TGF beta RI Inhibitors

TGFβs mediate their activity by high affinity binding to the TGFβ receptor type-II (TGFβ RII) with a cytoplasmic serine-threonine kinase domain. Biochemicals that inhibit TGF beta RI have many applications in biochemical and physiological research. Click on the product name to view detailed information such as the chemical structure and specific chemical properties for each of our TGF beta RI Inhibitors. In stock TGF beta RI Inhibitors are available for immediate shipping.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
A 83-01
A 83-01 is an inhibitor of TGF-β type I receptor kinase (ALK5), activin type IB receptor (ALK4), and nodal type I receptor (ALK7).
909910-43-6 sc-203791
sc-203791A
10 mg
50 mg
$190.00
$772.00
13
(1)
SB 431542
SB 431542 is a Potent, selective inhibitor of TGF-βRI, specifically at ALK5 and its relatives ALK4 and ALK7.
301836-41-9 sc-204265
sc-204265A
sc-204265B
1 mg
10 mg
25 mg
$74.00
$205.00
$400.00
43
(1)
Casein Kinase I Inhibitor, D4476
Casein Kinase I Inhibitor, D4476 is a cell-permeable triaryl substituted imidazolo compound that acts as a selective inhibitor of casein kinase 1 (CK1)
301836-43-1 sc-202522
1 mg
$95.00
6
(1)
TGF-beta RI Kinase Inhibitor V
TGF-β RI Kinase Inhibitor V is a TGF-β signaling blocker
627536-09-8 sc-203294
2 mg
$84.00
3
(1)
LY 364947
LY 364947 is a selective ATP-competitive inhibitor of TGF-β Receptor I kinase
396129-53-6 sc-203122
sc-203122A
5 mg
10 mg
$103.00
$150.00
4
(1)
TGF-beta RI Kinase Inhibitor VII
TGF-β RI Kinase Inhibitor VII is an inhibitor of ALK5/TGF-β Receptor I kinase activity
666729-57-3 sc-356133
5 mg
$195.00
0
(0)
TGF-beta RI Kinase Inhibitor III
TGF-β RI Kinase Inhibitor III is an inhibitor of activin receptor-like kinase 4
356559-13-2 sc-204341
2 mg
$198.00
0
(0)
TGF-beta RI Kinase Inhibitor VIII
TGF-β RI Kinase Inhibitor VIII is a potent ATP-competitive inhibitor against receptor TbR-I/ALK5
356559-20-1 sc-203295
2 mg
$100.00
2
(1)
ALK5 Inhibitor II
ALK5 Inhibitor II is an ATP-competitive inhibitor of TGF-β RI kinase and has been used as an to inhibit autophosphorylation of ALK5.
446859-33-2 sc-221234
sc-221234A
sc-221234B
sc-221234C
sc-221234D
sc-221234E
sc-221234F
1 mg
5 mg
10 mg
50 mg
100 mg
500 mg
1 g
$67.00
$90.00
$176.00
$620.00
$1,200.00
$4,212.00
$7,665.00
6
(1)
LY2157299
LY2157299 is a potent TGF β RI inhibitor
700874-72-2 sc-391123
sc-391123A
5 mg
10 mg
$200.00
$340.00
3
(1)