EGFR阻害剤

Santa Cruz Biotechnology now offers a broad range of EGFR Inhibitors. The EGF receptor family comprises several related receptor tyrosine kinases that are frequently overexpressed in a variety of carcinomas. Upregulation of EGFR is associated with tumor progression. Abrogation of EGFR may be achieved with the use of EGFR Inhibitors with potential results in cell cycle arrest, apoptosis or dedifferentiation of cancer cells. EGFR Inhibitors offered by Santa Cruz inhibit EGFR and, in some cases, other receptor tyrosine kinases and tumor progression related proteins. View detailed EGFR Inhibitor specifications, including EGFR Inhibitor CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

indicates a highly recommended product based on customer preference.

製品名/アプリケーション CAS カタログ # 数量 価格 引用文献 レーティング
Erlotinib Hydrochloride
Erlotinib Hydrochloride is a HER-1/EGFR tyrosine kinase inhibitor
183319-69-9 sc-202154
sc-202154A
10 mg
25 mg
$68.00
$112.00
27
(1)
Gefitinib
Gefitinib is an EGFR-tyrosine kinase inhibitor
184475-35-2 sc-202166
sc-202166A
sc-202166B
sc-202166C
100 mg
250 mg
1 g
5 g
$50.00
$100.00
$200.00
$325.00
47
(2)
AG-490
AG-490 is a tyrosine kinase inhibitor of JAK2, EGFR, JAK3 and Neu
133550-30-8 sc-202046
sc-202046A
10 mg
50 mg
$78.00
$312.00
23
(1)
Lapatinib ditosylate
Lapatinib ditosylate is a selective and effective inhibitor of ErbB-2 and EGFR dual tyrosine kinases
388082-78-8 sc-202205
sc-202205A
sc-202205B
10 mg
25 mg
5 mg
$63.00
$105.00
$38.00
14
(1)
Tyrphostin AG 1478
Tyrphostin AG 1478 is a potent and selective inhibitor of EGFR
175178-82-2 sc-200613
sc-200613A
5 mg
25 mg
$87.00
$400.00
13
(1)
CL-387,785
CL-387,785 is an irreversible inhibitor of EGF-receptor kinase activity
194423-06-8 sc-221429
1 mg
$134.00
0
(1)
Hypericin
Hypericin is a kinase inhibitor with antiviral activity
548-04-9 sc-3530
sc-3530A
1 mg
5 mg
$58.00
$200.00
10
(1)
Erbstatin Analog
Erbstatin Analog is a stable inhibitor of EGFR tyrosine kinase
63177-57-1 sc-200511
sc-200511A
5 mg
25 mg
$81.00
$299.00
4
(1)
CGP-74514A hydrochloride
CGP-74514A hydrochloride is a Cdk inhibitor
1173021-98-1 sc-300344
sc-300344A
5 mg
25 mg
$220.00
$796.00
0
(1)
Herbimycin A
Herbimycin A is an inhibitor of c-Abl, HSP 90, c-Src, c-Yes, Fes, and Ros
70563-58-5 sc-3516
sc-3516A
100 µg
1 mg
$166.00
$950.00
11
(1)
PD 168393
PD 168393 is a potent, cell-permeable, irreversible inhibitor of EGFR
194423-15-9 sc-222138
1 mg
$162.00
3
(1)
Daphnetin
Daphnetin is a coumarin analog that acts as an inhibitor of several protein kinases
486-35-1 sc-203022
10 mg
$80.00
0
(1)
Afatinib
Afatinib is an irreversible and potent EGFR/Neu inhibitor, inhibits EGFR phosphorylation.
