Histamine H1 Receptor Inhibitors
Santa Cruz Biotechnology now offers a broad range of Histamine H1 Receptor Inhibitors. Histamine is an inflammatory mediator that is ubiquitously expressed and has a broad range of pharmacologic effects. The effects of histamine are mediated by a family of G protein-coupled receptors, the Histamine H1, H2, H3 and H4 Receptors. Histamine H1 Receptor Inhibitors offered by Santa Cruz inhibit Histamine H1 Receptor and, in some cases, other inflammation and immune response related proteins. View detailed Histamine H1 Receptor Inhibitor specifications, including Histamine H1 Receptor Inhibitor CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.
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SEE ALSO...
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| PRODUCT NAME/Application | CAS | Catalog # | QUANTITY | Price | Citations | RATING | |
|---|---|---|---|---|---|---|---|
Ketotifen fumarateA histamine H1 antagonist and mast cell growth inhibitor |
34580-14-8 |
sc-201094 sc-201094A |
1 g 100 mg |
$62.00
$39.00 |
2 |
| |
LoratadineLoratadine is a peripheral histamine H1 receptor agonist |
79794-75-5 |
sc-203117 sc-203117A |
10 mg 50 mg |
$105.00
$446.00 |
1 |
| |
Chlorpromazine, HydrochlorideChlorpromazine, Hydrochloride is an inhibitor of PDE, D2DR, NOS1, and PLA2 |
69-09-0 |
sc-202537 sc-202537A sc-202537B sc-202537C sc-202537D |
500 mg 5 g 25 g 100 g 250 g |
$32.00
$48.00 $140.00 $480.00 $1,060.00 |
5 |
| |
TerfenadineTerfenadine is a histamine H1-receptor antagonist, which blocks HERG and KIR6 channels |
50679-08-8 |
sc-208421A sc-208421B sc-208421 |
500 mg 1 g 5 g |
$37.00
$64.00 $105.00 |
0 |
| |
AstemizoleAstemizole is a potent and selective H1-receptor antagonist that displays antihistamine and antimalarial activity |
68844-77-9 |
sc-201088 sc-201088A |
10 mg 50 mg |
$69.00
$275.00 |
2 |
| |
Methapyrilene HClMethapyrilene HCl is a specialty product for proteomics research |
135-23-9 |
sc-257708 |
1 g |
$94.00
|
0 |
| |
Diphenhydramine hydrochlorideDiphenhydramine hydrochloride is a histamine H1-receptor antagonist |
147-24-0 |
sc-204729 sc-204729A sc-204729B |
10 g 25 g 100 g |
$50.00
$80.00 $120.00 |
2 |
| |
Meclizine DihydrochlorideMeclizine Dihydrochloride is a histamine H1 receptor antagonist and PXR (pregnane X receptor) agonist |
1104-22-9 |
sc-211779A sc-211779 |
5 g 10 g |
$85.00
$150.00 |
2 |
| |
(S)-(+)-Dimethindene maleate(S)-(+)-Dimethindene maleate is a subtype-selective mAChR M2 antagonist and histamine H1 receptor antagonist |
121367-05-3 |
sc-361329 sc-361329A |
10 mg 50 mg |
$170.00
$700.00 |
0 |
| |
Mepyramine maleateMepyramine maleate is a histamine H1 receptor antagonist |
59-33-6 |
sc-203629 sc-203629A |
100 mg 1 g |
$65.00
$220.00 |
1 |
| |
Fluphenazine HydrochlorideFluphenazine Hydrochloride is a dopamine D1 and D2 receptor antagonist that can bind to histamine H1 |
146-56-5 |
