BIBP 3226 trifluoroacetate is a mixed NPY1-R (non-peptide neuropeptide Y Y1 receptor) and NPFF (neuropeptide FF) receptor inhibitor (Ki values are 1.1, 79, 108, > 1000, > 1000 and >1000 for rNPY1-R, hNPFF2, rNPFF, rNPY2-R, rNPY4-R and rNPY5-R respectively). Following i.c.v. administration, BIBP 3226 trifluoroacetate produces an anxiogenic-like effect in rats.
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Soluble in water (10 mM).
Store at -20° C
n20D 1.63 (Predicted)
α20/D 21.4°, c = 1 in water
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
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