AR Inhibitors

Santa Cruz Biotechnology now offers a broad range of AR Inhibitors. There are five general types of adrenergic receptors (ARs), designated α1, α2, β1, β2 and β3, which are found in different target tissues and differ in their affinities and responses to various agonists and antagonists. AR Inhibitors offered by Santa Cruz inhibit AR and, in some cases, other G protein-coupled receptor kinases (GRKs) and PKC-directed phosphorylation related proteins. View detailed AR Inhibitor specifications, including AR Inhibitor CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Rauwolscine dot HCl
Rauwolscine • HCl is a standard α-2-adrenergic (AR) antagonist
6211-32-1 sc-200151
100 mg
$98.00
0
(1)
ICI 89406
ICI 89406 is a β-adrenergic antagonist
53671-71-9 sc-361212
sc-361212A
10 mg
50 mg
$89.00
$510.00
0
(0)
Propranolol hydrochloride
Propranolol hydrochloride is a β1 and β2 adrenergic receptor blocker
3506-09-0 sc-3580
sc-3580B
1 g
5 g
$32.00
$117.00
6
(1)
Verapamil hydrochloride
Verapamil hydrochloride is a calcium channel protein inhibitor in cardiac muscle cells
152-11-4 sc-3590
sc-3590A
sc-3590B
100 mg
1 g
5 g
$25.00
$31.00
$90.00
18
(1)
Oxprenolol hydrochloride
Oxprenolol hydrochloride is a non-selective β-adrenergic antagonist that also displays intrinsic sympathomimetic activity
6452-73-9 sc-204152
sc-204152B
sc-204152C
sc-204152D
100 mg
2.5 g
10 g
50 g
$30.00
$1,900.00
$6,500.00
$13,000.00
2
(1)
Alfuzosin hydrochloride
Alfuzosin hydrochloride is an α 1 adrenoceptor antagonist
81403-68-1 sc-203812
sc-203812A
10 mg
50 mg
$79.00
$295.00
0
(1)
BRL-37344
BRL-37344 is a potent and selective β3-AR agonist
127299-93-8 sc-200154
5 mg
$105.00
3
(1)
S(-)-Propranolol hydrochloride
S(−)-Propranolol hydrochloride is a β-adrenergic receptor antagonist
4199-10-4 sc-200153
100 mg
$84.00
0
(1)
2-PMDQ
2-PMDQ is a potent and selective antagonist of the α1-AR adrenoceptor
139047-55-5 sc-203771
sc-203771A
10 mg
50 mg
$135.00
$560.00
0
(0)
Doxazosin Mesylate
Doxazosin Mesylate is an alpha-1-adrenoreceptor antagonist
77883-43-3 sc-205656
sc-205656A
50 mg
250 mg
$101.00
$390.00
2
(1)
Spironolactone
Spironolactone is a lactone for proteomic research
52-01-7 sc-204294
50 mg
$100.00
1
(1)
Phentolamine mesylate
Phentolamine mesylate is an α-adrenergic blocker
65-28-1 sc-205803
sc-205803A
50 mg
100 mg
$62.00
$125.00
1
(1)
Aaptamine
Aaptamine is a spongean alkaloid that can activate the p21 promoter in the absence of p53
85547-22-4 sc-202899
sc-202899A
1 mg
10 mg
$200.00
$750.00
0
(1)
Phentolamine hydrochloride
Phentolamine hydrochloride is an a-Adrenergic blocker
73-05-2 sc-205802
sc-205802A
sc-205802B
sc-205802C
sc-205802D
sc-205802E
sc-205802F
50 mg
100 mg
250 mg
500 mg
1 g
2 g
2.5 g
$75.00
$100.00
$220.00
$390.00
$750.00
$1,400.00
$1,700.00
1
(1)
Carnosol
Carnosol is a phytopolyphenol found in Rosemary that functions as an antioxidant, antimicrobial, & anticarcinogen
5957-80-2 sc-204672
sc-204672A
sc-204672B
sc-204672C
1 mg
5 mg
10 mg
50 mg
$79.00
$179.00
$578.00
$2,540.00
0
(0)
Galeterone