sc-205700 sc-205700A sc-205700B sc-205700C |
1 g 5 g 50 g 100 g |
$86.00
$224.00 $835.00 $1,215.00 |
0 |
| |
LidocaineLidocaine is a selective inverse peripheral histamine H1-receptor agonist |
137-58-6 |
sc-204056 sc-204056A |
50 mg 1 g |
$49.00
$125.00 |
0 |
| |
Cyproheptadine hydrochlorideCyproheptadine hydrochloride is a non-selective 5-HT2 antagonist |
969-33-5 |
sc-203557 |
50 mg |
$85.00
|
2 |
| |
Brompheniramine MaleateBrompheniramine Maleate is a histamine H1 receptors antagonist |
980-71-2 |
sc-210967 sc-210967A |
25 mg 250 mg |
$60.00
$200.00 |
1 |
| |
Doxepin hydrochlorideDoxepin hydrochloride is a highly potent histamine H1 antagonist with affinity to H4 receptor |
1229-29-4 |
sc-203930 |
1 g |
$50.00
|
0 |
| |
Hydroxyzine DihydrochlorideHydroxyzine Dihydrochloride is a hetercyclic H1 receptor antagonist |
2192-20-3 |
sc-205716 sc-205716A |
5 g 10 g |
$75.00
$103.00 |
0 |
| |
Antazoline hydrochlorideAntazoline hydrochloride is an anticholinergic and antihistamine agent |
2508-72-7 |
sc-203515 sc-203515A sc-203515B |
100 mg 1 g 5 g |
$65.00
$80.00 $200.00 |
0 |
| |
Fenspiride HydrochlorideFenspiride Hydrochloride is an α adrenergic and H1 histamine receptor antaonist |
5053-08-7 |
sc-207684 |
10 mg |
$145.00
|
0 |
| |
trans-Triprolidine hydrochloridetrans-Triprolidine hydrochloride is a potent H1 receptor antagonist |
6138-79-0 |
sc-204354 |
1 g |
$35.00
|
0 |
| |
Clemastine fumarateClemastine fumarate is a selective histamine H1 antagonist |
14976-57-9 |
sc-203897 |
100 mg |
$95.00
|
0 |
| |
ZotepineZotepine is an SR-2A and D2DR inhibitor and Histamine H1 receptor antagonist |
26615-21-4 |
sc-360895 sc-360895A |
10 mg 50 mg |
$66.00
$246.00 |
2 |
| |
OxatomideOxatomide is an H1-histamine receptor antagonist |
60607-34-3 |
sc-208136 |
10 mg |
$200.00
|
0 |
| |
Azelastine HClAzelastine HCl is an H1-receptor antagonist with antiallergic effects and disrupts TNF alpha activity |
79307-93-0 |
sc-201096 sc-201096A sc-201096B sc-201096C sc-201096D |
100 mg 250 mg 1 g 5 g 10 g |
$92.00
$200.00 $642.00 $1,950.00 $3,200.00 |
0 |
| |
Levocabastine HydrochlorideLevocabastine Hydrochloride is a histamine H1 receptor antagonist and anti-allergic agent |
79547-78-7 |
sc-201095 |
10 mg |
$184.00
|
4 |
| |
Cetirizine DihydrochlorideCetirizine Dihydrochloride is a Histamine H1 receptor inverse agonist |
83881-52-1 |
sc-202992 |
50 mg |
$59.00
|
0 |
| |
MirtazapineMirtazapine is a potent SR-2, SR-3, and Histamine H1 receptor antagonist |
85650-52-8 |
sc-204088 sc-204088A |
10 mg 50 mg |
$105.00
$409.00 |
0 |
| |
EbastineEbastine is an antagonist of the histamine H1-receptor |
90729-43-4 |
sc-205663 sc-205663A |
1 g 5 g |
$104.00
$420.00 |
1 |
| |
Pemirolast Potassium SaltPemirolast Potassium Salt is an inhibitor of mast cell mediator release |
100299-08-9 |
sc-208156 |
10 mg |
$165.00
|
0 |
| |
DesloratadineDesloratadine is a potent and selective H1-receptor agonist |
100643-71-8 |
