AR Activators

Santa Cruz Biotechnology now offers a broad range of AR Activators. There are five general types of adrenergic receptors (ARs), designated α1, α2, β1, β2 and β3, which are found in different target tissues and differ in their affinities and responses to various agonists and antagonists. AR Activators offered by Santa Cruz activate AR and, in some cases, other G protein-coupled receptor kinases (GRKs) and PKC-directed phosphorylation related proteins. View detailed AR Activator specifications, including AR Activator CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Zilpaterol
Zilpaterol is a growth promotant and b-andrenergic agonist
119520-05-7 sc-220402
sc-220402A
sc-220402A-CW
sc-220402B
5 mg
10 mg
10 mg
100 mg
$220.00
$533.00
$681.00
$5,300.00
0
(2)
Brimonidine Tartrate
Brimonidine Tartrate is an α-2 receptor agonist
70359-46-5 sc-217788
100 mg
$167.00
3
(1)
Dexmedetomidine hydrochloride
Dexmedetomidine hydrochloride is an active isomer of medetomide, a potent and highly selective α2-adrenoceptor agonist
145108-58-3 sc-205290
sc-205290A
10 mg
50 mg
$159.00
$490.00
0
(1)
(-)-Isoproterenol (+)-bitartrate salt
(−)-Isoproterenol (+)-bitartrate salt is a β-adrenoceptor agonist
54750-10-6 sc-252926
sc-252926A
sc-252926D
sc-252926B
sc-252926C
100 mg
500 mg
1 g
5 g
10 g
$95.00
$235.00
$397.00
$2,250.00
$4,300.00
0
(1)
Andarine
Andarine is an androgen receptor (AR) agonist with Ki of 4 nM
401900-40-1 sc-364405
sc-364405A
5 mg
50 mg
$255.00
$1,455.00
0
(0)
(+/-)-Epinephrine
(±)-Epinephrine is an adrenoceptor agonist
329-65-7 sc-252779
sc-252779A
5 g
25 g
$60.00
$140.00
1
(1)
Cimaterol
Cimaterol is an agonist of the β-AR adrenoreceptor
54239-37-1 sc-203549
sc-203549A
10 mg
50 mg
$115.00
$440.00
0
(1)
Rilmenidine hemifumarate
Rilmenidine hemifumarate is a selective ligand for I1-imidazoline and α2-AR agonist
207572-68-7 sc-203680
sc-203680A
5 mg
25 mg
$110.00
$550.00
0
(1)
UK 14,304
UK 14,304 is an α2-adrenergic receptor agonist
59803-98-4 sc-204373
sc-204373A
10 mg
50 mg
$110.00
$446.00
0
(0)
B-HT 920
B-HT 920 is a dopamine D2 receptor agonist, SR-3 antagonist and α2-adrenoceptor agonist
36085-73-1 sc-203523
sc-203523A
10 mg
50 mg
$89.00
$440.00
0
(0)
Cirazoline hydrochloride
Cirazoline hydrochloride is a selective α1 agonist
40600-13-3 sc-203550
10 mg
$129.00
0
(0)
Cimaterol-d7
Cimaterol-d7 is a labeled β-adrenergic agonist
1228182-44-2 sc-394133
10 mg
$600.00
0
(0)
(-)-Epinephrine-(+)-bitartrate
(−)-Epinephrine-(+)-bitartrate is an α,β-adrenergic receptor agonist
51-42-3 sc-204032
100 mg
$67.00
0
(1)
(+/-)-Synephrine
(±)-Synephrine is an α-adrenergic receptor agonist
94-07-5 sc-220182
25 g
$200.00
0
(0)
Naphazoline Hydrochloride
Naphazoline Hydrochloride is a producer ionotropic effects via α-adrenoceptor stimulation
550-99-2 sc-205764
sc-205764A
25 g
100 g
$49.00
$150.00
0
(0)
Xylazine
Xylazine is an α2 class of adrenergic receptor agonist
7361-61-7 sc-253838
1 g
$59.00
5
(0)
Z-Guggulsterone
Z-Guggulsterone is a selective antagonist of farnesoid X receptor and inhibitor of FXR transactivation.
