Inhibitors - Other

• 1-(5-Isoquinolinesulfonyl)-3-methylpiperazine
  A less potent inhibitor of protein kinase C than H-7.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208552	84477-73-6	C14H17N3O2S	5 g

• 1-(8-Chloro-5-isoquinolinesulfonyl)piperazine, Dihydrochloride
  Inhibits both Ca²⁺ dependent myosin phosphorylation by protein kinase C and MLC-Kinase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206110	355115-40-1	C13H16Cl3N3O2S	10 mg

• 1-Allylcyclopropane-1-sulfonyl Chloride
  A MEK inhibitor. Useful in the treatment of cancer and other hyperproliferative diseases.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206127	923032-59-1	C6H9ClO2S	50 mg

• 1-Benzyl-4-cyano-4-phenylpiperidine
  A piperidine derivative as calcium channel blockers.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208614	56243-25-5	C19H20N2	1 g

• 1-Hydroxycyclopropanecarboxylic Acid Phosphate, Biscyclohexylamine Salt
  A potent, reversible inhibitor of enzymes utilizing phosphoenolpyruvate (PEP), such as phosphoenolpyruvate carboxylase which catalyzes the carboxylation of PEP to produce oxaloacetate.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-213339	94017-79-5	C16H35N2O6P	10 mg

• 1-Methyl-D-tryptophan
  An inhibitor of IDO and IDO2, with selectivity for IDO2. Shown to reverse IDO-mediated suppression of immune response.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200313	110117-83-4	C12H14N2O2	50 mg

• 1-O-Acetyl-2,3,5-tri-O-benzoyl-α,β-D-ribofuranose
  This compound inhibits neutrophil-keyhole limpet hemocyanin adhesion

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206190	14215-97-5	C28H24O9	2.5 g

• 1-Thio-β-D-glucose tetraacetate
  Inhibits the Maillard reaction between glucose and glycine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205567	19879-84-6	C14H20O9S	250 mg/1 g

• 1,2-Isopropylidene Swainsonine

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-213452	N/A	C11H19NO3	1 mg

• 1,4-Dichloro-7-isoquinolinesulfonyl Chloride
  Intermediate of isoquinolinylguanidines as urokinase inhibitors.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206252	223671-80-5	C9H4Cl3NO2S	100 mg

• 1,4-Dideoxy-1,4-imino-D-arabinitol HCl
  A glycogen phosphorylase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220553	100937-52-8	C5H11NO3•HCl	10 mg/25 mg

• 1,5-Bis(4-Allyldimethylammoniumphenyl)pentan-3-one, Dibromide
  A selective inhibitor of acetylcholinesterase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206257	402-40-4	C27H38Br2N2O	100 mg

• 2-(5,5-Dimethyl-1,3,2-dioxaborinan-2-yl)benzoic Acid Ethyl Ester
  Boronic acid ester derivative that inhibits hormone-sensitive lipase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206328	346656-34-6	C14H19BO4	1 g

• 2-Acetamido-2-deoxy-6-O-(β-D-galactopyranosyl)-D-glucopyranose
  An inhibitor of lectins.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216163	50787-10-5	C14H25NO11	1 mg

• 2-Amino-4-isopropylamino-6-chlorotriazine
  Has been shown to inhibit the growth of plants.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206379	6190-65-4	C6H10ClN5	500 mg

• 2-Chloro-4-nitrophenyl-β-D-lactoside
  A substrate used for the determination of cellobiohydrolase I.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220712	120583-41-7	C18H24ClNO13	10 mg/50 mg

• 2-Fluoropalmitic acid
  Inhibitor of palmityl-CoA biosynthesis resulting in blockade of protein palmitoylation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202881	89270-22-4	C16H31FO2	1 mg/5 mg

• 2-Hexynyl-5’-N-ethylcarboxamidoadenosine
  This compound possesses high affinity to adenosine (A1 & A2) receptors, which inhibits radioligands from binding to these sites.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206449	141018-30-6	C18H24N6O4	5 mg

• 2-Hydroxymyristic acid
  An acid that has the capability to distinguish between myristoylation and palmitoylation, and is therefore able to inhibit protein myristoylation in cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202401	2507-55-3	C14H28O3	25 mg

