GABA Receptor Activators

Santa Cruz Biotechnology now offers a broad range of GABA Receptor Activators. In the central nervous system GABA functions as the main inhibitory transmitter by increasing a Cl- conductance that inhibits neuronal firing. GABA has been shown to activate both ionotropic (GABAA) and metabotropic (GABAB) receptors as well as a third class of receptors called GABAC. GABA Receptor Activators offered by Santa Cruz activate GABA Receptor and, in some cases, other ionotropic and metabotropic receptor related proteins. View detailed GABA Receptor Activator specifications, including GABA Receptor Activator CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Etomidate
Etomidate is a GABAA receptors agonist
33125-97-2 sc-203577
10 mg
$122.00
0
(0)
Securinine
Securinine is a GABA receptor antagonist
5610-40-2 sc-220097
sc-220097A
50 mg
100 mg
$175.00
$350.00
2
(1)
(+/-)-Baclofen
(±)-Baclofen is a selective agonist of the GABAB receptor
1134-47-0 sc-200464
sc-200464A
1 g
5 g
$49.00
$243.00
0
(1)
4-Imidazoleacetic acid hydrochloride
4-Imidazoleacetic acid hydrochloride is a competitive antagonist at GABAC receptors
3251-69-2 sc-254684
1 g
$119.00
0
(0)
Isoguvacine HCl
Isoguvacine⋅HCl is an agonist of Gamma-amino butyric acid receptors
68547-97-7 sc-200451
sc-200451A
10 mg
50 mg
$25.00
$108.00
2
(0)
Indiplon
Indiplon is a potent GABAAreceptor positive allosteric modulator
325715-02-4 sc-204011
sc-204011A
10 mg
50 mg
$129.00
$516.00
0
(0)
R-(+)-Baclofen hydrochloride
R-(+)-Baclofen hydrochloride is a seelctive GABAB receptor agonist
63701-55-3 sc-203229
sc-203229A
10 mg
50 mg
$30.00
$117.00
0
(0)
GABA
GABA is an inhibitory neurotransmitter in the CNS
56-12-2 sc-203053
sc-203053A
sc-203053B
sc-203053C
10 g
25 g
5 kg
10 kg
$40.00
$82.00
$390.00
$720.00
1
(1)
Hispidulin
Hispidulin is a potent benzodiazepine (BZD) receptor ligand
1447-88-7 sc-203999
sc-203999A
sc-203999B
sc-203999C
10 mg
100 mg
500 mg
1 g
$245.00
$970.00
$2,945.00
$5,300.00
1
(0)
Muscimol
Muscimol is a potent and specific GABAA receptor agonist/GABA analog
2763-96-4 sc-200460
sc-200460A
5 mg
25 mg
$96.00
$225.00
2
(1)
Valerenic acid
Valerenic acid is a positive allosteric modulator of the GABAA receptor
3569-10-6 sc-204377
sc-204377A
1 mg
10 mg
$53.00
$460.00
1
(1)
TACA
TACA is a GABAA and GABAC agonist
38090-53-8 sc-203705
sc-203705A
10 mg
50 mg
$90.00
$290.00
0
(0)
THIP hydrochloride
THIP hydrochloride is a GABAA receptor agonist and GABAC receptor antagonist
64603-91-4 sc-204342
50 mg
$149.00
0
(0)
ZAPA sulfate
ZAPA sulfate is a selective potent GABAA receptor agonist
92138-10-8 sc-200471
sc-200471A
5 mg
25 mg
$71.00
$275.00
0
(0)
SKF 97541
SK&F 97541 is a very potent GABAB agonist/GABAC antagonist
127729-35-5 sc-200469
sc-200469A
5 mg
25 mg
$101.00
$450.00
0
(0)
R-(+)-Baclofen (free base)
R-(+)-Baclofen (free base) is a selective GABAB receptor agonist
69308-37-8 sc-203228
sc-203228A
10 mg
50 mg
$50.00
$195.00
0
(0)
Loreclezole hydrochloride
Loreclezole hydrochloride is a subtype-selective GABAA receptor agonist
117857-45-1 sc-204061
sc-204061A
10 mg
50 mg
$195.00
$849.00
0
(0)
rac BHFF
rac BHFF is a GABAB receptor positive allosteric modulator
123557-91-5 sc-204228
sc-204228A
5 mg
25 mg
$110.00
$420.00
0
(0)
