PSB 0788A potent and selective Adenosine A2B-R antagonist

PSB 0788 (CAS 1027513-54-7)

  • bvseo_sdk, java_sdk, bvseo-3.2.0
  • CLOUD, getAggregateRating, 86ms
  • bvseo-msg: The resource to the URL or file is currently unavailable.;
Synonym: 8-[4-[4-(4-Chlorobenzyl)piperazide-1-sulfonyl)phenyl]]-1-propylxanthine
Application: A potent and selective Adenosine A2B-R antagonist
CAS Number: 1027513-54-7
Molecular Weight: 543.04
Molecular Formula: C25H27ClN6O4S
* Refer to Certificate of Analysis for lot specific data (including water content).
Submit a review for this product and receive 15 CruzCredits

PSB 0788 is a potent and selective Adenosine A2B-R antagonist (IC50 = 3.64 nM at human Adenosine A2B-R). It displays > 100-fold selectivity over human Adenosine A1-R, human Adenosine A2A-R and human Adenosine A3-R.

Physical State :
Solubility :
Soluble in DMSO (100 mM).
Storage :
Store at 4° C
Density :
1.41 g/cm3 (Predicted)
Refractive Index :
n20D 1.65 (Predicted)
IC50 :
Adenosine A2B-R: IC50 = 3.64 nM (human)
Ki Data :
Adenosine A2B-R: Ki= 0.39 nM (human); Adenosine A1 receptor: Ki= 386 nM (rat); Adenosine A3-R: Ki>1 µM (human); Adenosine A2a receptor: Ki= 1.73 µM (rat); Adenosine A1-R: Ki= 2.24 µM (human)
pK Values :
pKa: 7.37 (Predicted), pKb: 5.05 (Predicted)
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
PubChem CID :
MDL Number :

Download SDS (MSDS)

Certificate of Analysis

Adobe Acrobat Reader is required to reliably view,
print and comment on PDF documents

日本で購入を検討しています。日本での販売価格はいくらになりますでしょうか? ご教授いただけますと幸いです。

Asked by: tkht
Thank you for your question. Please contact our local distributors in Japan to confirm the price and lead time. The contact information can be found below. お問い合わせを頂きまして、誠にありがとうございました。お手数ですが、日本での購入は弊社の日本での代理店へお勧めします。納期と日本円での価格は代理店へご連絡ください。 代理店は下記の四社となります。
Answered by: Technical Support 8
Date published: 2017-06-20
  • y_2019, m_9, d_23, h_24CST
  • bvseo_bulk, prod_bvqa, vn_bulk_2.0.13
  • cp_1, bvpage1
  • co_hasquestionsanswers, tq_1
  • loc_en_US, sid_204217, prod, sort_[SortEntry(order=LAST_APPROVED_ANSWER_SUBMISSION_TIME, direction=DESCENDING)]
  • clientName_scbt
  • bvseo_sdk, java_sdk, bvseo-3.2.0
  • CLOUD, getContent, 140ms
  • bvseo_sdk, java_sdk, bvseo-3.2.0
  • CLOUD, getReviews, 38ms
  • bvseo-msg: The resource to the URL or file is currently unavailable.;

Santa Cruz Biotechnology, Inc. is a world leader in the development of products for the biomedical research market. Call us Toll Free at 1-800-457-3801.
Copyright © 2007-2019 Santa Cruz Biotechnology, Inc. All Rights Reserved. "Santa Cruz Biotechnology", and the Santa Cruz Biotechnology, Inc. logo, "Santa Cruz Animal Health", "San Juan Ranch", "Supplement of Champions", the San Juan Ranch logo, "Ultracruz", "Chemcruz", "Immunocruz", "Exactacruz", and "EZ Touch" are registered trademarks of Santa Cruz Biotechnology, Inc.
All trademarks are the property of their respective owners.