• 2-Iodo-5'-ethylcarboxamido-2',3'-O-isopropylidineadenosine

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216221	162936-24-5	C15H19IN6O4	10 mg

• 2-n-Butylthiophene
  Inhibitor of DMH-induced aberrant crypt formation in colon.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204617	1455-20-5	C8H12S	5 g/10 g

• 2-TEDC
  Potent inhibitor of 5-, 12-, and 15-lipoxygenase (IC₅₀ values are 0.09, 0.013 and 0.5 μM respectively).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203772	132465-10-2	C16H13NO4S	10 mg/50 mg

• 2,3-Butanedione 2-Monoxime
  Skeletal and cardiac muscle contraction inhibitor. Broad reversible inhibitor of myosin ATPase in eukaryotes. Shown to induce Ca²⁺ release from canine cardiac SR.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203774	57-71-6	C4H7NO2	500 mg

• 2,4-Dibenzyl-5-oxothiadiazolidine-3-thione
  A highly conserved, widely found and expressed Ser/Thr protein kinase that is active in the signal transduction cascades of multiple cellular processes. It is an analog of oxothadiazolidine-3-thione.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-213994	72966-20-2	C16H14N2OS2	5 mg

• 2,4-Diethylpyridine dicarboxylate

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202405	41438-38-4	C11H13NO4	10 mg/25 mg

• 2,4-Thiazolidinedione
  Inhibitor of enzyme.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216281	2295-31-0	C3H3NO2S	50 g

• 2,6-Anhydro-3-deoxy-D-glycero-D-galacto-non-2-enoic Acid
  Potential inhibitor of virus sialidase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206536	188854-96-8	C9H14O8	5 mg

• 2'-(N-Methylanthraniloyl)guanosine 3',5'-Cyclicmonophosphate, Sodium Salt
  Blue fluorescent derivative of cGMP, a useful substrate in the assay of cyclic nucleotide phosphodiesterases. Has been shown to inhibit calmodulin-dependent activation of cyclic nucleotide phosphodiestereases by peptide segments of HIV envelope glycoproteins.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206545	221905-46-0	C18H18N6NaO8P	5 mg

• 2',3'-Dideoxyadenosine
  Inhibitor of adenylate cyclase. Useful tool in antiviral and anticancer studies. Blocks viral reverse transcription from RNA to DNA. Inhibitor of adenosine deaminase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202406	4097-22-7	C10H13N5O2	1 mg/5 mg

• 2',4',6'-Trihydroxy-4-nitrodihydrochalcone

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216314	82628-82-8	C15H13NO6	10 mg

• 2',5'-Dideoxyadenosine 3'-monophosphate
  A non-cell-permeable, potent inhibitor of adenylyl cyclase. It is a precursor to 2',5'-Dideoxyadenosine 3'-triphosphate). IC₅₀ = 460 nM in detergent-dispersed rat brain preparation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214084	121878-11-3	C10H14N5O5P	5 mg

• (2S)-(+)-Amino-5-iodoacetamidopentanoic acid
  An irreversible inhibitor of ornithine decarboxylase and arginase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202409	35748-65-3	C7H13N2O3I	5 mg/25 mg

• 3-(N-Hydroxyamino)propyl Phosphonate

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-209484	66508-11-0	C3H10NO4P	25 mg

• 3-Amino-1,2,4-triazole
  An irreversible inhibitor of catalase activity. Inhibits imidazoleglycerol-phosphate dehydratase activity and histidine biosynthesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202016	61-82-5	C2H4N4	1 g

• 3-Keto-N-aminoethyl-N'-aminocaproyldihydrocinnamoyl Cyclopamine
  Cyclopamine demonstrates teratogenic properties and has been shown to reverse effects of oncogenic mutations in Smoothened and Patched. The KAAD derivative shows 10-20 fold higher potency than cyclopamine in inhibition of β-Galactosidase expression.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206652	306387-90-6	C44H63N3O4	250 µg

• 3-Nitropropionic acid
  A potent, irreversible inhibitor of mitochondrial complex II enzyme, which causes dysfunction and oxidative stress in mitochondria.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214148	504-88-1	C3H5NO4	1 g/10 g

