AR Inhibitors
Santa Cruz Biotechnology now offers a broad range of AR Inhibitors. There are five general types of adrenergic receptors (ARs), designated α1, α2, β1, β2 and β3, which are found in different target tissues and differ in their affinities and responses to various agonists and antagonists. AR Inhibitors offered by Santa Cruz inhibit AR and, in some cases, other G protein-coupled receptor kinases (GRKs) and PKC-directed phosphorylation related proteins. View detailed AR Inhibitor specifications, including AR Inhibitor CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.
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SEE ALSO...
- AR Antibodies for 10 µg trial size samples
- ChemCruz™ Chemical AR Activators for functional analysis of cellular responses to AR
| PRODUCT NAME/Application | CAS | Catalog # | QUANTITY | Price | Citations | RATING | |
|---|---|---|---|---|---|---|---|
Rauwolscine dot HClRauwolscine • HCl is a standard α-2-adrenergic (AR) antagonist |
6211-32-1 |
sc-200151 |
100 mg |
$98.00
|
0 |
| |
ICI 89406ICI 89406 is a β-adrenergic antagonist |
53671-71-9 |
sc-361212 sc-361212A |
10 mg 50 mg |
$89.00
$510.00 |
0 |
| |
Propranolol hydrochloridePropranolol hydrochloride is a β1 and β2 adrenergic receptor blocker |
3506-09-0 |
sc-3580 sc-3580B |
1 g 5 g |
$32.00
$117.00 |
8 |
| |
Verapamil hydrochlorideVerapamil hydrochloride is a calcium channel protein inhibitor in cardiac muscle cells |
152-11-4 |
sc-3590 sc-3590A sc-3590B |
100 mg 1 g 5 g |
$25.00
$31.00 $90.00 |
19 |
| |
Oxprenolol hydrochlorideOxprenolol hydrochloride is a non-selective β-adrenergic antagonist that also displays intrinsic sympathomimetic activity |
6452-73-9 |
sc-204152 sc-204152B sc-204152C sc-204152D |
100 mg 2.5 g 10 g 50 g |
$30.00
$1,900.00 $6,500.00 $13,000.00 |
2 |
| |
Alfuzosin hydrochlorideAlfuzosin hydrochloride is an α 1 adrenoceptor antagonist |
81403-68-1 |
sc-203812 sc-203812A |
10 mg 50 mg |
$79.00
$295.00 |
0 |
| |
BRL-37344BRL-37344 is a potent and selective β3-AR agonist |
127299-93-8 |
sc-200154 |
5 mg |
$105.00
|
3 |
| |
S(-)-Propranolol hydrochlorideS(−)-Propranolol hydrochloride is a β-adrenergic receptor antagonist |
4199-10-4 |
sc-200153 |
100 mg |
$84.00
|
1 |
| |
2-PMDQ2-PMDQ is a potent and selective antagonist of the α1-AR adrenoceptor |
139047-55-5 |
sc-203771 sc-203771A |
10 mg 50 mg |
$135.00
$560.00 |
0 |
| |
Doxazosin MesylateDoxazosin Mesylate is an alpha-1-adrenoreceptor antagonist |
77883-43-3 |
sc-205656 sc-205656A |
50 mg 250 mg |
$101.00
$390.00 |
2 |
| |
SpironolactoneSpironolactone is a lactone for proteomic research |
52-01-7 |
sc-204294 |
50 mg |
$100.00
|
1 |
| |
Phentolamine mesylatePhentolamine mesylate is an α-adrenergic blocker |
65-28-1 |
sc-205803 sc-205803A |