439081-18-2 sc-364398
sc-364398A
5 mg
10 mg
$100.00
$180.00
3
(2)
Lapatinib
Lapatinib is an antineoplastic agent used in breast cancer research
231277-92-2 sc-353658
100 mg
$399.00
23
(1)
PKC-412
PKC-412 is a broad spectrum tyrosine kinase inhibitor
120685-11-2 sc-200691
sc-200691A
1 mg
5 mg
$114.00
$450.00
8
(1)
PD 174265
PD 174265 is a potent, cell-permeable, reversible, and selective inhibitor of EGFR tyrosine kinase activity
216163-53-0 sc-204170
1 mg
$137.00
2
(1)
Tyrphostin 51
Tyrphostin 51 is a potent inhibitor of EGFRK activity showing mixed competitive inhibition with ATP and substrate1-3.
122520-90-5 sc-200545
sc-200545A
5 mg
25 mg
$58.00
$299.00
0
(1)
Butein
Butein is inhibits the tyrosine kinase activity of the EGF receptor and p60c-src
487-52-5 sc-202510
sc-202510A
5 mg
50 mg
$169.00
$300.00
4
(1)
Vatalanib Dihydrochloride
Vatalanib Dihydrochloride is a potent inhibitor of EGFR- and RET-dependent tumor cell proliferation and survival
212141-51-0 sc-202379
sc-202379A
5 mg
25 mg
$125.00
$374.00
0
(1)
PP 3
PP 3 is a negative control for the Src family protein tyrosine kinase inhibitor PP2
5334-30-5 sc-203213
sc-203213A
sc-203213B
1 mg
5 mg
10 mg
$80.00
$127.00
$176.00
1
(1)
Tyrphostin 47
Tyrphostin 47 is a potent inhibitor of EGFR kinase activity
122520-86-9 sc-200543
sc-200543A
5 mg
25 mg
$77.00
$309.00
4
(1)
AG 494
AG 494 is a potent and selective inhibitor of EGFR tyrosine kinase
133550-35-3 sc-202043
sc-202043A
10 mg
50 mg
$69.00
$255.00
0
(1)
Tyrphostin AG 112
Tyrphostin AG 112 is an EGFR inhibitor
144978-82-5 sc-222381
sc-222381A
sc-222381B
sc-222381C
1 mg
5 mg
25 mg
50 mg
$23.00
$50.00
$200.00
$350.00
0
(0)
WHI-P 154
WHI-P 154 is a JAK3 inhibitor which inhibits other common kinases
211555-04-3 sc-204395
sc-204395A
10 mg
50 mg
$109.00
$615.00
0
(1)
RPI-1
RPI-1 is a cell-permeable ATP-competitive tyrosine kinase inhibitor
269730-03-2 sc-255524
sc-255524A
5 mg
10 mg
$150.00
$182.00
4
(1)
AZD8931
AZD8931 is a potent inhibitor of EGFR phosphorylation
848942-61-0 sc-364426
sc-364426A
5 mg
10 mg
$255.00
$480.00
0
(0)
CUDC-101
CUDC-101 is a potent inhibitor to HDAC, EGFR and HER2
1012054-59-9 sc-364474
sc-364474A
10 mg
50 mg
$190.00
$700.00
0
(0)
Tyrphostin A1
Tyrphostin A1 is an inactive Tyrphostin used as a negative control for Tyrphostin A23
2826-26-8 sc-3559
sc-3559A
25 mg
100 mg
$147.00
$179.00
1
(0)
Compound 56
Compound 56 is a potent and specific inhibitor of the tyrosine kinase activity of the epidermal growth factor
171745-13-4 sc-203430
500 µg
$164.00
2
(1)
XL647
XL647 is a potent and selective EGFR phosphorylation inhibitor
651031-01-5 sc-364659
sc-364659A
5 mg
10 mg
$305.00
$560.00
1
(0)
AG 43
AG 43 is a useful negative control in EGFR tyrosine kinase assays
5553-97-9 sc-202916
5 mg
$52.00
0
(0)
(+)shy-Aeroplysinin-1
(+)-Aeroplysinin-1 is a compound that is an inhibitor of EGFR kinase
