GR 103691A potent and selective receptor antagonist for D3DR

GR 103691 (CAS 162408-66-4)

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Synonym: 4′-Acetyl-N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-[1,1′-biphenyl]-4-carboxamide
Application: A potent and selective receptor antagonist for D3DR
CAS Number: 162408-66-4
Purity: ≥98%
Molecular Weight: 485.63
Molecular Formula: C30H35N3O3
* Refer to Certificate of Analysis for lot specific data (including water content).
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GR 103691 is an effective and selective receptor antagonist of the D3DR (dopamine D3 receptor). GR 103691 was shown to have higher selectivity for D3DR (dopamine D3 receptor) over the D2DR (dopamine D2 receptor) and D4DR (dopamine D4 receptor) sites by greater than 100-fold.

Physical State :
Solid
Solubility :
Soluble in DMSO (>5 mg/ml at 60° C).
Storage :
Store at 4° C
Melting Point :
~294.22° C (Predicted)
Boiling Point :
~688.72° C at 760 mmHg (Predicted)
Density :
~1.1 g/cm3 (Predicted)
Refractive Index :
n20D 1.58 (Predicted)
Ki Data :
D3DR: Ki= 0.32 nM (human)
pK Values :
pKb: 7.87
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
WGK Germany :
3
PubChem CID :
4302960
MDL Number :
MFCD00936840
SMILES :
CC(=O)C1=CC=C(C=C1)C2=CC=C(C=C2)C(=O)NCCCCN3CCN(CC3)C4=CC=CC=C4OC

Download SDS (MSDS)

Certificate of Analysis

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