50 mg 100 mg |
$62.00
$125.00 |
1 |
| |
AaptamineAaptamine is a spongean alkaloid that can activate the p21 promoter in the absence of p53 |
85547-22-4 |
sc-202899 sc-202899A |
1 mg 10 mg |
$200.00
$750.00 |
0 |
| |
Phentolamine hydrochloridePhentolamine hydrochloride is an a-Adrenergic blocker |
73-05-2 |
sc-205802 sc-205802A sc-205802B sc-205802C sc-205802D sc-205802E sc-205802F |
50 mg 100 mg 250 mg 500 mg 1 g 2 g 2.5 g |
$75.00
$100.00 $220.00 $390.00 $750.00 $1,400.00 $1,700.00 |
1 |
| |
CarnosolCarnosol is a phytopolyphenol found in Rosemary that functions as an antioxidant, antimicrobial, & anticarcinogen |
5957-80-2 |
sc-204672 sc-204672A sc-204672B sc-204672C |
1 mg 5 mg 10 mg 50 mg |
$79.00
$179.00 $578.00 $2,540.00 |
0 |
| |
GaleteroneGaleterone is an antagonist to LNCaP AR |
851983-85-2 |
sc-364495 sc-364495A |
5 mg 25 mg |
$183.00
$550.00 |
1 |
| |
RX 821002 hydrochlorideRX 821002 hydrochloride is a selective α2-adrenoceptor antagonist |
109544-45-8 |
sc-203686 sc-203686A |
10 mg 50 mg |
$69.00
$259.00 |
0 |
| |
PhenoxybenzaminePhenoxybenzamine is a non-specific irreversible adrenergic (AR) antagonist |
63-92-3 |
sc-3581 sc-3581A |
200 mg 1 g |
$23.00
$74.00 |
3 |
| |
IsotetrandrineIsotetrandrine is a biscoclaurine alkaloid inhibitor of G protein activation of PLA2 |
477-57-6 |
sc-200869 sc-200869A |
1 mg 5 mg |
$69.00
$251.00 |
0 |
| |
Sotalol hydrochlorideSotalol hydrochloride is a potent β adrenergic antagonist |
959-24-0 |
sc-203699 sc-203699A |
10 mg 50 mg |
$60.00
$235.00 |
1 |
| |
1,3-Dimethyl-8-phenylxanthineCAS: 961-45-5, MF: C13H12N4O2, MW: 256.26, Purity: ≥98% |
961-45-5 |
sc-253981 |
100 mg |
$110.00
|
0 |
| |
Doxepin hydrochlorideDoxepin hydrochloride is a highly potent histamine H1 antagonist with affinity to H4 receptor |
1229-29-4 |
sc-203930 |
1 g |
$32.00
|
0 |
| |
(R)-(+)-Propranolol hydrochloride(R)-(+)-Propranolol hydrochloride is a less active anantiomer the non-selective beta blocker propranolol |
5051-22-9 |
sc-203678 sc-203678A |
100 mg 1 g |
$69.00
$325.00 |
0 |
| |
Fenspiride HydrochlorideFenspiride Hydrochloride is an α adrenergic and H1 histamine receptor antaonist |
5053-08-7 |
sc-207684 |
10 mg |
$145.00
|
0 |
| |
Clomipramine hydrochlorideClomipramine hydrochloride is a selective ST, SLC6A2, and DAT inhibitor |
17321-77-6 |
sc-203898 |
1 g |
$36.00
|
2 |
| |
ent-Levobunolol, Hydrochlorideent-Levobunolol, Hydrochloride is an enantiomer of levobunolol |
27867-05-6 |
sc-211411 |
100 mg |
$220.00
|
0 |
| |
Propafenone HydrochloridePropafenone Hydrochloride is a sodium channel protein inhibitor |
34183-22-7 |
sc-204863 sc-204863A sc-204863B sc-204863C |
1 g 5 g 25 g 100 g |
$21.00
$64.00 $190.00 $481.00 |
0 |
| |
Acebutolol HydrochlorideAcebutolol Hydrochloride is a β-AR antagonist |