28656-91-9 sc-202445
100 µg
$36.00
0
(1)
Lavendustin C
Lavendustin C is an inhibitor of CaMKII
125697-93-0 sc-202207
sc-202207B
sc-202207A
sc-202207C
1 mg
5 mg
10 mg
50 mg
$82.00
$180.00
$320.00
$1,400.00
0
(1)
PD 153035
PD 153035 is an extremely potent and specific inhibitor of EGFR tyrosine kinase activity
153436-54-5 sc-205909
5 mg
$68.00
3
(1)
OSI-420, Free Base (Desmethyl Erlotinib)
OSI-420, Free Base (Desmethyl Erlotinib) is a metabolite of Erlotinib
183321-86-0 sc-212485
1 mg
$254.00
1
(1)
WZ 4002
WZ 4002 is an EGFR phosphorylation inhibitor
1213269-23-8 sc-364655
sc-364655A
10 mg
50 mg
$180.00
$744.00
1
(2)
Tyrphostin B44, (+) enantiomer
Tyrphostin B44, (+) enantiomer is an EGFR kinase inhibitor
133550-37-5 sc-203305
5 mg
$30.00
0
(0)
Angiogenesis Inhibitor
Angiogenesis Inhibitor is a cell-permeable indolinone
186611-44-9 sc-221253
10 mg
$198.00
0
(0)
PD 161570
PD 161570 is a selective FGFR inhibitor
192705-80-9 sc-361284
sc-361284A
5 mg
25 mg
$112.00
$446.00
0
(0)
Neratinib
Neratinib is a potent and selective inhibitor of EGFR and HER2
698387-09-6 sc-364549
sc-364549A
sc-364549B
sc-364549C
sc-364549D
5 mg
25 mg
100 mg
500 mg
1 g
$80.00
$200.00
$360.00
$720.00
$1,200.00
1
(1)
HDS 029
HDS 029 is A potent inhibitor of EGF receptor family
881001-19-0 sc-203995
sc-203995A
1 mg
10 mg
$105.00
$215.00
0
(0)
Erlotinib-d6, Hydrochloride Salt
Erlotinib-d6, Hydrochloride Salt is a labeled form of Erlontinib HCl, a potent EGFR autophosphorylation inhibitior
sc-218329
1 mg
$180.00
6
(0)
Lavendustin C methyl ester
Lavendustin C methyl ester is an inhibitor of EGFR tyrosine kinase activity
sc-221838
sc-221838A
1 mg
5 mg
$26.00
$137.00
0
(0)
Lapatinib-13C2,15N Ditosylate
Lapatinib-13C2,15N Ditosylate is an inhibitor of ErbB1 and ErbB2 tyrosine kinases
sc-280905
500 µg
$250.00
0
(0)
JAK3 Inhibitor V
JAK3 Inhibitor V is a selective JAK3 inhibitor
4452-06-6 sc-295218
10 mg
$239.00
0
(0)
RO 106-9920
RO 106-9920 is a NF-kB-dependent cytokine expression, 5-LO, and EGFR inhibitor
62645-28-7 sc-203240
sc-203240A
1 mg
5 mg
$135.00
$575.00
5
(1)
Tyrphostin A25
Tyrphostin A25 is a cell-permeable, reversible, and competitive protein tyrosine kinase (PTK) substrate inhibitor
118409-58-8 sc-3555A
sc-3555
5 mg
25 mg
$67.00
$276.00
8
(1)
Tyrphostin AG 99
Tyrphostin AG 99 is a potent, cell-permeable and reversible inhibitor of EGFR and EGF-dependent cell proliferation
118409-59-9 sc-202847
sc-202847A
5 mg
25 mg
$54.00
$184.00
0
(1)
Lavendustin A
Lavendustin A is a selective and potent inhibitor of the receptor tyrosine kinase
125697-92-9 sc-200539
sc-200539A
1 mg
5 mg
$116.00
$456.00
0
(1)
Tyrphostin B42
Tyrphostin B42 is a potent JAK2 inhibitor
133550-30-8 sc-3556
5 mg
$26.00
3
(1)
AG 555
AG 555 is a potent epidermal growth factor receptor kinase inhibitor
133550-34-2 sc-203500