sc-202133 sc-202133A |
100 mg 500 mg |
$85.00
$384.00 |
3 |
| |
Olopatadine HydrochlorideOlopatadine Hydrochloride is a dual acting histamine H1-receptor antagonist and mast cell stabilizer |
140462-76-6 |
sc-212473 |
25 mg |
$140.00
|
0 |
| |
(S)-Azelastine Hydrochloride(S)-Azelastine Hydrochloride is n orally active Histamine H1 Receptor |
153408-27-6 |
sc-208363 |
1 mg |
$250.00
|
0 |
| |
(R)-Azelastine HydrochlorideAn orally active Histamine H1 Receptor |
153408-28-7 |
sc-208236 |
1 mg |
$250.00
|
0 |
| |
Fexofenadine HClFexofenadine HCl is an antihistamine that inhibits Cox-1, Cox-2, and is a histamine H1 receptor agonist |
153439-40-8 |
sc-203047 sc-203047A |
10 mg 50 mg |
$95.00
$399.00 |
0 |
| |
Asenapine maleateAsenapine maleate is An antagonist of noradrenalin, dopamine, 5-HT and receptors |
65576-45-6 |
sc-361110 sc-361110A |
10 mg 50 mg |
$145.00
$615.00 |
0 |
| |
Iso LoratadineIso Loratadine is an isomer of loratadine used to prepare tricyclic amides and ureas |
170727-59-0 |
sc-394085 |
5 mg |
$300.00
|
0 |
| |
4-Diphenylmethoxy-1-methylpiperidine hydrochloride4-Diphenylmethoxy-1-methylpiperidine hydrochloride is n inhibitor of Histamine H1 Receptor |
132-18-3 |
sc-254657 |
10 g |
$67.00
|
0 |
| |
Mianserin hydrochlorideMianserin hydrochloride is a non-selective 5-HT2 receptor antagonist with moderate affinity for 5-HT6 |
21535-47-7 |
sc-358986 |
100 mg |
$105.00
|
1 |
| |
Phenindamine HydrochloridePhenindamine Hydrochloride is a Histamine H1 receptor inhibitor |
5503-08-2 |
sc-460196 |
50 mg |
$280.00
|
0 |
| |
FexofenadineFexofenadine is A metabolite of of terfenadine, a H1-Histamine receptor antagonist |
83799-24-0 |
sc-218475 |
100 mg |
$200.00
|
1 |
| |
Chlorpheniramine MaleateChlorpheniramine Maleate is an antagonist of the histamine H1-receptor |
113-92-8 |
sc-204684 sc-204684A |
5 g 25 g |
$29.00
$49.00 |
1 |
| |
(S)-Cetirizine Dihydrochloride(S)-Cetirizine Dihydrochloride is a nonsedating type histamine H1-receptor antagonist |
163837-48-7 |
sc-208364 |
2.5 mg |
$250.00
|
0 |
| |
Olopatadine N-OxideOlopatadine N-Oxide is an active metabolite of Olopatadine |
203188-31-2 |
sc-212474 |
2.5 mg |
$280.00
|
0 |
| |
Fexofenadine-d6Fexofenadine-d6 is a H1-Histamine receptor antagonist |
548783-71-7 |
sc-211506 |
1 mg |
$210.00
|
2 |
| |
Doxylamine SuccinateDoxylamine Succinate is a H1 histamine receptor antagonist |
562-10-7 |
sc-211381 |
100 mg |
$100.00
|
1 |
| |
Epinastine HydrochlorideEpinastine Hydrochloride is a tetracyclic, histamine H1 receptor antagonist |
108929-04-0 |
sc-211420 |
10 mg |
$86.00
|
0 |
| |
Azelastine-13C,d3Azelastine-13C,d3 is A H1-histamine receptor antagonist |
58581-89-8 (unlabeled) |
sc-217683 |
1 mg |
$250.00
|
0 |
| |
Rupatadine FumarateRupatadine Fumarate is a dual histamine H1 and PAF antagonist |
182349-12-8 |
sc-212795 |
10 mg |
$160.00
|
0 |
| |
Diphenhydramine-d6 HydrochlorideDiphenhydramine-d6 Hydrochloride is a labeled H1-Histamine receptor antagonist |