34381-68-5 |
sc-217555 |
10 g |
$220.00
|
0 |
| |
Levobunolol, HydrochlorideLevobunolol, Hydrochloride is a β-adrenoceptor antagonist |
27912-14-7 |
sc-211734 sc-211734A |
100 mg 250 mg |
$700.00
$600.00 |
0 |
| |
2-Hydroxy-flutamide2-Hydroxy-flutamide is an inhibitor of proliferation of estradiol-induced growth of MCF-7 breast cancer cells |
52806-53-8 |
sc-205574 sc-205574A |
10 mg 25 mg |
$140.00
$368.00 |
0 |
| |
Urapidil HClUrapidil HCl is an adrenergic α1-AR antagonist and a serotonin 5-HT1A (SR-1A) receptor agonist |
64887-14-5 |
sc-200155 |
100 mg |
$120.00
|
0 |
| |
Maprotiline HydrochlorideMaprotiline Hydrochloride is A norepinephrine reuptake inhibitor shown to block apoptosis of spiny neurons |
10347-81-6 |
sc-200156 |
1 g |
$72.00
|
5 |
| |
Fenoldopam hydrochlorideFenoldopam hydrochloride is a selective D1-like dopamine receptor partial agonist |
67227-56-9 |
sc-279160 |
10 mg |
$159.00
|
0 |
| |
MirtazapineMirtazapine is a potent SR-2, SR-3, and Histamine H1 receptor antagonist |
85650-52-8 |
sc-204088 sc-204088A |
10 mg 50 mg |
$105.00
$409.00 |
0 |
| |
CarazololCarazolol is A high affinity β-adrenergic receptor antagonist |
57775-29-8 |
sc-257215 sc-257215A |
10 mg 200 mg |
$50.00
$250.00 |
0 |
| |
Dimebolin dihydrochlorideDimebolin dihydrochloride is a histamine, AR, and Ca channel inhibitor |
97657-92-6 |
sc-294348 sc-294348A sc-294348B |
1 mg 5 mg 50 mg |
$37.00
$96.00 $384.00 |
0 |
| |
Cyanopindolol hemifumarateCyanopindolol hemifumarate is a SR-1A/SR-1B antagonist |
106469-57-2 |
sc-203906 sc-203906A |
10 mg 25 mg |
$159.00
$693.00 |
0 |
| |
Niguldipine hydrochlorideNiguldipine hydrochloride is a selective α 1-adrenoceptor antagonist and dihydropyridine calcium channel blocker |
113317-61-6 |
sc-201471 sc-201471A |
10 mg 50 mg |
$77.00
$312.00 |
0 |
| |
Naftopidil hydrochlorideNaftopidil hydrochloride is an α1-AR adrenoceptor antagonist |
57149-07-2 (free base) |
sc-203151 sc-203151A |
10 mg 50 mg |
$55.00
$175.00 |
0 |
| |
S-(+)-Niguldipine hydrochlorideS-(+)-Niguldipine hydrochloride is a calcium channel protein inhibitor |
113165-32-5 |
sc-203248 |
10 mg |
$124.00
|
0 |
| |
(S)-Timolol Maleate(S)-Timolol Maleate is a selective β1-AR receptor antagonist |
26921-17-5 |
sc-203297 sc-203297A |
100 mg 250 mg |
$59.00
$122.00 |
0 |
| |
ARC 239 dihydrochlorideARC 239 dihydrochloride is a selective α2B-AR adrenoreceptor antagonist |
67339-62-2 |
sc-203518 |
5 mg |
$125.00
|
1 |
| |
Betaxolol hydrochlorideBetaxolol hydrochloride is a selective β1-AR adrenoceptor antagonist |
63659-19-8 |
sc-203527 sc-203527A |
10 mg 50 mg |
$125.00
$480.00 |
0 |
| |
2-MPMDQ2-MPMDQ is a selective α1-AR adrenoceptor antagonist |
149847-77-8 |
sc-203770 sc-203770A |
10 mg 50 mg |
$129.00
$548.00 |
