (5 mM with gentle warming).
Storage :
Store at 4° C
Melting Point :
335.65° C (Predicted)
Boiling Point :
~636.1° C at 760 mmHg (Predicted)
Density :
~2.0 g/cm3 (Predicted)
Refractive Index :
n20D 1.75 (Predicted)
IC50 :
Glutamate receptor ionotropic, AMPA: IC50 = 164 µM (rat)
Ki Data :
Glutamate receptor ionotropic, AMPA: Ki>100 µM (rat); Glutamate receptor ionotropic kainate 2: Ki>100 µM (rat)
pK Values :
pKa: 2.12 (Predicted), pKb: 9.03 (Predicted)
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
PubChem CID :
6604913
MDL Number :
MFCD06411591
SMILES :
C1=CC(=CC=C1CN2C(=O)C(=CN(C2=O)C[[email protected]@H](C(=O)O)N)I)C(=O)O

Download SDS (MSDS)

Certificate of Analysis

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