147-24-0 (unlabeled) |
sc-218244 |
1 mg |
$250.00
|
0 |
| |
Loratadine-d4Loratadine-d4 is a labelled histamine H1-receptor inhibitor |
381727-27-1 |
sc-280929 |
1 mg |
$300.00
|
0 |
| |
Chlorprothixene HydrochlorideChlorprothixene Hydrochloride is a D2DR inhibitor |
6469-93-8 |
sc-211077 |
1 g |
$30.00
|
1 |
| |
HydroxyzineHydroxyzine is an H1 receptor antagonist |
68-88-2 |
sc-207748 |
500 mg |
$240.00
|
0 |
| |
Orphenadrine Citrate SaltOrphenadrine Citrate Salt is a histaminergic compound |
4682-36-4 |
sc-212481 |
5 g |
$45.00
|
0 |
| |
Promethazine HydrochloridePromethazine Hydrochloride is an antagonist of the histamine H1-receptor |
58-33-3 |
sc-212586A sc-212586 |
50 mg 100 mg |
$70.00
$90.00 |
0 |
| |
rac-N-Demethyl dimethindene-d3 hydrobromideCAS: 151562-10-6 (unlabeled free base), MF: C19H19D3N2•HBr, MW: 362.32 |
151562-10-6 (unlabeled free base) |
sc-500664 |
1 mg |
$280.00
|
0 |
| |
Astemizole-d3Astemizole-d3 is a labeled histamine H1-receptor anatagonist |
1189961-39-4 |
sc-217667 |
1 mg |
$450.00
|
0 |
| |
Cetirizine-d8, DihydrochlorideCetirizine-d8, Dihydrochloride is A nonsedating type histamine H1-receptor antagonist |
2070015-04-0 |
sc-217874 |
1 mg |
$285.00
|
0 |
| |
alpha-Hydroxy olopatadineα-Hydroxy olopatadine is an inhibitor of Histamine H1 Receptor. |
1331822-32-2 |
sc-489117 |
1 mg |
$300.00
|
0 |
| |
Hydroxyzine-d8 DihydrochlorideHydroxyzine-d8 Dihydrochloride is a H1 receptor antagonist |
sc-280807 |
1 mg |
$300.00
|
0 |
| ||
Hydroxyzine-d8Hydroxyzine-d8 is a H1 receptor antagonist |
68-88-2 (unlabeled) |
sc-280806 |
1 mg |
$165.00
|
0 |
| |
Olopatadine-d6 HydrochlorideOlopatadine-d6 Hydrochloride is a labeled Olopatadine |
1217229-05-4 |
sc-219484 |
1 mg |
$280.00
|
0 |
| |
Trimipramine-d3 Maleate SaltTrimipramine-d3 Maleate Salt is a serotonin transport blocker that also blocks norepinephrine uptake |
521-78-8 (unlabeled) |
sc-220342 |
1 mg |
$200.00
|
0 |
| |
Mebhydroline 1,5-naphthalenedisulfonate saltMebhydroline 1,5-naphthalenedisulfonate salt is a H1 histamine receptor antagonist |
6153-33-9 |
sc-263459 |
1 g |
$20.00
|
0 |
| |
Desmethyl NizatidineDesmethyl Nizatidine is a main metabolite of Nizatidine |
82586-78-5 |
sc-391545 |
2.5 mg |
$280.00
|
0 |
| |
AcrivastineAcrivastine is a second-generation antihistamine |
87848-99-5 |
sc-357283 sc-357283A |
10 mg 50 mg |
$100.00
$304.00 |
0 |
| |
Pheniramine maleate saltPheniramine maleate salt is A H1 histamine receptor antagonist |
132-20-7 |
sc-253258 |
5 g |
$110.00
|
0 |
| |
Bepotastine besilateBepotastine besilate is an inhibitor of Histamine H1 Receptor. |
190786-44-8 |
sc-482068 |
10 mg |
$79.00
|
0 |
| |
Desmethyl doxylamine |
1221-70-1 |
sc-500284 sc-500284A |
100 mg 1 g |
$300.00
$2,400.00 |
0 |
| |
Diphenylamine HydrochlorideDiphenylamine Hydrochloride is a antagonist of histamine H1 receptor |
537-67-7 |
sc-485023 |
25 g |
$68.00
|
0 |
|