0 |
| |
(±)-Bisoprolol hemifumarate(±)-Bisoprolol hemifumarate is a selective β1-AR antagonist |
104344-23-2 |
sc-203531 sc-203531B sc-203531A |
10 mg 25 mg 50 mg |
$115.00
$190.00 $462.00 |
0 |
| |
Efaroxan hydrochlorideEfaroxan hydrochloride is a potent α2-AR adrenoceptor antagonist |
89197-00-2 |
sc-203573 sc-203573A |
10 mg 50 mg |
$125.00
$525.00 |
0 |
| |
(R)-Phenoxybenzamine Hydrochloride(R)-Phenoxybenzamine Hydrochloride is an irreversible α-adrenergic antagonist |
16053-59-1 |
sc-391970 |
5 mg |
$280.00
|
0 |
| |
HEAT hydrochlorideHEAT hydrochloride is a very selective α1-AR adrenoceptor antagonist |
30007-39-7 |
sc-203996 sc-203996A |
10 mg 50 mg |
$115.00
$440.00 |
0 |
| |
UrapidilUrapidil is an a1-adrenergic antagonist with high affinity for 5-hydroxytryptamine sites. |
34661-75-1 |
sc-391143 sc-391143A |
500 mg 5 g |
$120.00
$762.00 |
0 |
| |
SDZ 21009SDZ 21009 is a β-AR, SR-1A, and SR-1B antagonist |
39731-05-0 |
sc-203695 sc-203695A |
10 mg 50 mg |
$200.00
$825.00 |
0 |
| |
BMY 7378 dihydrochlorideBMY 7378 dihydrochloride is a SR-1A agonist and a selective α1D-AR antagonist |
21102-95-4 |
sc-203849 sc-203849A |
10 mg 50 mg |
$44.00
$205.00 |
0 |
| |
BucindololBucindolol is a non-selective β-AR adrenoceptor antagonist with additional α1-adrenoceptor blocking activity. |
71119-11-4 |
sc-203860 sc-203860A |
10 mg 50 mg |
$235.00
$750.00 |
1 |
| |
CGP 12177 hydrochlorideCGP 12177 hydrochloride is a β1/β2-AR adrenoreceptor agonist |
81047-99-6 |
sc-203878 sc-203878A |
10 mg 50 mg |
$75.00
$172.00 |
0 |
| |
CGP 20712 DihydrochlorideCGP 20712 Dihydrochloride is a highly potent and selective β1-AR antagonist |
1216905-73-5 |
sc-203879 sc-203879A |
10 mg 50 mg |
$210.00
$865.00 |
0 |
| |
Idazoxan hydrochlorideIdazoxan hydrochloride is an α2-AR adrenoceptor antagonist and I2 imidazoline receptor agonist. |
79944-56-2 |
sc-204006 sc-204006A |
10 mg 50 mg |
$125.00
$495.00 |
2 |
| |
N-(4-Amino-6,7-dimethoxyquinazol-2-yl)-N-methyl-2-cyanoethylamine |
76362-28-2 |
sc-211970 |
100 mg |
$280.00
|
0 |
| |
JP 1302 dihydrochlorideJP 1302 dihydrochloride is a selective α2C-AR |
80259-18-3 |
sc-204026 sc-204026A |
10 mg 50 mg |
$185.00
$772.00 |
0 |
| |
Nebivolol hydrochlorideNebivolol hydrochloride is a highly selective β1-adrenoceptor antagonist |
152520-56-4 |
sc-204122 sc-204122A |
10 mg 50 mg |
$139.00
$224.00 |
0 |
| |
2-phenyl-amino-N6-endo-norbornyladenine2-phenyl-amino-N6-endo-norbornyladenine is an A3 AR antagonist |
863202-33-9 |
sc-205088 sc-205088A |
500 µg 1 mg |
$208.00
$368.00 |
1 |
| |
rac Nebivolol Hydrochloriderac Nebivolol Hydrochloride is a racimic mixture of β1-Adrenergic blocker (β1-AR) used as an antihypertensive |
169293-50-9 |
sc-391275 |
10 mg |
$220.00
|
0 |
| |
