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NOMBRE DEL PRODUCTO NÚMERO DE CATÁLOGODESCRIPCIÓNMENCIONESCLASIFICACIÓN
1-(1-Naphthyl)piperazine·HClsc-201139A mixed modulator of serotonin 5-HT receptors. Demonstrates agonism of the 5-HT1A receptors and antagonism of the 5-HT2A/2C receptors. NÚMERO DE CAS 57536-86-4

Clomipramine hydrochloridesc-203898Clomipramine hydrochloride (Anafranil) is an ST (serotonin transporter/SERT), SLC6A2 (norepinephrine transporter/NET), and DAT (dopamine transporter) blocker with Ki of 0.14, 54 and 3 nM, respectively. NÚMERO DE CAS 17321-77-6

RS-127445sc-364604RS-127445 is a high affinity 5-HT2B receptor antagonist with modest efficacy against 5-HT2A/C and 5-HT5/6/7. NÚMERO DE CAS 199864-87-4

1-Methylpsilocinsc-2037641-Methylpsilocin is a potent and selective SR-2C agonist. NÚMERO DE CAS 1465-16-3

Citalopram hydrobromidesc-203551Citalopram hydrobromide is a salt form of Citalopram (sc-201123). Citalopram is a selective inhibitor of ST (5-hydroxytryptamine/serotonin transporter) and therefore is a potent and selective serotonin reuptake inhibitor. NÚMERO DE CAS 59729-32-7

1-Phenylbiguanidesc-222728 NÚMERO DE CAS 102-02-3

Mesulergine hydrochloridesc-361251Mesulergine hydrochloride is a D2-like dopamine receptor partial agonist and a SR-2A/SR-2C antagonist. NÚMERO DE CAS 64795-35-3

1-Phenylbiguanide hydrochloridesc-2034551-Phenylbiguanide hydrochloride is a SR-3 agonist. NÚMERO DE CAS 55-57-2

Indatraline hydrochloridesc-203605Indatraline hydrochloride is a strong monoamine uptake inhibitor which inhibits the transporters ST (serotonin/SERT), DAT (dopamine), and SLC6A2 (noradrenalin/NET). NÚMERO DE CAS 86939-10-8

BIMU 8sc-362714BIMU 8 is a potent SR-4 full agonist. NÚMERO DE CAS 134296-40-5

2-[1-(4-Piperonyl)piperazinyl]benzothiazolesc-2037672-[1-(4-Piperonyl)piperazinyl]benzothiazole is a SR-4 agonist with moderate activity as a SR-3 antagonist.

Fluoxetine HClsc-201125Fluoxetine is an ST (5-hydroxytryptamine/serotonin/5-HT reuptake) inhibitor. NÚMERO DE CAS 56296-78-7

3
2-Methylserotonin·HClsc-2011362-Methylserotonin·HCl is a SR-3 agonist shown to have low binding activity for SR-1A, SR-1B, SR-1C, and SR-2 binding sites. NÚMERO DE CAS 78263-90-8

Milnacipran hydrochloridesc-204086Milnacipran inhibits both SLC6A2 (norepinephrine transporter/NET) and ST (norepinephrine transporter/SERT) with IC50 of 77 nM and 420 nM, respectively. NÚMERO DE CAS 101152-94-7

3-AQCsc-2037763-AQC is a competitive SR-3 antagonist, almost 100 times more potent than tropisetron, but with widely differing activity in various tissues.

3-Oxo Citalopramsc-209668An intermediate of Citalopram and a potent and selective inhibitor of the 5-hydroxytryptamine transporter (serotonin). NÚMERO DE CAS 372941-54-3

4-[3-(Benzotriazol-1-yl)propyl]-1-(2-methoxyphenyl)piperazine oxalatesc-220919Strong pre- and postsynaptic 5-HT1A receptor antagonist.

Sertraline HClsc-201104Sertraline HCl is a selective and potent inhibitor of ST (serotonin transporter), increasing availability of serotonin in the brain. NÚMERO DE CAS 79559-97-0

1
4F 4PP oxalatesc-2037824F 4PP oxalate is a selective SR-2A antagonist.

Graminesc-255191 NÚMERO DE CAS 87-52-5

B-HT 920sc-203523B-HT 920 is a dopamine D2 receptor agonist, SR-3 antagonist and α2-adrenoceptor agonist. It also displays antiparkinsonian activity. NÚMERO DE CAS 36085-73-1

5-Carboxamidotryptamine maleatesc-2034775-Carboxamidotryptamine maleate is a SR-1 agonist with high affinity at SR-1A, SR-1B, SR-1D, SR-5 and SR-7. NÚMERO DE CAS 74885-09-9

(5-Hydroxy-1H-indol-3-yl)acetic acidsc-299847 NÚMERO DE CAS 1321-73-9

5-Nonyloxytryptamine oxalatesc-2034805-Nonyloxytryptamine oxalate is a selective SR-1B agonist. It is inactive as a SR-1A agonist (Ki at SR-1B = 1 nM, selectivity over SR-1B > 300-fold). NÚMERO DE CAS 157798-12-4