Galeterone is an antagonist to LNCaP AR
851983-85-2 sc-364495
sc-364495A
5 mg
25 mg
$183.00
$550.00
1
(0)
RX 821002 hydrochloride
RX 821002 hydrochloride is a selective α2-adrenoceptor antagonist
109544-45-8 sc-203686
sc-203686A
10 mg
50 mg
$69.00
$259.00
0
(0)
Phenoxybenzamine
A non-specific irreversible adrenergic (AR) antagonist
63-92-3 sc-3581
sc-3581A
200 mg
1 g
$23.00
$74.00
3
(1)
Isotetrandrine
Isotetrandrine is a biscoclaurine alkaloid inhibitor of G protein activation of PLA2
477-57-6 sc-200869
sc-200869A
1 mg
5 mg
$69.00
$251.00
0
(1)
Sotalol hydrochloride
Sotalol hydrochloride is a potent β adrenergic antagonist
959-24-0 sc-203699
sc-203699A
10 mg
50 mg
$60.00
$235.00
0
(1)
1,3-Dimethyl-8-phenylxanthine
CAS: 961-45-5, MF: C13H12N4O2, MW: 256.26, Purity: ≥98%
961-45-5 sc-253981
100 mg
$110.00
0
(0)
Doxepin hydrochloride
Doxepin hydrochloride is a highly potent histamine H1 antagonist with affinity to H4 receptor
1229-29-4 sc-203930
1 g
$32.00
0
(1)
(R)-(+)-Propranolol hydrochloride
(R)-(+)-Propranolol hydrochloride is a less active anantiomer the non-selective beta blocker propranolol
5051-22-9 sc-203678
sc-203678A
100 mg
1 g
$69.00
$325.00
0
(0)
Fenspiride Hydrochloride
Fenspiride Hydrochloride is an α adrenergic and H1 histamine receptor antaonist
5053-08-7 sc-207684
10 mg
$145.00
0
(0)
Clomipramine hydrochloride
Clomipramine hydrochloride is a selective ST, SLC6A2, and DAT inhibitor
17321-77-6 sc-203898
1 g
$36.00
2
(1)
ent-Levobunolol, Hydrochloride
ent-Levobunolol, Hydrochloride is an enantiomer of levobunolol
27867-05-6 sc-211411
100 mg
$220.00
0
(0)
Propafenone Hydrochloride
Propafenone Hydrochloride is a sodium channel protein inhibitor
34183-22-7 sc-204863
sc-204863A
sc-204863B
sc-204863C
1 g
5 g
25 g
100 g
$21.00
$64.00
$190.00
$481.00
0
(1)
Acebutolol Hydrochloride
Acebutolol Hydrochloride is a β-AR antagonist
34381-68-5 sc-217555
10 g
$220.00
0
(1)
Levobunolol, Hydrochloride
Levobunolol, Hydrochloride is a β-adrenoceptor antagonist
27912-14-7 sc-211734
sc-211734A
100 mg
250 mg
$700.00
$600.00
0
(1)
2-Hydroxy-flutamide
2-Hydroxy-flutamide is an inhibitor of proliferation of estradiol-induced growth of MCF-7 breast cancer cells
52806-53-8 sc-205574
sc-205574A
10 mg
25 mg
$140.00
$368.00
0
(1)
Urapidil HCl
Urapidil HCl is an adrenergic α1-AR antagonist and a serotonin 5-HT1A (SR-1A) receptor agonist
64887-14-5 sc-200155
100 mg
$120.00
0
(0)
Maprotiline Hydrochloride
Maprotiline Hydrochloride is A norepinephrine reuptake inhibitor shown to block apoptosis of spiny neurons
10347-81-6 sc-200156
1 g
$72.00
4
(1)
Fenoldopam hydrochloride
Fenoldopam hydrochloride is a selective D1-like dopamine receptor partial agonist
67227-56-9 sc-279160
10 mg
$159.00
0
(0)
Mirtazapine
Mirtazapine is a potent SR-2, SR-3, and Histamine H1 receptor antagonist
85650-52-8 sc-204088
sc-204088A
10 mg
50 mg
$105.00
$409.00
0
(1)
Carazolol
Carazolol is A high affinity β-adrenergic receptor antagonist
57775-29-8 sc-257215
sc-257215A
10 mg
200 mg
$50.00
$250.00
0
(1)
Dimebolin dihydrochloride
