G Protein AntagonistA G protein inhibitor of M2 muscarinic cholinergic receptors.

G Protein Antagonist (CAS 143675-79-0)

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Synonym: pGlu-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH2
Application: A G protein inhibitor of M2 muscarinic cholinergic receptors.
CAS Number: 143675-79-0
Purity: ≥90%
Molecular Weight: 1093.26
Molecular Formula: C57H64N12O9S
* Refer to Certificate of Analysis for lot specific data (including water content).

This product has been shown to inhibit the activation of Gαi or Gαo by M2 muscarinic cholinergic receptor.


References

1. Mukai, H., et al. 1992. J. Biol. Chem. 267: 16237-16243. PMID: 1379592

Physical State :
Solid
Solubility :
Soluble in water, and 30% acetonitrile / water (1 mg/ml).
Storage :
Desiccate at -20° C
Density :
~1.37 g/cm3 (Predicted)
Refractive Index :
n20D ~1.68 (Predicted)
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
WGK Germany :
3
PubChem CID :
44134914
MDL Number :
MFCD03444578
SMILES :
CSCC[C@H](NC(=O)[C@H](NC(=O)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](NC(=O)[C@H](CCC(=O)N)NC(=O)[C@@H]1CCC(=O)N1)Cc1c[nH]c2ccccc12)Cc1c[nH]c2ccccc12)Cc1c[nH]c2ccccc12)C(=O)N

Download SDS (MSDS)

Certificate of Analysis

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