• 3-O-Methyl-N-acetyl-D-glucosamine
  An analog of N-acetyl-D-glucosamine shown to inhibit N-acetylglucosamine kinase and N-acetylmannosamine kinase, without inhibiting glucokinase - potentially useful for accurate assay of glucokinase activity in pancreatic islets and liver tissues.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202886	94825-74-8	C9H17NO6	5 mg

• 3-Phenylpropyl isothiocyanate
  Synthetic phenyl isothiocyanate that has been found to induce Phase II detoxifying enzymes. Also inhibits chemically induced carcinogenesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204620	2627-27-2	C10H11NS	5 g/10 g

• 3,4-Dihydroxyphenyl Ethanol
  Inhibits 5-lipoxygenase and 12-lipoxygenase. Scavenges reactive oxygen species and protects against oxidative damage. Increases cytosolic Ca²⁺ levels.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202887	10597-60-1	C8H10O3	10 mg

• 3,7-Dimethyl-8-(p-sulfonamidophenyl)xanthine
  A weak water soluble A2 -adenosine receptor antagonist.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-209733	149981-21-5	C13H13N5O4S	50 mg

• 3,7-Dimethyl-8-p-sulfophenylxanthine
  A weak water soluble A2 -adenosine receptor antagonist.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-209734	149981-20-4	C13H12N4O5S	25 mg

• 3'-Deoxy-3'-fluorothymidine-5'-monophosphate Disodium Salt
  A fluoronated analog of thymidine-5'-O-monophosphate. A substrate of Mycobacterium tuberculosis thymidylate kinase with a Km of 30 μM.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216619	N/A	C10H12FN2Na2O7P	1 mg

• 3',4',5',5,7-Pentamethoxyflavanone

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216630	479672-30-5	C20H22O7	10 mg

• (3R,5S)-Fluvastatin Sodium Salt
  An anti-lipemic synthetic HMG-CoA reductase inhibitor that contains residual sodium chloride which is quantified on the certificate of analysis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206732	94061-80-0	C24H25FNNaO4	1 mg

• (3S,5R) Fluvastatin Sodium Salt
  Antilipemic. A synthetic HMG-CoA reductase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206738	155229-76-8	C24H25FNNaO4	1 mg

• 3α-Mannobiose
  Postulated to be the major antigenic determinant of yeast in cell walls. An inhibitor of fimbrial lectins from enterobacteria.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216644	23745-85-9	C12H22O11	1 mg/5 mg

• 4-[(1-oxo-7-phenylheptyl)amino]-(4R)-octanoic acid
  Phospholipase A2 (PLA2) catalyzes the hydrolysis of fatty acids at the sn-2 position of glycerophospholipids, liberating arachidonic acid for subsequent eicosanoid synthesis. Three primary types of PLA2 exist: secretory (sPLA2), calcium-independent cytosolic (iPLA2), and calcium-dependent cytosolic (cPLA2). Of these three enzymes, cPLA2 is the rate-limiting stimulus for release of arachidonic acid whereas sPLA2 amplifies the action of cPLA2 and regulates foam cell formation and phagocytosis. This chemical, a simple amide based on (R)-α-norleucine, is a selective and potent inhibitor of sPLA2. It exhibits 95% inhibition (XI(50) = 0.003) of sPLA2 at 0.091 mole fraction without affecting the activities of cPLA2 or iPLA2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-223602	1101136-50-8	C21H33NO3	1 mg/5 mg

• 4-Aminobenzoyl-Gly-Pro-D-Leu-D-Ala hydroxamic acid
  This compound inhibits collagenase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214226	124168-73-6	C23H34N6O6	5 mg

• 4-Chloro-1H-pyrazolo[3,4-d]pyrimidine
  This has a SK channel blocker effect.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216799	5399-92-8	C5H3ClN4	250 mg

• 4-Chloro-DL-phenylalanine methyl ester hydrochloride
  Tryptophan hydroxylase inhibitor. This can cross the blood brain barrier better than p-chlorophenylalanine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-238813	14173-40-1	C10H12ClNO2 ·HCl	1 g/5 g

• 4-Chlorophenylguanidine hydrochloride
  Potent and specific inhibitor of urokinase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203474	14279-91-5	C7H8CIN3 HCl	100 mg

