CYP3A4 Substrates

Cytochrome P450 (CYP) proteins are heme-thiolate monooxygenases that mediate NADPH-dependent electron transport and function to oxidize a variety of structurally unrelated compounds, including steroids, fatty acids and xenobiotics. Biochemicals that act as substrates for CYP3A4 have many applications in biochemical and physiological research. Click on the product name to view detailed information such as the chemical structure and specific chemical properties for each of our CYP3A4 Substrates biochemicals. In stock CYP3A4 Substrates are available for immediate shipping.

PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Vinblastine Sulfate
Vinblastine Sulfate is an anti-mitotic agent which arrests the cell cycle in the G2/M-phase
143-67-9 sc-201447
sc-201447A
10 mg
50 mg
$99.00
$390.00
9
(1)
Verapamil hydrochloride
Verapamil hydrochloride is a calcium channel protein inhibitor in cardiac muscle cells
152-11-4 sc-3590
sc-3590A
sc-3590B
100 mg
1 g
5 g
$25.00
$31.00
$90.00
21
(1)
Vincristine Sulfate
Vincristine Sulfate is a cell cycle arresting, apoptotic inducing alkaloid
2068-78-2 sc-201434
sc-201434A
5 mg
25 mg
$108.00
$319.00
12
(2)
Clarithromycin
Clarithromycin is a macrolide antibiotic and protein synthesis inhibitor
81103-11-9 sc-205634
sc-205634A
100 mg
250 mg
$69.00
$113.00
1
(1)
Clarithromycin-N-methyl-d3
Clarithromycin-N-methyl-d3 (contains 2% d0) is a deuterium-labeled clarithromycin derivative and a CYP4A inhibitor and substrate
sc-217926
5 mg
$280.00
0
(0)
(R)-(+)-Warfarin
(R)-(+)-Warfarin is a CYP1A2/3A4 substrate
5543-58-8 sc-255498
5 mg
$592.00
0
(0)