Dimebolin dihydrochloride is a histamine, AR, and Ca channel inhibitor
97657-92-6 sc-294348
sc-294348A
sc-294348B
1 mg
5 mg
50 mg
$37.00
$96.00
$384.00
0
(0)
Cyanopindolol hemifumarate
Cyanopindolol hemifumarate is a SR-1A/SR-1B antagonist
106469-57-2 sc-203906
sc-203906A
10 mg
25 mg
$159.00
$693.00
0
(0)
Niguldipine hydrochloride
Niguldipine hydrochloride is a selective α 1-adrenoceptor antagonist and dihydropyridine calcium channel blocker
113317-61-6 sc-201471
sc-201471A
10 mg
50 mg
$77.00
$312.00
0
(0)
Naftopidil hydrochloride
Naftopidil hydrochloride is an α1-AR adrenoceptor antagonist
57149-07-2 (free base) sc-203151
sc-203151A
10 mg
50 mg
$55.00
$175.00
0
(1)
S-(+)-Niguldipine hydrochloride
S-(+)-Niguldipine hydrochloride is a calcium channel protein inhibitor
113165-32-5 sc-203248
10 mg
$124.00
0
(0)
(S)-Timolol Maleate
(S)-Timolol Maleate is a selective β1-AR receptor antagonist
26921-17-5 sc-203297
sc-203297A
100 mg
250 mg
$59.00
$122.00
0
(1)
ARC 239 dihydrochloride
ARC 239 dihydrochloride is a selective α2B-AR adrenoreceptor antagonist
67339-62-2 sc-203518
5 mg
$125.00
0
(0)
Betaxolol hydrochloride
Betaxolol hydrochloride is a selective β1-AR adrenoceptor antagonist
63659-19-8 sc-203527
sc-203527A
10 mg
50 mg
$125.00
$480.00
0
(1)
2-MPMDQ
2-MPMDQ is a selective α1-AR adrenoceptor antagonist
149847-77-8 sc-203770
sc-203770A
10 mg
50 mg
$129.00
$548.00
0
(0)
(±)-Bisoprolol hemifumarate
(±)-Bisoprolol hemifumarate is a selective β1-AR antagonist
104344-23-2 sc-203531
sc-203531B
sc-203531A
10 mg
25 mg
50 mg
$115.00
$190.00
$462.00
0
(0)
Efaroxan hydrochloride
Efaroxan hydrochloride is a potent α2-AR adrenoceptor antagonist
89197-00-2 sc-203573
sc-203573A
10 mg
50 mg
$125.00
$525.00
0
(0)
(R)-Phenoxybenzamine Hydrochloride
(R)-Phenoxybenzamine Hydrochloride is an irreversible α-adrenergic antagonist
16053-59-1 sc-391970
5 mg
$280.00
0
(0)
HEAT hydrochloride
HEAT hydrochloride is a very selective α1-AR adrenoceptor antagonist
30007-39-7 sc-203996
sc-203996A
10 mg
50 mg
$115.00
$440.00
0
(0)
Urapidil
Urapidil is an a1-adrenergic antagonist with high affinity for 5-hydroxytryptamine sites.
34661-75-1 sc-391143
sc-391143A
500 mg
5 g
$120.00
$762.00
0
(0)
SDZ 21009
SDZ 21009 is a β-AR, SR-1A, and SR-1B antagonist
39731-05-0 sc-203695
sc-203695A
10 mg
50 mg
$200.00
$825.00
0
(0)
BMY 7378 dihydrochloride
BMY 7378 dihydrochloride is a SR-1A agonist and a selective α1D-AR antagonist
21102-95-4 sc-203849
sc-203849A
10 mg
50 mg
$44.00
$205.00
0
(0)
Bucindolol
Bucindolol is a non-selective β-AR adrenoceptor antagonist
71119-11-4 sc-203860
sc-203860A
10 mg
50 mg
$235.00
$750.00
1
(1)
CGP 12177 hydrochloride
CGP 12177 hydrochloride is a β1/β2-AR adrenoreceptor agonist
81047-99-6 sc-203878
sc-203878A
10 mg
50 mg
$75.00
$172.00
0
(0)
CGP 20712 Dihydrochloride
CGP 20712 Dihydrochloride is a highly potent and selective β1-AR antagonist
1216905-73-5 sc-203879
sc-203879A
10 mg
50 mg
$210.00
$865.00
0
(0)
Idazoxan hydrochloride
Idazoxan hydrochloride is an α2-AR adrenoceptor antagonist and I2 imidazoline receptor agonist.