1,1-Dichloro-2,2-bis(4-chlorophenyl)ethene1,1-Dichloro-2,2-bis(4-chlorophenyl)ethene is a potent androgen receptor antagonist |
72-55-9 |
sc-251534 |
1 g |
$55.00
|
0 |
| |
(S)-(-)-Verapamil Hydrochloride(S)-(−)-Verapamil Hydrochloride is an isomer that inhibits the p-glycoprotein efflux pump in MDR tumor cell lines |
36622-29-4 |
sc-208338 |
1 mg |
$350.00
|
0 |
| |
AsenapineAsenapine is a combined 5HT2, adrenergic, and D2 receptor antagonist |
65576-45-6 |
sc-210839 |
10 mg |
$280.00
|
0 |
| |
rac Propranolol-d7rac Propranolol-d7 is an anti-hypertensive, anti-anginal and anti-arrhythmic β-AR (β-Adrenergic receptor) blocker |
98897-23-5 |
sc-212742 |
5 mg |
$225.00
|
1 |
| |
8-Benzyloxy-5-((R)-2-bromo-1-hydroxyethyl)-1H-quinolinone8-Benzyloxy-5-((R)-2-bromo-1-hydroxyethyl)-1H-quinolinone is a chemical used in the preparation of phenylethanolamine derivatives |
530084-79-8 |
sc-396009 |
2.5 mg |
$280.00
|
0 |
| |
Spironolactone-d6 (Major)Spironolactone-d7 (Major) is a renal competitive MCR (aldosterone receptor) antagonist |
52-01-7 unlabeled |
sc-220132 sc-220132A |
1 mg 10 mg |
$250.00
$2,000.00 |
0 |
| |
BenzoestrolBenzoestrol is a nonsteroidal estrogen antagonist |
85-95-0 |
sc-210870 |
5 mg |
$300.00
|
0 |
| |
(R,R)-Labetalol Hydrochloride(R,R)-Labetalol Hydrochloride is A competitive antagonist at both α-and β-adrenergic receptor sites |
75659-08-4 |
sc-212635 |
1 mg |
$350.00
|
0 |
| |
Tolazoline HydrochlorideTolazoline Hydrochloride is a peripheral vasodilator |
59-97-2 |
sc-213056 sc-213056A sc-213056B |
10 g 25 g 100 g |
$45.00
$90.00 $180.00 |
0 |
| |
Chlorprothixene HydrochlorideChlorprothixene Hydrochloride is a D2DR inhibitor |
6469-93-8 |
sc-211077 |
1 g |
$30.00
|
0 |
| |
BRL 44408 MALEATEBRL 44408 MALEATE is a selective α2A-AR antagonist |
118343-19-4 |
sc-217791 |
10 mg |
$143.00
|
0 |
| |
AzaperoneAzaperone is an α-adrenergic, dopamine and histamine receptor inhibitor |
1649-18-9 |
sc-210851 |
100 mg |
$284.00
|
0 |
| |
Mirtazapine-d3Mirtazapine-d3 is an α2-Adrenergic blocker |
1216678-68-0 |
sc-218855 |
1 mg |
$300.00
|
0 |
| |
Sotalol-d6 HydrochlorideSotalol-d6 Hydrochloride is A deuterium labeled β-adronergic blocker |
1246820-85-8 |
sc-220127 |
1 mg |
$280.00
|
1 |
| |
Trimipramine-d3 Maleate SaltTrimipramine-d3 Maleate Salt is a serotonin transport blocker that also blocks norepinephrine uptake |
521-78-8 (unlabeled) |
sc-220342 |
1 mg |
$200.00
|
0 |
| |
Imiloxan HydrochlorideImiloxan Hydrochloride is a highly selective α2B-AR antagonist |
81167-22-8 |
sc-224023 sc-224023A |
5 mg 25 mg |
$211.00
$849.00 |
0 |
| |
Labetalol hydrochlorideLabetalol hydrochloride is a competitive α-AR (α-adrenoceptor) and β-AR (β-adrenoceptor) antagonist with antihypertensive propertie |
32780-64-6 |
sc-252942 |
5 g |
$77.00
|
0 |
|