sc-203500A
10 mg
50 mg
$69.00
$330.00
3
(1)
AG 556
AG 556 is inhibitor of EGFR kinase autophosphorylation over HER1/2 autophosphorylation
133550-41-1 sc-202044
sc-202044A
5 mg
25 mg
$30.00
$62.00
0
(0)
RG-13022
RG-13022 is an inhibitor of the EGF and PDGF receptor tyrosine kinases
136831-48-6 sc-200591
sc-200591A
5 mg
10 mg
$95.00
$175.00
1
(0)
Lavendustin B
Lavendustin B is a tyrosine kinase inhibitor
125697-91-8 sc-200595
sc-200595A
1 mg
5 mg
$64.00
$249.00
1
(0)
Tyrphostin RG 14620
Tyrphostin RG 14620 is a non-phenolic tyrphostin analog selective for the EGF receptor
136831-49-7 sc-200593
sc-200593A
5 mg
10 mg
$64.00
$130.00
0
(0)
DAPH
DAPH is an inhibitor of EGFR kinase 3
145915-58-8 sc-200698
5 mg
$130.00
0
(0)
AG 825
AG 825 is a selective ErbB2 (Neu) inhibitor and apoptosis inducer
149092-50-2 sc-202045
sc-202045A
sc-202045B
sc-202045C
2 mg
5 mg
10 mg
100 mg
$45.00
$90.00
$175.00
$1,700.00
0
(1)
PD 158780 solution
PD 158780 solution is a potent tyrosine kinase inhibitor
171179-06-9 sc-202758
500 µg
$159.00
0
(0)
BPIQ-II HCl Salt
BPIQ-II HCl Salt is a specific and potent EGFR tyrosine kinase activity inhibitor
171179-32-1 (free base) sc-221375
1 mg
$203.00
0
(0)
EGFR/ErbB-2 抑制剤
EGFR/ErbB-2 Inhibitor is a potent reversible inhibitor of EGFR and c-erbB2
179248-61-4 sc-203935
1 mg
$99.00
0
(0)
Didesmethyl Erlotinib Hydrochloride Salt
Didesmethyl Erlotinib Hydrochloride Salt is a metabolite of Erlotinib
183320-12-9 sc-207566
1 mg
$350.00
0
(0)
Desmethyl Erlotinib Acetate
Desmethyl Erlotinib Acetate is a derivative of Ertolinib, a potent EGFR inhibitor
183320-15-2 sc-218150
1 mg
$350.00
0
(0)
PD 153035 Hydrochloride
PD 153035 Hydrochloride is a potent inhibitor of epidermal growth factor (EGF) receptor tyrosine kinase
183322-45-4 sc-205963
sc-205963A
10 mg
50 mg
$125.00
$525.00
0
(1)
3-(4-Isopropylbenzylidenyl)shyindolin-2-one
3-(4-Isopropylbenzylidenyl)indolin-2-one is a non-selective inhibitor of RTKs
186611-55-2 sc-202413
sc-202413A
1 mg
5 mg
$39.00
$206.00
0
(0)
BIBX 1382
BIBX 1382 is a potent, reversible, selective inhibitor of EGFR
196612-93-8 sc-202497
5 mg
$180.00
0
(0)
GW2974
GW2974 is a selective dual EGFR and Neu (ErbB-2) inhibitor
202272-68-2 sc-252869
25 mg
$240.00
0
(0)
PD 166285
PD 166285 is an inhibitor of RTK, c-Src, FGFR1, Wee 1, and PDGFRβ
212391-63-4 sc-208153
5 mg
$100.00
1
(1)
Pelitinib
Pelitinib is an EGFR inhibitor
257933-82-7 sc-208155
5 mg
$350.00
0
(0)
Canertinib
Canertinib is an irreversible pan-erbB tyrosine kinase inhibitor
267243-28-7 sc-207397
10 mg
$220.00
1
(0)
ZM 323881 hydrochloride
ZM 323881 hydrochloride is a receptor tyrosine kinase inhibitor of VEGFR-2 (Flk-1), PDGFR-beta, EGFR, and FGFR1
324077-30-7 sc-296861
sc-296861A
1 mg
10 mg
$105.00
$164.00
1
(0)
Vandetanib
Vandetanib is an antagonist of VEGFR (Flk and Flk) and EGFR families.