SB 205384
SB 205384 is a GABAA receptor modulator
160296-13-9 sc-204263
sc-204263A
10 mg
50 mg
$195.00
$825.00
0
(1)
Org 20599
Org 20599 is a positive allosteric modulator and agonist of GABA receptors
156685-94-8 sc-204150
sc-204150A
10 mg
50 mg
$185.00
$781.00
0
(0)
U 89843A
U 89843A is a positive allosteric modulator of GABAA receptors
157013-85-9 sc-204361
sc-204361A
10 mg
50 mg
$125.00
$525.00
0
(0)
5-Nitro-alpha-oxo-N-(1R)-phenylethyl]-1H-indole-3-acetamide
TCS 1205 is a GABAA α2 agonist
355022-97-8 sc-358561
sc-358561A
10 mg
50 mg
$135.00
$595.00
0
(0)
DS2
DS2 is a positive allosteric modulator of δ-subunit containing GABAA receptors
374084-31-8 sc-294421
sc-294421A
10 mg
25 mg
$170.00
$715.00
0
(0)
AA 29504
AA 29504 is a positive allosteric modulator of GABAA receptors
945828-50-2 sc-361096
sc-361096A
5 mg
25 mg
$83.00
$350.00
0
(0)
(S)-Baclofen
(S)-Baclofen is a specific GABA-B receptor agonist
66514-99-6 sc-396081
sc-396081A
sc-396081B
sc-396081C
10 mg
25 mg
50 mg
100 mg
$250.00
$500.00
$930.00
$2,000.00
0
(0)
Chlormezanone
Chlormezanone is a compound acting at the benzodiazapine site of GABAA receptors
80-77-3 sc-203887
1 g
$67.00
0
(0)
CL 218872
CL 218872 is a benzodiazepine agonist selective for α1 subunit-containing GABAA receptors
66548-69-4 sc-203552
sc-203552A
10 mg
50 mg
$85.00
$319.00
0
(0)
CGS 20625
CGS 20625 is a central benzodiazepine receptor partial agonist
111205-55-1 sc-203545
sc-203545A
10 mg
50 mg
$169.00
$712.00
0
(0)
Primidone
Primidone is a compound that potentiates GABA receptor function
125-33-7 sc-204861
5 g
$37.00
0
(0)
Acamprosate Calcium
Acamprosate Calcium is a GABA receptor agonist and glutamatergic systems modulator
77337-73-6 sc-210733
100 mg
$140.00
0
(0)
L-838417
L-838417 is a subtype-selective GABAA receptor partial agonist
286456-42-6 sc-211693
5 mg
$209.00
0
(0)
Ganaxolone
Ganaxolone is a potent stereoselective modulator of GABAA receptors
38398-32-2 sc-203586
sc-203586A
10 mg
50 mg
$129.00
$560.00
0
(1)
7-Chloro-1-methyl-5-phenyl-[1,2,4]triazolo[4,3-a]quinolin-4-amine
7-Chloro-1-methyl-5-phenyl-[1,2,4]triazolo[4,3-a]quinolin-4-amine is an impurity of alprazolam
448950-89-8 sc-396449
5 mg
$300.00
0
(0)
Bretazenil
84379-13-5 sc-252512
5 mg
$150.00
0
(0)
Safranal
A chemical responsible for Saffron smell that is also a proposed GABA A receptor agonist activity in vitro
116-26-7 sc-472985
sc-472985A
sc-472985C
sc-472985B
sc-472985D
5 g
10 g
25 g
50 g
100 g
$100.00
$190.00
$370.00
$650.00
$1,150.00
0
(0)
Progabide
Progabide is a GABAA and GABAB receptor agonistic
62666-20-0 sc-476638
sc-476638A
100 mg
5 mg
$300.00
$20.00
0
(0)
1-Methyl-4-imidazoleacetic acid hydrochloride
1-Methyl-4-imidazoleacetic acid hydrochloride is a metabolite
35454-39-8 sc-222712
sc-222712A
10 mg
250 mg
$60.00
$600.00
0
(0)
5-Oxo-Zaleplon
5-Oxo-Zaleplon is a metabolite of Zaleplon, a selective non-benzodiazepine GABAA receptor agonist
159225-99-7 sc-478295
10 mg
$300.00
0
(0)
Baclofen-d4
Baclofen-d4 is a specific GABA-B receptor agonist
1189938-30-4 sc-217694
sc-217694A
1 mg
10 mg
$450.00
$2,900.00
0
(0)
3-Aminopropylphosphonic acid
3-Aminopropylphosphonic acid is a GABAB receptor agonist
13138-33-5 sc-251943
1 g
$142.00
0
(1)

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