CGP 46381 CAS: 123691-14-5
MF: C10H22NO2P
MW: 219.26
A selective GABAB receptor antagonist.

CGP 46381 (CAS 123691-14-5)

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Application: CGP 46381 is a selective GABAB receptor antagonist
CAS Number: 123691-14-5
Molecular Weight: 219.26
Molecular Formula: C10H22NO2P
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data (including water content).
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CGP 46381 is a selective GABAB receptor antagonist (IC50 = 4.9 μM).

Physical State :
Solid
Solubility :
Soluble in water (100 mM).
Storage :
Store at room temperature
Melting Point :
84.78° C (Predicted)
Boiling Point :
441.21° C at 760 mmHg (Predicted)
Density :
1.08 g/cm3 (Predicted)
Refractive Index :
n20D 1.49 (Predicted)
IC50 :
GABA-B receptor 1: IC50 = 4 µM (rat)
pK Values :
pKa: 2.88 (Predicted), pKb: 10.44 (Predicted)
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
PubChem CID :
MDL Number :
MFCD00910404
SMILES :
C1CCC(CC1)CP(=O)(CCCN)O

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Certificate of Analysis

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CGP 46381 (CAS 123691-14-5)  Product Citations

See how others have used CGP 46381 (CAS 123691-14-5). Click on the entry to view the PubMed entry .

Citations 1 to 3 of 3 total

PMID: # 25241062  Neuroscience. 254-61.

PMID: # 25114926  Biomed Res Int. 871735.

PMID: # 24682435  Heart Vessels. 249-57.

Citations 1 to 3 of 3 total
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