Venlafaxine Hydrochloridesc-201102Venlafaxine Hydrochloride is a dual ST and SLC6A2 (serotonin and noradrenalin re-uptake) inhibitor that displays ~ 30-fold higher affinity for ST (SERT) than SLC6A2 (NET). NÚMERO DE CAS 99300-78-4

8-Hydroxy-DPAT • HBrsc-2011298-Hydroxy-DPAT HBr is a SR-1A agonist with high affinity for SR-1A and SR-7 subtypes. NÚMERO DE CAS 87394-87-4

3
8-Hydroxy-PIPAT oxalatesc-3610908-Hydroxy-PIPAT oxalate is a high affinity SR-1A agonist. NÚMERO DE CAS 159651-91-9

(±)α-Methylserotonin maleatesc-201134(±)α-Methylserotonin maleate is a racemic mixture of α-methylserotonin maleate. it is a serotonin receptor agonist with preference for SR-2A, SR-2B, SR-2C. NÚMERO DE CAS 304-52-9

Almotriptan Hydrochloridesc-210786A Serotonin 5HT1B /1D-receptor agonist. NÚMERO DE CAS 154323-46-3

Altanserin hydrochloridesc-203504Altanserin hydrochloride is a selective and potent SR-2A antagonist. In addition, it can be used to determine malfunction in serotonergic neurotransmission. NÚMERO DE CAS 76330-71-7

Amperozide hydrochloridesc-203512Atypical antipsychotic which displays a high affinity for 5-HT2 receptors (Ki = 26 nM) and a low affinity for D2 receptors. Supresses ethanol drinking in genetically ethanol-preferring rats. NÚMERO DE CAS 75558-90-6

Urapidil HClsc-200155Urapiidil HCl is an adrenergic α1-AR antagonist and a serotonin 5-HT1A (SR-1A) receptor agonist. NÚMERO DE CAS 64887-14-5

Anpirtoline hydrochloridesc-201108Anpirtoline hydrochloride is a selective agonist of SR-1B. It shows strong selectivity at SR-1B over the SR-1A and SR-2 subtypes. Anpirtoline is also described to produce antagonism at the SR-3. NÚMERO DE CAS 98330-05-3

AS 19sc-203826AS 19 is reported to be a potent SR-7 agonist.

Asenapine maleatesc-361110Asenapine maleate is an antagonist of noradrenalin, dopamine, 5-HT and histamine receptor subtypes. NÚMERO DE CAS 65576-45-6

Azasetron Hydrochloridesc-210852A 5-HT3 receptor antagonist which is used as an anti-emetic. NÚMERO DE CAS 123040-69-7

BP 554 maleatesc-203851BP 554 maleate is a selective SR-1A agonist. NÚMERO DE CAS 82900-57-0

BRL 15572 hydrochloridesc-202979BRL 15572 hydrochloride is a selective SR-1D antagonist, displaying 60-fold selectivity over SR-1B, and exhibiting little or no affinity for a range of other receptor types. NÚMERO DE CAS 193611-72-2

BRL 54443sc-203855BRL 54443 is a potent SR-1E and SR-1F agonist. NÚMERO DE CAS 57477-39-1

BRL 54443 maleate saltsc-300302BRL 54443 maleate salt has been shown to be a potent agonist for the 5-HT1E/1F serotonin receptor. NÚMERO DE CAS 1197333-54-2

Bupropion HClsc-201121Bupropion HCl is a non-selective inhibitor of dopamine and SLC6A2 (Ki values are 1.4 μM for SLC6A2, 2.8 μM for dopamine, and 45 μM for serotonin). NÚMERO DE CAS 31677-93-7

Buspirone hydrochloridesc-202982Buspirone hydrochloride is a SR-1A partial agonist. NÚMERO DE CAS 33386-08-2

BW 723C86 hydrochloridesc-203428BW 723C86 hydrochloride is an activator of SR-2B. NÚMERO DE CAS 160521-72-2

CGS 12066B dimaleatesc-201106CGS 12066B dimaleate is a pyrroloquinoxaline agonist of SR-1B. It is described to be selective for SR-1B, with a 10-fold selectivity over SR-1A receptor and a 1000-fold selectivity over SR-2C. NÚMERO DE CAS 109028-10-6

CGS-12066A maleate saltsc-3003455-HT1B serotonin receptor agonist. NÚMERO DE CAS 109028-09-3

Cinanserinsc-201110Serotonin 5-HT2 antagonist. NÚMERO DE CAS 1166-34-3

Cinanserin hydrochloridesc-361149Cinanserin hydrochloride is a 5-HT2 antagonist. NÚMERO DE CAS 1166-34-3 (non-salt)

cis-Urocanic acidsc-214741This 5-HT agonist is a product of uv isomerization of trans-urocanic acid in skin. This leads to immunosuppression via activation of 5-HT2A receptor. NÚMERO DE CAS 7699-35-6

rac-trans-Sertralinesc-212762Used in the treatment of menopause and mood, anxiety, and cognitive disorders NÚMERO DE CAS 79836-45-6