443913-73-3 sc-220364
sc-220364A
5 mg
50 mg
$167.00
$1,353.00
0
(1)
EGFR Inhibitor III
EGFR Inhibitor III is which inhibits EGFR- kinase activity, blocking phosphorylation
733009-42-2 sc-221580
5 mg
$379.00
0
(0)
EGFR 抑制剤
EGFR Inhibitor is a highly selective, cell-permeable EGFR inhibitor
879127-07-8 sc-203934
1 mg
$99.00
0
(1)
JNJ 28871063 hydrochloride
A potent inhibitor of ErbB receptors
944341-54-2 sc-204025
sc-204025A
10 mg
50 mg
$209.00
$880.00
1
(0)
EGF/FGF/PDGF receptor tyrosine kinase 抑制剤
EGF/FGF/PDGF receptor tyrosine kinase inhibitor is a tyrosine kinase inhibitor that inhibits human FGFR-1, PDGFR-β, c-Scr, & EGFR
1135256-66-4 sc-221579
2 mg
$290.00
1
(1)
AST 1306
AST 1306 is a potent and selective inhibitor of EGFR phosphorylation
1050500-29-2 sc-364413
sc-364413A
5 mg
10 mg
$420.00
$600.00
0
(0)
2prime-Thioadenosine
2′-Thioadenosine is a potent, selective inhibitor of ErbB1/ErbB2
60239-18-1 (non-salt) sc-220826
2 mg
$270.00
0
(0)
Gefitinib hydrochloride salt
Gefitinib hydrochloride salt is a potent inhibitor of EGFR tyrosine kinase activity
184475-55-6 sc-337854
1 g
$300.00
1
(0)
ARRY334543
ARRY334543 is a potent and selective EGFR phosphorylation inhibitor
845272-21-1 sc-364410
sc-364410A
5 mg
10 mg
$487.00
$667.00
0
(0)
Src/EGFR 抑制剤
Src/EGFR Inhibitor is a synthetic inhibitor for Src and EGFR
131023-24-0 sc-3050
0.5 mg
$90.00
0
(0)
Gefitinib O-Methyl-D3
Gefitinib O-Methyl-D3 is an derivative of Gefitinib, an EGFR inhibitor
sc-218566
1 mg
$300.00
0
(0)
OSI-420-d4, Free Base (Desmethyl Erlotinib-d4)
OSI-420-d4, Free Base (Desmethyl Erlotinib-d4) is a labeled metabolite of Erlotinib, an EGFR inhibitor
sc-219500
1 mg
$600.00
0
(0)
LFM-A12
LFM-A12 is a potent and specific inhibitor of EGFR tyrosine kinase activity
sc-295360
sc-295360A
500 µg
1 mg
$296.00
$400.00
0
(0)
BPDQ
BPDQ is a potent, reversible, and specific inhibitor of EGFR tyrosine kinase
169205-87-2 sc-311299
1 mg
$160.00
0
(0)
Tyrphostin AG 528
Tyrphostin AG 528 is an inhibitor of EGFR tyrosine kinase activity
133550-49-9 sc-216034
5 mg
$42.00
0
(0)
BPIQ-I
BPIQ-I is a potent and specific inhibitor of tyrosine kinase activity of EGFR
174709-30-9 sc-202507
1 mg
$150.00
0
(0)
Gefitinib 2hydrochloride salt
Gefitinib 2hydrochloride salt is a potent and selective inhibitor of EGFR kinase
184475-56-7 sc-337853
