CB1 Activators

The cannabinoid receptors (CB1 and CB2) are G-protein coupled receptors that inhibit adenylate cyclase activity in response to psychoactive cannabinoids. Biochemicals that activate CB1 have many applications in biochemical and physiological research. Click on the product name to view detailed information such as the chemical structure and specific chemical properties for each of our CB1 Activators biochemicals. In stock CB1 Activators are available for immediate shipping.

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PRODUCT NAME/ApplicationCASCatalog #QUANTITYPriceCitationsRATING
Rimonabant
An immunomodulatory CB1 receptor inverse agonist
168273-06-1sc-205491
sc-205491A
5 mg
10 mg
$66.00
$152.00
11
(1)
Magnolol
An inhibitor of NO and TNF-α production
528-43-8sc-204797
sc-204797A
5 mg
25 mg
$42.00
$185.00
0
(0)
Oleamide
A CB1, 5-HT2A and 2C receptor agonist
301-02-0sc-358696
10 mg
$59.00
0
(1)
Leelamine HCl
A weak CB1 receptor agonist and PDK inhibitor
1446-61-3sc-200375
sc-200375A
10 mg
50 mg
$122.00
$520.00
0
(0)
ABN-CBD
An agonist of the novel cannabinoid receptor GPR55
22972-55-0sc-203488
10 mg
$225.00
0
(0)
Olvanil
A TRPV1 agonist more potent than capsaicin
58493-49-5sc-201454
sc-201454A
5 mg
25 mg
$47.00
$201.00
0
(0)
CP-55,940
A potent non-selective cannabinoid receptor agonist
83002-04-4sc-200359
sc-200359A
5 mg
25 mg
$162.00
$638.00
1
(1)
Arvanil
A cannabinoid CB1 and vanilloid TRPV1 (VR) agonist
128007-31-8sc-202065
5 mg
$62.00
0
(0)
DEA
An endocannabinoid agonist of the CB1 receptor
150314-35-5sc-203024
5 mg
$55.00
0
(0)
(R)-Methanandamide
A potent CB1 agonist and VR agonist
157182-49-5sc-200792
sc-200792A
5 mg
25 mg
$55.00
$172.00
1
(1)
ACEA
A potent and selective agonist of the CB1 receptors
220556-69-4sc-202902
sc-202902A
5 mg
25 mg
$69.00
$285.00
2
(1)
Arachidonylcyclopropylamide (ACPA)
A cannabinoid CB1 receptor agonist
229021-64-1sc-200795
sc-200795A
10 mg
50 mg
$62.00
$179.00
6
(1)
CB 13
A potent CB1/CB2 receptor agonist with limited brain penetration
432047-72-8sc-203870
sc-203870A
10 mg
50 mg
$115.00
$473.00
0
(0)
Anandamide
An endogenous cannabinoid receptor ligand
94421-68-8sc-396321
sc-396321A
5 mg
25 mg
$62.00
$190.00
1
(0)
Mead acid ethanolamide
A cannabinoid CB1 and CB2 agonist equipotent with anandamide1
169232-04-6sc-202704
sc-202704A
1 mg
10 mg
$87.00
$825.00
0
(0)
Arachidonamide (20:4, n-6)
A weak cannabinoid CB1 and CB2 agonist
85146-53-8sc-221258
sc-221258A
10 mg
50 mg
$96.00
$364.00
0
(0)
AM 1172
A potent and selective inhibitor of anandamide uptake and FAAH
251908-92-6sc-202456
sc-202456A
10 mg
50 mg
$200.00
$650.00
0
(0)
N-Arachidonoyl-L-serine
An endocannabinoid-like compound and CB1/CB2 agonist
187224-29-9sc-202718
10 mg
$230.00
1
(0)
Palmitoyl Ethanolamide-d4
A useful deuterium labeled palmitoyl ethanolamide
1159908-45-8sc-224199
sc-224199A
100 µg
500 µg
$28.00
$127.00
0
(0)
N-Arachidonyl maleimide
A highly potent and irreversible inhibitor
876305-42-9sc-394306
sc-394306A
5 mg
25 mg
$112.00
$421.00
0
(0)
Arachidonoyl 2prime-fluoroethylamide
A CB1 receptor agonist
166100-37-4sc-202469
5 mg
$200.00
0
(0)
Dihomo-gamma-linolenylethanolamide
A CB1 and CB2 agonist and adenylyl cyclase inhibitor
150314-34-4sc-202137
5 mg
$55.00
0
(0)
Yangonin
One of the major components of kava extract
500-62-9sc-205889
sc-205889A
5 mg
10 mg
$263.00
$500.00
0
(0)
MDA 19
A selective human peripheral cannabinoid CB2 receptor agonist
1048973-47-2sc-358804
sc-358804A
1 mg
5 mg
$27.00
$120.00
0
(0)
CB-52
A stable analog of THC and AEA with high affinity for central CB1 and peripheral CB2 receptors
sc-221404
sc-221404A
1 mg
5 mg
$38.00
$170.00
0
(0)
Arachidonoyl-1-thio-Glycerol
A thiol analog of 2-arachidonoyl glycerol
1309664-54-7sc-221265
sc-221265A
1 mg
5 mg
$44.00
$198.00
0
(0)
RVD-Hpalpha
A selective CB1receptor agonist which increases intracellular Ca2+ levels in cells expressing CB receptors in vitro
sc-361323
1 mg
$185.00
0
(0)

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