Cisapridesc-203894Cisapride is a SR-4 agonist that stimulates intestinal ACh. NÚMERO DE CAS 81098-60-4

Nemonapridesc-204123Nemonapride is a highly selective D2DR antagonist and potent SR-1A agonist. NÚMERO DE CAS 75272-39-8

3
Citalopramsc-201123A selective inhibitor of the 5-hydroxytryptamine transporter (serotonin) and therefore is a potent and selective serotonin reuptake inhibitor. NÚMERO DE CAS 59729-33-8

Citalopram N-Oxidesc-207444A metabolite of Citalopram and a potential selective inhibitor of the 5-hydroxytryptamine transporter (serotonin). NÚMERO DE CAS 63284-72-0

CJ 033466sc-205257CJ 033466 is a selective and potent SR-4 partial agonist. It’s selectivity for SR-4 is substantially greater than that of other serotonin receptors and D2 receptors. NÚMERO DE CAS 519148-48-2

CP 809101 hydrochloridesc-205277CP 809101 hydrochloride is a potent and selective SR-2C agonist. NÚMERO DE CAS 479683-64-2

CP 93129 dihydrochloridesc-203904CP 93129 dihydrochloride is a selective SR-1B agonist. NÚMERO DE CAS 127792-75-0

WAY 208466 dihydrochloridesc-361404WAY 208466 dihydrochloride is a high affinity, selective SR-6 (5-HT6) receptor agonist. NÚMERO DE CAS 633304-27-5

CP 94253 hydrochloridesc-203905CP 94253 hydrochloride is a potent, selective SR-1B agonist. NÚMERO DE CAS 131084-35-0

Cyanopindolol hemifumaratesc-203906Cyanopindolol hemifumarate is a SR-1A and SR-1B antagonist. It is also a β-adrenergic antagonist. NÚMERO DE CAS 106469-57-2

Cyproheptadine hydrochloridesc-203557Migraine prophylactic and Non-selective 5HT2 antagonist. NÚMERO DE CAS 969-33-5

Demethylchloro Citalopram Hydrochloridesc-207519A derivative of Citalopram and a potentially useful internal standard. NÚMERO DE CAS 64372-52-7

Dibenzepine HClsc-201115Dibenzepine HCl is a tricyclic antidepressant used in the treatment of depression especially endogenous depression. NÚMERO DE CAS 315-80-0

Didemethylchloro Citalopram Hydrochloridesc-207565A derivative of Citalopram and potentially useful as an internal standard. NÚMERO DE CAS 887354-48-5

Quetiapine Fumaratesc-219681Quetiapine fumarate is an inhibitor of D2DR and SR-2A. NÚMERO DE CAS 111974-72-2

Dihydroergocristine mesylatesc-201117Dihydroergocristine mesylate demonstrates antagonism at serotonin receptors (SR) and partial agonism/antagonism of dopaminergic and adrenergic receptors. NÚMERO DE CAS 24730-10-7

2
Dihydroergotamine Methanesulfonate Saltsc-294343A competitive serotonin antagonist and vasoconstrictor. NÚMERO DE CAS 11032-41-0

Dolasetronsc-204733An antiserotonin used as an antiemetic to prevent nausea and vomiting brought on by chemotherapy or general anaesthesia. NÚMERO DE CAS 115956-12-2

Eicosapentaenoyl Serotoninsc-358802Eicosapentaenoyl serotonin is a hybrid molecule patterned after arachidonoyl serotonin (sc-201460). NÚMERO DE CAS 199875-71-3

Pindololsc-204847Pindolol is a SR-1A/SR-1B antagonist with similar affinity for each subtype. NÚMERO DE CAS 13523-86-9

Eltoprazine hydrochloridesc-203574Eltoprazine hydrochloride is a SR-1 and SR-2C receptor partial agonist. NÚMERO DE CAS 98224-03-4

EMD 386088 hydrochloridesc-203575EMD 386088 hydrochloride is a potent SR-6 receptor agonist that displays selectivity to other serotonin receptors. NÚMERO DE CAS 54635-62-0

ent-Frovatriptansc-207622Serotonin 5-HT1B/1D receptor agonist. It is a triptan drug for the treatment of migraine headaches. Frovatriptan causes vasoconstriction of arteries and veins that supply blood to the head. NÚMERO DE CAS 158930-18-8

Roxindole hydrochloridesc-203685Selective and potent presynaptic D-2 dopamine autoreceptor agonist. Inhibits serotonin (5-HT) uptake. NÚMERO DE CAS 112192-04-8

Fananserinsc-203951Fananserin is a potent serotonin SR-2A and dopamine D4 antagonist, with efficacy against histamine H1, α1 and SR-1A. NÚMERO DE CAS 127625-29-0