79944-56-2 sc-204006
sc-204006A
10 mg
50 mg
$125.00
$495.00
2
(0)
N-(4-Amino-6,7-dimethoxyquinazol-2-yl)-N-methyl-2-cyanoethylamine
76362-28-2 sc-211970
100 mg
$280.00
0
(0)
JP 1302 dihydrochloride
JP 1302 dihydrochloride is a selective α2C-AR
80259-18-3 sc-204026
sc-204026A
10 mg
50 mg
$185.00
$772.00
0
(0)
Nebivolol hydrochloride
Nebivolol hydrochloride is a highly selective β1-adrenoceptor antagonist
152520-56-4 sc-204122
sc-204122A
10 mg
50 mg
$139.00
$224.00
0
(0)
2-phenyl-amino-N6-endo-norbornyladenine
2-phenyl-amino-N6-endo-norbornyladenine is an A3 AR antagonist
863202-33-9 sc-205088
sc-205088A
500 µg
1 mg
$208.00
$368.00
1
(0)
rac Nebivolol Hydrochloride
rac Nebivolol Hydrochloride is a racimic mixture of β1-Adrenergic blocker (β1-AR) used as an antihypertensive
169293-50-9 sc-391275
10 mg
$220.00
0
(0)
1,1-Dichloro-2,2-bis(4-chlorophenyl)ethene
1,1-Dichloro-2,2-bis(4-chlorophenyl)ethene is a potent androgen receptor antagonist
72-55-9 sc-251534
1 g
$55.00
0
(0)
(S)-(-)-Verapamil Hydrochloride
(S)-(−)-Verapamil Hydrochloride is an isomer that inhibits the p-glycoprotein efflux pump in MDR tumor cell lines
36622-29-4 sc-208338
1 mg
$350.00
0
(0)
Asenapine
Asenapine is a combined 5HT2, adrenergic, and D2 receptor antagonist
65576-45-6 sc-210839
10 mg
$280.00
0
(0)
rac Propranolol-d7
rac Propranolol-d7 is an anti-hypertensive, anti-anginal and anti-arrhythmic β-AR (β-Adrenergic receptor) blocker
98897-23-5 sc-212742
5 mg
$225.00
1
(0)
8-Benzyloxy-5-((R)-2-bromo-1-hydroxyethyl)-1H-quinolinone
8-Benzyloxy-5-((R)-2-bromo-1-hydroxyethyl)-1H-quinolinone is a chemical used in the preparation of phenylethanolamine derivatives
530084-79-8 sc-396009
2.5 mg
$280.00
0
(0)
Spironolactone-d6 (Major)
Spironolactone-d7 (Major) is a renal competitive MCR (aldosterone receptor) antagonist
52-01-7 unlabeled sc-220132
sc-220132A
1 mg
10 mg
$250.00
$2,000.00
0
(0)
Benzoestrol
Benzoestrol is a nonsteroidal estrogen antagonist
85-95-0 sc-210870
5 mg
$300.00
0
(0)
(R,R)-Labetalol Hydrochloride
(R,R)-Labetalol Hydrochloride is A competitive antagonist at both α-and β-adrenergic receptor sites
75659-08-4 sc-212635
1 mg
$350.00
0
(0)
Tolazoline Hydrochloride
Tolazoline Hydrochloride is a peripheral vasodilator
59-97-2 sc-213056
sc-213056A
sc-213056B
10 g
25 g
100 g
$45.00
$90.00
$180.00
0
(1)
Chlorprothixene Hydrochloride
Chlorprothixene Hydrochloride is a D2DR inhibitor
6469-93-8 sc-211077
1 g
$30.00
0
(1)
BRL 44408 MALEATE
BRL 44408 MALEATE is a selective α2A-AR antagonist
118343-19-4 sc-217791
10 mg
$143.00
0
(0)
Azaperone
Azaperone is an α-adrenergic, dopamine and histamine receptor inhibitor
1649-18-9 sc-210851
100 mg
$284.00
0
(0)
Mirtazapine-d3
Mirtazapine-d3 is an α2-Adrenergic blocker
1216678-68-0 sc-218855
1 mg
$300.00
0
(0)
Sotalol-d6 Hydrochloride
Sotalol-d6 Hydrochloride is A deuterium labeled β-adronergic blocker
1246820-85-8 sc-220127
1 mg
$280.00
0
(0)
Trimipramine-d3 Maleate Salt
Trimipramine-d3 Maleate Salt is a serotonin transport blocker that also blocks norepinephrine uptake
521-78-8 (unlabeled) sc-220342
1 mg
$200.00
0
(0)
Imiloxan Hydrochloride
Imiloxan Hydrochloride is a highly selective α2B-AR antagonist
81167-22-8 sc-224023
sc-224023A
5 mg
25 mg
$211.00
$849.00
0
(0)
Labetalol hydrochloride
Labetalol hydrochloride is a competitive α-AR (α-adrenoceptor) and β-AR (β-adrenoceptor) antagonist with antihypertensive propertie
32780-64-6 sc-252942
5 g
$77.00
0
(1)

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