39025-23-5 sc-204414
sc-204414A
10 mg
25 mg
$205.00
$360.00
16
(1)
Tizanidine • HCl
Tizanidine • HCl is a centrally acting α2-adrenergic (α2-AR) agonist
64461-82-1 sc-200148
sc-200148A
100 mg
500 mg
$61.00
$247.00
0
(1)
Carvedilol
Carvedilol is an α1- and β-adrenergic receptor antagonist
72956-09-3 sc-200157
sc-200157A
sc-200157B
sc-200157C
sc-200157D
100 mg
1 g
10 g
25 g
100 g
$57.00
$80.00
$133.00
$265.00
$667.00
1
(1)
Isoproterenol Hydrochloride
Isoproterenol Hydrochloride is a selective β-adrenergic agonist
51-30-9 sc-202188
sc-202188A
100 mg
500 mg
$20.00
$30.00
2
(0)
Clonidine hydrochloride
Clonidine hydrochloride is an antihypertensive α2-adrenergic receptor agonist
4205-91-8 sc-203002
1 g
$360.00
11
(0)
Dobutamine Hydrochloride
Dobutamine Hydrochloride is a dopamine derived β1-AR agonist
49745-95-1 sc-203031
sc-203031A
10 mg
50 mg
$58.00
$183.00
1
(1)
Formoterol fumarate
Formoterol fumarate is a potent β2-AR agonist
43229-80-7 sc-203050
sc-203050A
10 mg
50 mg
$125.00
$525.00
3
(1)
Clonidine-d4 Hydrochloride
Clonidine-d4 Hydrochloride is an a2-adrenergic agonist
67151-02-4 sc-217935
1 mg
$280.00
0
(0)
L-(ndash)-Norepinephrine-(+)-bitartrate
L-(–)-Norepinephrine-(+)-bitartrate is a α,β-adrenoceptor (AR) agonist
69815-49-2 sc-203093
100 mg
$80.00
0
(1)
Octopamine Hydrochloride
Octopamine Hydrochloride is an activator of β3-AR and α2A-AR adrenoceptors
770-05-8 sc-203168
sc-203168A
1 g
5 g
$50.00
$85.00
0
(1)
Oxymetazoline Hydrochloride
Oxymetazoline Hydrochloride is is an α1-AR and α2-AR adrenergic receptor agonist.
2315-02-8 sc-203172B
sc-203172
sc-203172C
sc-203172A
1 g
5 g
10 g
25 g
$53.00
$120.00
$208.00
$480.00
1
(0)
Salbutamol hemisulfate
Salbutamol hemisulfate is a β2-AR adrenergic receptor agonist
51022-70-9 sc-203373
250 mg
$119.00
0
(0)
Guanabenz acetate
Guanabenz acetate is an α2A-AR agonist and IGRS selective ligand
23256-50-0 sc-203590
sc-203590A
sc-203590B
sc-203590C
sc-203590D
100 mg
500 mg
1 g
10 g
25 g
$98.00
$450.00
$800.00
$4,000.00
$7,000.00
2
(2)
(R)-(-)-Phenylephrine hydrochloride
(R)-(−)-Phenylephrine hydrochloride is an α1-adrenoceptor agonist
61-76-7 sc-203677
100 mg
$43.00
1
(1)
Moxonidine hydrochloride
Moxonidine hydrochloride is an Imidazoline receptor and an α2-adrenergic agonist
75438-57-2 sc-204096
sc-204096A
10 mg
50 mg
$121.00
$495.00
0
(0)
A 61603 HYDROBROMIDE
A 61603 HYDROBROMIDE is a potent α-adrenoceptor agonist
107756-30-9 sc-203789
sc-203789A
10 mg
50 mg
$139.00
$645.00
0
(0)
CL 316243 disodium salt
CL 316243 disodium salt is a highly selective, thermogenic β3-adrenoceptor agonist and anti-obesity agent.
151126-84-0 sc-203895
sc-203895A
10 mg
50 mg
$220.00
$825.00
10
(2)
Guanfacine hydrochloride
Guanfacine hydrochloride is a selective α2A-AR adrenoceptor agonist
29110-48-3 sc-203988
sc-203988A
10 mg
50 mg
$65.00
$225.00
0
(0)
L-755,507
L-755,507 is a very potent, selective β3-adrenergic receptor partial agonist and enhancer of CRISPR-mediated HDR efficiency.