Fluperlapinesc-201119Fluperlapine is an atypical antipsychotic agent and ligand for the serotonin receptors 5-HT6/5-HT7. NÚMERO DE CAS 67121-76-0

2
Fluvoxamine maleatesc-203582A selective serotonin reuptake inhibitor with high affinity for the 5-HT transporter (Ki = 1.6 nM). NÚMERO DE CAS 61718-82-9

SKF 38393 HClsc-203264SKF 38393 HCl is a selective dopamine D1DR agonist that seems to be correlated to induced desynchronization of electroencephalographic activity in rats. NÚMERO DE CAS 81633-77-4

GR 113808sc-361189A robust and selective receptor antagonist of SR-4. NÚMERO DE CAS 144625-51-4

GR 125487 sulfamatesc-361190GR 125487 sulfamate is a selective and effective receptor antagoonist of SR-4 antagonist. NÚMERO DE CAS 144625-67-2

GR 127935 hydrochloride hydratesc-250068A selective, potent and orally active 5-HT1B/1D serotonin receptor antagonist. NÚMERO DE CAS 148642-42-6 (anhydrous)

GR 55562 dihydrochloridesc-361196GR 55562 dihydrochloride is a selective SR-1B (SR-1Bβ) antagonist. It has been shown to express weak binding at a number of serotonin receptor subtypes. NÚMERO DE CAS 172854-55-6

Granisetron hydrochloridesc-203984Granisetron hydrochloride is a SR-3 antagonist that possesses potent antiemetic activity. NÚMERO DE CAS 107007-99-8

Indorenate hydrochloridesc-2040125-HT receptor agonist with high affinity for 5-HT1A receptors (pKd = 7.8) and lower affinity for 5-HT1B and 5-HT2C receptors (pKd values are 5.44 and 6.49 respectively). Possesses anti-hypertensive, anorectic, and anxiolytic activity in vivo. NÚMERO DE CAS 72318-55-9

Ipsapironesc-203607Ipsapirone is a SR-1A agonist that has been found to selectively bind SR-1 receptors. It is also an anti-apoptotic agent that augments NF-κB, Bcl-XL, catalase, and XIAP expressions in neurons. NÚMERO DE CAS 95847-70-4

Isamoltane hemifumaratesc-203608Isamoltane hemifumarate is a SR-1B antagonist, with approximately 30-fold selective over SR-1B. Isamoltane hemifumarate possesses affinity for β-adrenergic receptors. NÚMERO DE CAS 55050-95-8

Ketanserin tartratesc-201131Ketanserin tartrate is a seletive serotonin agonist with reported ability to distinguish between various serotonin receptor subtypes. NÚMERO DE CAS 83846-83-7

L-694,247sc-361223L-694,247 is known to be a highly potent and selective SR-1D agonist. NÚMERO DE CAS 137403-12-4

Lofepraminesc-203624Serotonin and noradrenalin re-uptake inhibitor (SNRI) that is metabolized to desipramine (sc-200158, sc-207535). Produces inhibition of liver tryptophan pyrollase activity in vitro and displays antidepressant properties in vivo.Lofepramine has also been shown to be effective against Multiple Sclerosis in combination with L-phenylalanine. NÚMERO DE CAS 23047-25-8

LP 12 hydrochloride hydratesc-300940This product is a 5-HT7 receptor agonist found to display selectivity over D2, 5-Ht1A and 5-HT2A.

Zotepinesc-360895Zotepine is a SR-2A and D2DR inhibitor (Ki values are 0.69 and 2.3 nM respectively). Zotepine is also a potent histamine H1 receptor antagonist (IC50 = 8.0 nM). NÚMERO DE CAS 26615-21-4

LP 44sc-224044LP 44 is a high affinity SR-7 agonist. NÚMERO DE CAS 824958-12-5

LY 344864 hydrochloridesc-361245LY 344864 hydrochloride is a potent and selective SR-1F agonist. NÚMERO DE CAS 186544-26-3

LY-310,762 hydrochloridesc-300941LY-310,762 hydrochloride is a selective and potent SR-1D antagonist. NÚMERO DE CAS 192927-92-7

m-Chlorophenylbiguanide hydrochloridesc-203125m-Chlorophenylbiguanide hydrochloride is a potent and selective SR-3 agonist. NÚMERO DE CAS 2113-05-5

McN 5652, (+/-)sc-203627Potent, orally active 5-HT uptake inhibitor. Inhibits dopamine and noradrenaline uptake in vitro NÚMERO DE CAS 96795-89-0

MDL 11,939sc-204069MDL 11,939 is a potent, selective SR-2 antagonist. NÚMERO DE CAS 107703-78-6

2
MDL 72832 hydrochloridesc-204070Potent, selective and stereospecific ligand for central and peripheral 5-HT1A recognition sites. NÚMERO DE CAS 113777-33-6

