Histamine Receptor Activators

Histamine is an inflammatory mediator that is ubiquitously expressed and has a broad range of pharmacologic effects. The effects of histamine are mediated by a family of G protein-coupled receptors, the Histamine H1, H2, H3 and H4 Receptors. Histamine Receptor Activators offered by Santa Cruz activate Histamine Receptor and, in some cases, other inflammation and immune response related proteins. View detailed Histamine Receptor Activator specifications, including Histamine Receptor Activator CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Amthamine
Amthamine is a very selective agonist of the histamine H2-receptor
142437-67-0 sc-201087
5 mg
$84.00
0
(0)
Dimaprit dihydrochloride
Dimaprit dihydrochloride is a specific agonist of the histamine H2-receptor
23256-33-9 sc-201090
100 mg
$94.00
0
(0)
Histamine dihydrochloride
Histamine dihydrochloride is a potent vasodilator and endogenous histamine receptor agonist
56-92-8 sc-202650
sc-202650A
sc-202650B
5 g
25 g
500 g
$40.00
$177.00
$481.00
1
(1)
Loratadine
Loratadine is a peripheral histamine H1 receptor agonist
79794-75-5 sc-203117
sc-203117A
10 mg
50 mg
$105.00
$446.00
1
(1)
4-Methylhistamine dihydrochloride
4-Methylhistamine dihydrochloride is a H4 receptor agonist
36376-47-3 sc-203475
sc-203475A
10 mg
50 mg
$175.00
$739.00
5
(1)
Imetit dihydrobromide
Imetit dihydrobromide is a high affinity agonist at the histamine H3- and H4-receptors
32385-58-3 sc-203602
10 mg
$110.00
0
(0)
Immethridine dihydrobromide
Immethridine dihydrobromide is a strong and highly selective histamine H3 receptor agonist
87976-03-2 sc-203603
sc-203603A
10 mg
50 mg
$145.00
$615.00
0
(0)
VUF 8430 dihydrobromide
VUF 8430 dihydrobromide is a potent histamine H4 receptor full agonist
100130-32-3 sc-203719
sc-203719A
5 mg
50 mg
$68.00
$548.00
0
(0)
Histamine, free base
Histamine, free base is a compound that activates NOS which results in the release of NO
51-45-6 sc-204000
sc-204000A
sc-204000B
1 g
5 g
25 g
$90.00
$272.00
$950.00
6
(1)
HTMT dimaleate
HTMT dimaleate is a mixed H1/H2 histamine agonist that is significantly more potent than histamine itself
195867-54-0 sc-204003
sc-204003A
10 mg
50 mg
$149.00
$615.00
0
(0)
Immepip dihydrobromide
Immepip dihydrobromide is an H3 and H4 receptor agonist
164391-47-3 sc-204010
sc-204010A
10 mg
50 mg
$155.00
$615.00
0
(0)
(+)-alpha-Methylhistamine dihydrobromide
(+)-α-Methylhistamine dihydrobromide is a less active enantiomer of H3 agonist R-(−)-α-methylhistamine
75614-93-6 sc-204426
sc-204426A
10 mg
50 mg
$119.00
$510.00
0
(0)
Proxyfan oxalate
Proxyfan oxalate is a high affinity histamine H3 receptor ligand
177708-09-7 sc-204867
sc-204867A
10 mg
50 mg
$139.00
$585.00
0
(0)
Histamine-α,α,β,β-d4 Dihydrochloride
Histamine-α,α,β,β-d4 Dihydrochloride is a deuterated analog of histamine
344299-48-5 sc-218580
sc-218580A
sc-218580B
sc-218580C
1 mg
2.5 mg
5 mg
10 mg
$290.00
$590.00
$1,095.00
$2,015.00
0
(0)
Histamine bisphosphate monohydrate
A potent histamine receptor agonist
51-74-1 sc-250117
5 g
$77.00
0
(0)
2-((3-Trifluoromethyl)phenyl)histamine dimaleate
2-((3-Trifluoromethyl)phenyl)histamine dimaleate is an extremely potent and selective H1 receptor agonist
162049-83-4 sc-251656
5 mg
$99.00
0
(0)