159182-43-1 sc-204045
sc-204045A
10 mg
50 mg
$165.00
$700.00
2
(1)
Medetomidine hydrochloride
Medetomidine hydrochloride is a potent and highly selective α2-adrenoceptor agonist used as an anesthetic and analgesic.
86347-15-1 sc-204073
sc-204073A
10 mg
50 mg
$119.00
$475.00
2
(1)
Detomidine HCl
Detomidine HCl is an α2-adrenergic agonist
90038-01-0 sc-357329
sc-357329A
25 mg
100 mg
$192.00
$444.00
0
(0)
Synephrine Hydrochloride
Synephrine Hydrochloride is an α-adrenergic receptor agonist (α1A-AR)
5985-28-4 sc-394099
5 g
$150.00
0
(0)
UK 14,304 tartrate
UK 14,304 tartrate is an α2-adrenoceptor agonist
59803-99-5 sc-204374
sc-204374A
10 mg
50 mg
$139.00
$575.00
0
(0)
Ritodrine
Ritodrine is a β2-adrenoceptor agonist that acts as an adrenergic receptor stimulant
23239-51-2 sc-204882
sc-204882A
250 mg
1 g
$100.00
$335.00
1
(0)
Adrafinil
Adrafinil is an α-adrenergic agonist
63547-13-7 sc-207263
sc-207263A
10 mg
100 mg
$250.00
$600.00
0
(0)
p-Aminoclonidine
CAS: 73217-88-6, MF: C9H10Cl2N4•HCl, MW: 281.57
73217-88-6 sc-296001
sc-296001A
1 mg
5 mg
$136.00
$444.00
0
(0)
4-Amino-3-chloro-5-(trifluoromethyl)benzoic Acid
4-Amino-3-chloro-5-(trifluoromethyl)benzoic Acid is a mabuterol intermediate
95656-52-3 sc-394146
250 mg
$280.00
0
(0)
1-[4-Amino-3-chloro-5-(trifluoromethyl)phenyl]-2-bromo-ethanone
1-[4-Amino-3-chloro-5-(trifluoromethyl)phenyl]-2-bromo-ethanone is a mabuterol intermediate
97760-87-7 sc-394147
50 mg
$280.00
0
(0)
A 80426 mesylate
A 80426 mesylate is a high affinity alpha2-adrenoceptor antagonist
152148-63-5 sc-361095
sc-361095A
10 mg
50 mg
$145.00
$645.00
0
(0)
Cl-4AS-1
Cl-4AS-1 is an inhibitor of 5α-Reductase 1 and 5α-Reductase 2
188589-66-4 sc-361152
sc-361152A
10 mg
50 mg
$195.00
$825.00
0
(0)
Brimonidine-d4 D-Tartrate
Brimonidine-d4 D-Tartrate is a labelled Brimonidine and α 2 receptor agonist
1316758-27-6 sc-217789
1 mg
$250.00
0
(0)
Cimbuterol
Cimbuterol is an adrenergic agonist
54239-39-3 sc-391935
sc-391935A
sc-391935B
sc-391935C
10 mg
25 mg
100 mg
250 mg
$158.00
$350.00
$1,400.00
$2,800.00
0
(0)
Tetrahydrozoline-d4 Hydrochloride
Tetrahydrozoline-d4 Hydrochloride is an AR (αreceptor) agonist
sc-220222
1 mg
$250.00
0
(0)
Salmeterol
Salmeterol is a potent and selective β2-AR agonist
89365-50-4 sc-224277
sc-224277A
10 mg
50 mg
$186.00
$562.00
1
(1)
Dihydroergotamine (+)-tartrate salt
Dihydroergotamine (+)-tartrate salt is a vascular SR (serotonin receptor) activator
5989-77-5 sc-263091
100 mg
$165.00
0
(0)
(±)-Epinephrine hydrochloride
(±)-Epinephrine hydrochloride is an adrenergic receptor agonist
329-63-5 sc-252780
sc-252780A
5 g
25 g
$63.00
$267.00
0
(1)
Isoetharine mesylate salt
Isoetharine mesylate salt is a β-AR (β-adrenergic receptor) agonist
7279-75-6 sc-252918
1 g
$58.00
0
(0)

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