MDL 73005EF hydrochloridesc-204071MDL 73005EF hydrochloride is a potent and selective SR-1A partial agonist with putative anxiolytic properties. NÚMERO DE CAS 124756-23-6

MDL-72222sc-201132MDL-72222 is a potent and highly selective antagonist at neuronal 5-hydroxytryptamine receptors, especially SR-3. NÚMERO DE CAS 40796-97-2

Melperone hydrochloridesc-204074Melperone hydrochloride is an atypical neuroleptic; 5-HT2A receptor antagonist and D2DR inhibitor. NÚMERO DE CAS 1622-79-3

Metergolinesc-204079Antagonist at 5-HT1, 5-HT2, and 5-HT7 serotonin receptors; also 5-HT1D ligand. moderate affinity for 5-HT6 and high affinity for 5-HT7. Analgesic; antipyretic. NÚMERO DE CAS 17692-51-2

Methiothepin maleatesc-203630Has moderate affinity for 5-ht5 and high affinity for 5-ht6 and 5-HT7. Also antagonist at 5-HT1 and 5-HT2 Potent 5-HT2 antagonist, also active as 5-HT1 antagonist. Differentiates 5-HT1D sub-types. NÚMERO DE CAS 20229-30-5

Methylergometrine maleatesc-203631Active metabolite of methysergide. Used as an oxytocic. NÚMERO DE CAS 113-42-8

Mexiletine hydrochloridesc-203633A use dependent blocker of sodium channels in skeletal muscle tissue. NÚMERO DE CAS 5370-01-4

Mianserin hydrochloridesc-3589865-HT2/5-HT1 antagonist. Has moderate affinity for 5-ht6 Non-selective 5-HT2 receptor antagonist. Has moderate affinity for 5-HT6. Antidepressant. NÚMERO DE CAS 21535-47-7

Mirtazapinesc-204088Mirtazapine is a potent SR-2 and SR-3 antagonist. In addition, it is a moderately potent α2 adrenoceptor and histamine H1-antagonist. NÚMERO DE CAS 85650-52-8

MK 212 hydrochloridesc-203634MK 212 hydrochloride is a SR-2C agonist. NÚMERO DE CAS 64022-27-1

ML 10302sc-363330 NÚMERO DE CAS 148868-55-7

ML 10302 hydrochloridesc-204089ML 10302 hydrochloride is a potent SR-4 partial agonist that displays > 680-fold selectivity over SR-3. NÚMERO DE CAS 148868-55-7

MM 77 dihydrochloridesc-204090MM 77 dihydrochloride is a highly potent and fairly selective SR-1A (postsynaptic) antagonist. NÚMERO DE CAS 159311-94-1

MMTCsc-201063MMTC is endogenous to the rat brain and to human urine. As a result of its antioxidant properties, MMTC may be neuroprotective. NÚMERO DE CAS 1210-56-6

Mosapride citratesc-203635Mosapride citrate is a selective SR-4 agonist and SR-3 antagonist. NÚMERO DE CAS 112885-42-4

N-Desmethyl Escitalopramsc-355637 NÚMERO DE CAS 144025-14-9

N-Methylquipazine dimaleatesc-203639N-Methylquipazine dimaleate is a tertiary amine analog of quipazine that is an agonist at SR (SR-3) with an affinity similar to that of quipazine, but which lacks affinity for central SR-1B. NÚMERO DE CAS 28614-26-8

NAN-190sc-201138NAN-190 is a SR-1A antagonist. NÚMERO DE CAS 115338-32-4

Naratriptan Hydrochloridesc-212362A triptan drug which is used for the treatment of migraine headaches. NÚMERO DE CAS 143388-64-1

NAS-181sc-203640NAS-181 is a selective SR-1B antagonist. It increases synthesis and metabolism of serotonin in the brain. NÚMERO DE CAS 205242-62-2

Nefazodone hydrochloridesc-203156Nefazodone hydrochloride is a SR-2A antagonist and inhibitor of serotonin and noradrenalin uptake. NÚMERO DE CAS 82752-99-6

NPEC-caged serotoninsc-359015NPEC ((N)-1-(2-nitrophenyl)ethyl) is a caged version of serotonin.

NPS ALX Compound 4a dihydrochloridesc-204134NPS ALX Compound 4a dihydrochloride is a competitive SR-6 antagonist displaying preference over other serotonin and D2 receptors. NÚMERO DE CAS 299433-10-6

Olanzapinesc-212469Olanzapine is a Serotonin 5-HT2A and D2DR inhibitor with anti-cholinergic activity. NÚMERO DE CAS 132539-06-1

Oleamidesc-358696Oleamide acts as an agonist at the CB1 cannabinoid receptor. Oleamide also appears to potentiate the actions of 5-HT on 5-HT2A and 2C receptors. NÚMERO DE CAS 301-02-0