1 g
$1,950.00
0
(0)
Canertinib Dihydrochloride
Canertinib Dihydrochloride is a water-soluble, EGFR, HER2, and ErbB-4 tyrosine kinase inhibitor
289499-45-2 sc-396066
25 mg
$113.00
0
(0)
GW 583340 dihydrochloride
GW 583340 dihydrochloride is a potent inhibitor of EGFR/Neu (EGFR/ErbB2)
388082-81-3 sc-224012
sc-224012A
1 mg
5 mg
$215.00
$850.00
0
(0)
BIBU 1361 dihydrochloride
BIBU 1361 dihydrochloride is a selective EGFR kinase inhibitor
793726-84-8 sc-203844
sc-203844A
1 mg
10 mg
$95.00
$209.00
0
(0)
TAK 285
TAK 285 is a potent and selective EGFR and HER2 inhibitor
871026-44-7 sc-364627
sc-364627A
5 mg
10 mg
$405.00
$700.00
0
(0)
3-(4-Hydroxybenzylidenyl)shyindolin-2-one
3-(4-Hydroxybenzylidenyl)indolin-2-one is a selective receptor tyrosine kinase (RTK) inhibitor shown to inhibit FLK-1 RTK
293302-14-4 sc-202412
sc-202412A
1 mg
5 mg
$55.00
$216.00
0
(0)
WZ 3146
WZ 3146 is a mutant EGFR phosphorylation inhibitor
1214265-56-1 sc-364654
sc-364654A
5 mg
10 mg
$305.00
$480.00
0
(0)
WZ8040
WZ8040 is a potent inhibitor of EGFR T790M
1214265-57-2 sc-364656
sc-364656A
5 mg
10 mg
$255.00
$480.00
0
(0)
O-Desmethyl Gefitinib
O-Desmethyl Gefitinib is a major metabolite of Gefitinib
847949-49-9 sc-212448
1 mg
$220.00
0
(0)
O-Desmorpholinopropyl Gefitinib
A metabolite of gefitinib, an EGFR inhibitor
184475-71-6 sc-212456
1 g
$300.00
0
(0)
TAK 165
TAK 165 is a selective, potent, and irreversible ErbB2 and EGFR inhibitor
366017-09-6 sc-361372
sc-361372A
10 mg
50 mg
$139.00
$781.00
0
(0)
CGP 74514A
CGP 74514A is An inhibitor of CDK1/cyclin B, PKCα, PKA, and EGFR
sc-391004
sc-391004B
5 mg
25 mg
$80.00
$279.00
0
(0)
Erlotinib, Free Base
Erlotinib, Free Base is a tyrosine kinase inhibitor
183321-74-6 sc-396113
sc-396113A
sc-396113B
sc-396113C
500 mg
1 g
5 g
10 g
$74.00
$120.00
$272.00
$475.00
35
(0)
O-tert-Butyl-dimethylsilyl Curcumin
O-tert-Butyl-dimethylsilyl Curcumin is a protected Curcumin
911292-36-9 sc-396137
100 mg
$210.00
0
(0)
Tyrphostin AG 30
Tyrphostin AG 30 is a potent PTK inhibitor
122520-79-0 sc-202042
sc-202042A
5 mg
10 mg
$33.00
$80.00
0
(0)
PD 158780
PD 158780 is a potent tyrosine kinase inhibitor that can permeate cells
171179-06-9 sc-358789
10 mg
$127.00
0
(0)
AST-1306
897383-62-9 sc-503138
5 mg
$450.00
0
(0)

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