CinanserinA serotonin 5-HT2 antagonist

Cinanserin (CAS 1166-34-3)

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Application: A serotonin 5-HT2 antagonist
CAS Number: 1166-34-3
Molecular Weight: 340.5
Molecular Formula: C20H24N2OS
* Refer to Certificate of Analysis for lot specific data (including water content).
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Cinanserin is a SR (serotonin 5-HT2) antagonis1,2.


References

1: J.E. Leysen et al. Life. Sci. 1981 28 1015 2: P.J. Pauwels et al. Life. Sci. 1990 47 2009

Physical State :
Solid
Solubility :
Soluble in ethanol, and methanol.
Storage :
Store at -20° C
IC50 :
Serotonin 2b (5-HT2b) receptor: IC50 = 2 nM (Rattus norvegicus); Serotonin 2a (5-HT2a) receptor: IC50 = 14.8 nM (Rattus norvegicus); Serotonin 2c (5-HT2c) receptor: IC50 = 2 nM (Rattus norvegicus)
Ki Data :
Serotonin 2a (5-HT2a) receptor: Ki= 4.5 nM (Rattus norvegicus); Serotonin 2c (5-HT2c) receptor: Ki= 3.8 nM (Rattus norvegicus); Serotonin 2b (5-HT2b) receptor: Ki= 4 nM (Rattus norvegicus); Serotonin 1b (5-HT1b) receptor: Ki= 1000 nM (Rattus norvegicus)
pK Values :
pKa: 13.46, pKb: 9.38
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
PubChem CID :
5475158
MDL Number :
MFCD00600248
SMILES :
CN(C)CCCSC1=CC=CC=C1NC(=O)/C=C/C2=CC=CC=C2

Download SDS (MSDS)

Certificate of Analysis

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