Olanzapine Lactam Impuritysc-361832 NÚMERO DE CAS 1017241-34-7

Olanzapine Thiolactam Impuritysc-361833 NÚMERO DE CAS 1017241-36-9

Ondansetron hydrochloride dihydratesc-205778A serotonin-3 (5-HT3) receptor antagonists, used to prevent radiosurgery-induced nausea and vomiting, along with the modulation of alcohol intoxiccation. NÚMERO DE CAS 99614-01-4

Ondansetronsc-201127An antagonist of the serotonin 5-HT3 receptor. Demonstrates anti-emetic effects. NÚMERO DE CAS 99614-02-5

Ondansetron hydrochloridesc-204147Ondansetron hydrochloride is a selective SR-3 antagonist. It is antiemetic and preventis emesis induced by cytotoxic drugs and radiation. NÚMERO DE CAS 103639-04-9

Org 12962 HClsc-301505Org 12962 HCl is a selective SR-2C agonist. NÚMERO DE CAS 210821-63-9

p-MPPF dihydrochloridesc-301510This product is a selective 5-HT1A serotonin receptor antagonist. It has been found to be more potent than p-MPPI. NÚMERO DE CAS 223699-41-0

Paroxetine maleatesc-203658Highly potent and selective 5-HT uptake inhibitor that binds with high affinity to the serotonin transporter (Ki = 0.05 nM). NÚMERO DE CAS 64006-44-6

Pizotifen malatesc-201143A potent inhibitor of SR-2 receptor activity with potential embryotoxic effects in mice. Also been reported to have acute antagonistic affects on central muscarinic receptors. NÚMERO DE CAS 5189-11-7

PNU 109291sc-204203PNU 109291 is a potent and highly selective SR-1D agonist. NÚMERO DE CAS 187665-60-7

PNU 142633sc-204204PNU 142633 is a very selective, high affinity SR-1D agonist. NÚMERO DE CAS 187665-65-2

PNU 22394 hydrochloridesc-204851PNU 22394 hydrochloride is a potent SR-2C agonist and partial SR-2A/SR-2B agonist. NÚMERO DE CAS 15923-78-1

Quipazine dimaleatesc-201145Quipazine dimaleate is a studied SR-3 agonist with a certain amount of SR-2A subtype stimulation as well. NÚMERO DE CAS 5786-68-5

5
Hymenidinsc-202177Antagonist of serotonergic receptors. Inhibitor of CDK5/p25 (IC50=4µM) and GSK-3β (IC50=12µM). NÚMERO DE CAS 107019-95-4

R-96544 hydrochloridesc-204223R-96544 hydrochloride is a potent, selective SR-2 antagonist. NÚMERO DE CAS 167144-79-8

(R)-Citalopram Oxalatesc-219751A derivative of Citalopram and a potential selective inhibitor of 5-hydroxytryptamine transporter (serotonin). NÚMERO DE CAS 219861-53-7

Ramosetronsc-204873A serotonin 5HT3 receptor antagonist for the treatment of nausea and vomiting in post-operative cases. NÚMERO DE CAS 132036-88-5

Risperidonesc-204881Risperidone is an atypical antipsychotic agent that displays SR-2A inhibition. Risperidone also displays high inhibition of D2DR. NÚMERO DE CAS 106266-06-2

Ritanserinsc-203681Potent and long-acting 5-HT2 receptor antagonist (Ki = 0.39 nM). Anxiolytic in vivo. NÚMERO DE CAS 87051-43-2

Ro 04-6790sc-204238Ro 04-6790 is a potent and selective SR-6 antagonist. NÚMERO DE CAS 202466-68-0

Ro 60-0175 fumaratesc-204890Ro 60-0175 fumarate is a potent, selective SR-2 agonist. Ro 60-0175 shows selectivity for the SR-2C subtype. NÚMERO DE CAS 169675-09-6

RS 102221 hydrochloride hydratesc-361310RS 102221 hydrochloride hydrate has been reported to be a selective and potent SR-2C antagonist. NÚMERO DE CAS 185376-97-0 (free base)

RS 127445 hydrochloridesc-204244RS 127445 hydrochloride is a high affinity SR-2B antagonist (pKi = 9.5). It displays 1000-fold selectivity for SR-2B with good bioavailability. NÚMERO DE CAS 199864-87-4

RS 16566 dihydrochloridesc-361311RS 16566 dihydrochloride has been reported to be a high affinity ligand for the (R)-zacopride binding site. NÚMERO DE CAS 175729-69-8

RS 23597-190 hydrochloridesc-203243RS 23597-190 hydrochloride is a selective and competitive SR-4 antagonist. NÚMERO DE CAS 149719-06-2

RS 39604 hydrochloridesc-361313Has been shown to be a selective and potent SR-4 antagonist, with a relatively long half life. NÚMERO DE CAS 167710-87-4

RS 56812 hydrochloridesc-361315RS 56812 hydrochloride is an extremely potent and selective SR-3 partial agonist. NÚMERO DE CAS 143137-35-3

RS 67333 hydrochloridesc-361316RS 67333 hydrochloride is an extremely selective and potent SR-4 partial agonist. NÚMERO DE CAS 168986-60-5

