FXR Activators

NR (nuclear receptor) proteins comprise a large family of nuclear hormone receptor transcription factors that are characterized by discrete domains which function in DNA and ligand binding. Biochemicals that activate FXR have many applications in biochemical and physiological research. Click on the product name to view detailed information such as the chemical structure and specific chemical properties for each of our FXR Activators biochemicals. In stock FXR Activators are available for immediate shipping.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
GW 9662
GW 9662 is a selective, irreversible, and effective PPARγ antagonist that also acts as a FXR and PXR agonist
22978-25-2 sc-202641
5 mg
Fexaramine is a potent, selective FXR activator
574013-66-4 sc-203580
10 mg
50 mg
SR 12813
SR 12813 is a PXR agonist that activates the farnesoid X receptor (FXR) at μM concentrations
126411-39-0 sc-204296
10 mg
50 mg
GW 4064
GW 4064 is a novel nonsteroidal FXR nuclear receptor activator
278779-30-9 sc-218577
5 mg