GPR Activators

G protein-coupled receptors (GPRs), also known as seven transmembrane receptors, heptahelical receptors or 7TM receptors, comprise a superfamily of proteins that play a role in many different stimulus-response pathways. Biochemicals that activate GPR have many applications in biochemical and physiological research. Click on the product name to view detailed information such as the chemical structure and specific chemical properties for each of our GPR Activators biochemicals. In stock GPR Activators are available for immediate shipping.

PRODUCT NAME/ApplicationCASCatalog #QUANTITYPriceCitationsRATING
Lipoxin A4
A trihydroxy fatty acid produced through 15-HETE metabolism
89663-86-5sc-201060
sc-201060A
sc-201060B
sc-201060C
25 µg
50 µg
100 µg
250 µg
$330.00
$471.00
$900.00
$1,980.00
0
(1)
Kynurenic acid
An antagonist of NMDA and AMPA/kainate receptors
492-27-3sc-202683
sc-202683A
sc-202683B
250 mg
1 g
5 g
$20.00
$50.00
$127.00
2
(1)
O-1602
A cannabidiol analog and activator of the GRP55 receptor
317321-41-8sc-202745
sc-202745A
1 mg
5 mg
$200.00
$400.00
0
(0)
Rosmarinic Acid
An activator of GPR35
20283-92-5sc-202796
sc-202796A
10 mg
50 mg
$31.00
$88.00
2
(1)
GW 9508
An aminophenylpropanoate agonist at the GRP40/FFA1 receptor
885101-89-3sc-203069
10 mg
$125.00
0
(0)
Tamoxifen Citrate
An antiestrogen with potent anti-cancer and PKC inhibitory activities
54965-24-1sc-203288
100 mg
$79.00
10
(1)
ABN-CBD
An agonist of the novel cannabinoid receptor GPR55
22972-55-0sc-203488A
sc-203488B
sc-203488
sc-203488C
1 mg
5 mg
10 mg
25 mg
$30.00
$135.00
$225.00
$525.00
0
(0)
MRS 2690
A potent agonist of the GPR105 receptor
15039-58-4sc-204104
1 mg
$398.00
0
(0)
PSN 375963 hydrochloride
An agonist of the GPR119 receptor
388575-52-8sc-204219
sc-204219A
10 mg
50 mg
$175.00
$739.00
0
(0)
TUG-424
An agonist of GPR40/FFA1
1082058-99-8sc-222379
sc-222379A
5 mg
25 mg
$234.00
$693.00
0
(0)
Kynurenic acid sodium salt
An antagonist of NDMA receptors
492-27-3 (non-salt)sc-358835
100 mg
$99.00
0
(1)
AS 1269574
A GPR119 receptor agonist
330981-72-1sc-361109
sc-361109A
10 mg
50 mg
$155.00
$620.00
0
(0)
Pamoic acid disodium salt
An agonist that induces GPR35 internalization and activates ERK1/2
6640-22-8sc-362777
25 g
$63.00
0
(0)
PF9 tetrasodium salt
A potent GPR17 agonist
851265-78-6sc-362783
1 mg
$235.00
0
(0)
TC-O 9311
A potent agonist of GPR139
444932-31-4sc-362802
sc-362802A
10 mg
50 mg
$116.00
$620.00
0
(0)
Compound 10
An activator of GPR35
123021-85-2sc-364688
sc-364688A
5 mg
25 mg
$84.00
$358.00
0
(0)

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