RS 67506 hydrochloridesc-361317RS 67506 hydrochloride has been reported to be a selective and potent SR-4 partial agonist. NÚMERO DE CAS 168986-61-6

RU 24969 hemisuccinatesc-204896RU 24969 hemisuccinate is a potent SR-1A/SR-1B and moderate SR-2C agonist that may also release serotonin. NÚMERO DE CAS 107008-28-6

S 14506sc-205497S 14506 is a full, highly potent and selective SR-1A agonist. NÚMERO DE CAS 135721-98-1

(S)-Citalopram N-Oxidesc-212881A derivative of Citalopram and a potential selective inhibitor of the 5-hydroxytryptamine transporter (serotonin). NÚMERO DE CAS 917482-45-2

(S)-WAY 100135 dihydrochloridesc-361330(S)-WAY 100135 dihydrochloride has been shown to be a selective and potent SR-1B antagonist. NÚMERO DE CAS 133025-23-7 (free base)

Sarpogrelate hydrochloridesc-296371Sarpogrelate hydrochloride is a selective SR-2A antagonist NÚMERO DE CAS 135159-51-2

SB 200646 hydrochloridesc-361332SB 200646 hydrochloride is a SR-2C/SR-2B antagonist with a selective affinity for SR-1A. NÚMERO DE CAS 143797-63-1

SB 204741sc-224279SB 204741 is a potent, selective SR-2B antagonist. NÚMERO DE CAS 152239-46-8

SB 206553 hydrochloridesc-361334SB 206553 hydrochloride is a selective and potent SR-2B/SR-2C antagonist. NÚMERO DE CAS 158942-04-2

SB 216641 hydrochloridesc-361335SB 216641 hydrochloride has been reported as a selective SR-1B antagonist with approximately 25-fold selectivity over SR-1D and little or no affinity for a range of other receptor types. NÚMERO DE CAS 193611-67-5

SB 221284sc-224281SB 221284 is a potent, SR-2C and SR-2B antagonist. NÚMERO DE CAS 196965-14-7

SB 224289 hydrochloridesc-361336SB 224289 hydrochloride has been shown to be a selective SR-1B antagonist. SB 224289 hydrochloride has been found to display more than a 60 fold selectivity for SR-1B over other serotonin receptors. NÚMERO DE CAS 180083-23-2

SB 228357sc-361337SB 228357 is a SR-2C and SR-2B receptor antagonist. NÚMERO DE CAS 181629-93-6

SB 258585 hydrochloridesc-361339SB 258585 hydrochloride has been found to be a selective and potent SR-6 antagonist. This compound displays more than a 160-fold selectivity over other serotonin receptor subtypes. NÚMERO DE CAS 209480-63-7

SB 269970 hydrochloridesc-361342SB 269970 hydrochloride has been shown to be a selective and potent SR-7 antagonist. NÚMERO DE CAS 201038-74-6

SB 399885 hydrochloridesc-204264SB 399885 hydrochloride is a potent, brain penetrant, and orally active SR-6 antagonist. NÚMERO DE CAS 402713-80-8

SB-258585 dihydrochloridesc-3017895-HT6 serotonin receptor antagonist.

SB203186sc-203257Potent 5-HT4 serotonin receptor antagonist. NÚMERO DE CAS 207572-69-8

SDZ 205-557 hydrochloridesc-204273SDZ 205-557 hydrochloride acts as a SR-3 and SR-4 antagonist. NÚMERO DE CAS 137196-67-9

SDZ SER 082 fumaratesc-361356SDZ SER 082 fumarate has been reported to be a selectiveSR-2C/SR-2B antagonist with low affinity for SR-1A. NÚMERO DE CAS 141474-54-6

Serotonin • HClsc-201146Serotonin • HCl is a tryptophan amino acid neurotransmitter located in the central nervous system, which functions as an endogenous serotonin receptor agonist in a variety of biochemical processes. NÚMERO DE CAS 153-98-0

9
Spiperone hydrochloridesc-204293Spiperone hydrochloride is an analogue of Spiperone. Spiperone (sc-204293) is an SR-2A and selective D2DR inhibitor. NÚMERO DE CAS 749-02-0 (anhydrous)

Spiroxatrine (R 5188)sc-201148Spiroxatrine (R 5188) is a SR-1A antagonist. NÚMERO DE CAS 1054-88-2

SR 57227 hydrochloridesc-204301SR 57227 hydrochloride is a potent, selective SR-3 agonist. NÚMERO DE CAS 77145-61-0

ST 1936 oxalatesc-364625St 1936 oxalate is a potent and selective agonist of 5-HT6 receptor. ST 1936 oxalate also displays moderate affinity for human α2 adrenergic receptors. NÚMERO DE CAS 1210-81-7

Sumatriptan succinatesc-204314A selective 5-HT1 receptor agonist with specificity towards 5-HT1D, 5-HT1B and 5-HT1A, which is carried through cells via liposomes. NÚMERO DE CAS 103628-48-4

Tandospirone hydrochloridesc-204320Tandospirone hydrochloride is a SR-1A partial agonist that displays selectivity over SR-2, SR-1C, α1, α2, D1 and D2 receptors. NÚMERO DE CAS 87760-53-0

TCB-2sc-204325TCB-2 is a high affinity SR-2A agonist. NÚMERO DE CAS 912440-88-1

Tegaserod, Maleatesc-212993Tegaserod maleate is a SR-4 partial agonist. NÚMERO DE CAS 189188-57-6

Tianeptine sodium saltsc-204345A selective facilitator of 5-HT uptake in vitro and in vivo with reported inhibition of dopamine uptake. NÚMERO DE CAS 30123-17-2

4
Trimipramine Maleate Saltsc-213120A serotonin transport blocker that also blocks norepinephrine uptake. Categorized as a antidepressant. NÚMERO DE CAS 521-78-8

Tropanyl-3,5-dimethylbenzoatesc-204357Tropanyl-3,5-dimethylbenzoate is an antagonist of SR-3.

Tropisetron hydrochloridesc-204930Tropisetron hydrochloride is an orally active and potent SR-3 antagonist. It is alos a selective, partial agonist at a7 nicotinic receptors. NÚMERO DE CAS 105826-92-4

U 92016Asc-204363Selective 5-HT1A receptor agonist that displays high intrinsic activity (Ki values are 0.4, 7.7 and 36 nM for 5-HT1A, 5-HT1D and D2 receptors respectively and > 1000 nM for 5-HT2, D1, α1 and α2 receptors). Produces hypotension, hypothermia and 5-HT behavioral syndrome following p.o. administration. NÚMERO DE CAS 149654-41-1

VER-3323 hemifumarate saltsc-301968This product has been shown to be a 5-HT2C/ 5-HT2B serotonin receptor agonist.

WAY 161503 hydrochloridesc-204392WAY 161503 hydrochloride is a potent and selective SR-2C agonist. NÚMERO DE CAS 75704-24-4

WAY 629 hydrochloridesc-204393WAY 629 hydrochloride is a selective SR-2C agonist. NÚMERO DE CAS 57756-45-3

WAY-100135sc-364647WAY-100135 is a potent, selective 5-HT1A receptor antagonist (IC50 = 15 nM). It is selective over 5-HT1B, 1C, 2,α1, α2 and D2 receptors (IC50 > 1000 nM). NÚMERO DE CAS 149055-79-8

Xaliproden hydrochloridesc-203721Xaliproden hydrochloride is a full agonist at SR-1A. It increases motoneuron survival and promotes effects of NGF on neurite outgrowth in vitro. NÚMERO DE CAS 90494-79-4

Y-25130 Hydrochloridesc-201150Y-25130 is a potent and selective SR-3 antagonist with antiemetic effects. NÚMERO DE CAS 123040-16-4

3
Zacopride hydrochloridesc-203723Zacopride hydrochloride is a highly potent SR-3 antagonist and SR-4 agonist. NÚMERO DE CAS 90182-92-6

Zimelidine dihydrochloridesc-203725Selective 5-HT uptake inhibitor; selective over noradrenalin and dopamine uptake (IC50 values are 0.33, 8.2 and 12 μM respectively). Modulates nociception and induces hyperglycemia in vivo, and is an orally active antidepressant. NÚMERO DE CAS 56775-88-3

Ziprasidone hydrochloride monohydratesc-204419Ziprasidone hydrochloride monohydrate is an atypical antipsychotic that displays combined SR-2A and D2DR inhibition. NÚMERO DE CAS 138982-67-9

Octoclothepin maleate saltsc-253215Octoclothepin maleate salt is an SR-2A inhibitor as well as a D2DR inhibitor. NÚMERO DE CAS 4789-68-8

WAY-100635 maleate saltsc-264493WAY-100635 maleate salt is a potent, selective and high affinity SR-2B antagonist. NÚMERO DE CAS 634908-75-1

Duloxetine Hydrochloridesc-207599A dual serotonin and norepinephrine reuptake inhibitor (SNRI) that is used in the treatment of stress urinary incontinence, as well as depression. NÚMERO DE CAS 136434-34-9

Agomelatinesc-207266This compound is a melatoninergic agonist and selective antagonist of 5-HT2C receptors. It has been shown to be active in several animal models of depression. NÚMERO DE CAS 138112-76-2

Trazodone Hydrochloridesc-213097An Antidepressant. NÚMERO DE CAS 25332-39-2

CP 135807sc-361155CP 135807 is a selective receptor agonist of SR-1D. CP 135807 has been shown to dose-dependently lower the extracellular serotonin concentration. NÚMERO DE CAS 151272-90-1

L-703,664 succinatesc-361225L-703,664 succinate has been shown to be a SR-1D agonist with selectivity over other receptors. NÚMERO DE CAS 144776-01-2