• 4-Formylpiperidine-1-carboxylic Acid tert-Butyl Ester
  Intermediate for polycyclic indazole derivatives which are ERK inhibitors.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216846	137076-22-3	C11H19NO3	100 mg

• 4-Hydroxynonenal
  Aldehydic product formed by peroxidation of ω-6-unsaturated fatty acids. Irreversibly inhibits Na⁺-K⁺-ATPase activity (IC₅₀ = 120 µM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202019	75899-68-2	C9H16O2	1 mg

• 4-Methylpyrazole hydrochloride
  Alcohol dehydrogenase inhibitor. Antidote in methanol and ethylene glycol poisoning.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214254	56010-88-9	C4H6N2•HCl	100 mg/500 mg

• 4-Oxatetradecanoic acid
  Analog of myristate with same chain length but a polar oxygen atom incorporated in place of a methylene group, resulting in reduced hydrophobicity. Inhibits HIV replication.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202422	7420-16-8	C13H26O3	10 mg

• (4-Sulfamoylphenyl)hydrazine Hydrochloride

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217009	4392-54-5	C6H10ClN3O2S	1 g

• 4,5,6,7-Tetrabromobenzimidazole
  A selective ATP-competitive inhibitor of protein kinase CK2 from such divergent sources as yeast, rat liver, Neurospora erassa and Candida tropicalis, with Ki values in the range of 0.5-1uM. It is virtually inactive against PKA, PKC, and a very weak

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217031	577779-57-8	C7H2Br4N2	25 mg

• 4'-Demethylepipodophyllotoxin
  A potent inhibitor of microtubule assembly.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206950	6559-91-7	C21H20O8	10 mg

• 4'-Deoxyphlorizin
  Inhibitor of the glucose transport system.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206951	4319-68-0	C21H24O9	1 g

• 4'-Hydroxy Atomoxetine
  A metabolite of Tomoxetine (Atomoxetine, LY 139603).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217050	435293-66-6	C17H21NO2	1 mg

• 4'-Hydroxy Atomoxetine β-D-Glucuronide
  A metabolite of Tomoxetine (Atomoxetine, LY 139603).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-210189	540729-08-6	C23H29NO8	1 mg

• 4'-Hydroxy Atomoxetine β-D-Glucuronide-d3
  A labeled metabolite of Tomoxetine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217051	N/A	C23H26D3NO8	5 mg

• 4'-Hydroxy Atomoxetine-d3
  A labeled metabolite of Tomoxetine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217052	N/A	C17H18D3NO2	1 mg

• 4E1RCat

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361085	328998-25-0	C28H18N2O6	10 mg/50 mg

• 5-Cyanoindole
  Inhibitor of enzyme.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217174	15861-24-2	C9H6N2	1 g

• 5-epi-Isofagomine
  Strongly and selectively inhibits β-Glucosidase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207026	202979-51-9	C6H13NO3	5 mg

• 5-Ethynyl-1-(β-D-ribofuranosyl)-imidazo-4-carbonitrile

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217178	126004-13-5	C11H11N3O4	5 mg

• 5-Iodo-1-(2',3',5'-tri-O-acetyl-β-D-ribofuranosyl)-imidazo-4-carbonitrile

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217209	N/A	C15H16IN3O7	5 mg

• 5-Iodonaphthalene-1-sulfonylchloride
  A synthetic intermediate.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-210352	110448-35-6	C10H6ClISO2	100 mg

• 6-Aminonicotinamide
  An inhibitor of the NADP+-dependent enzyme, 6-phosphogluconate dehydrogenase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-278446	329-89-5	C6H7N3O	1 g/5 g

• 5HPP-33

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214349	105624-86-0	C20H21NO3	5 mg/25 mg

• 6-ECDCA
  A novel derivative of cholic acid which acts as a potent and selective FXR agonist (EC₅₀= 99nM) displaying anticholeretic activity in an in vivo rat model of cholestasis. It not only inhibits vascular smooth muscle cell inflammation and migration but also promotes adipocyte differentiation and regulates adipose cell function in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-280538	459789-99-2	C26H44O4	5 mg/25 mg

• 6-Methoxypurine
  Phosphoribosyltransferase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-291383	1074-89-1	N/A	250 mg/1 g

• 6-Nitroindazole
  Anticonvulsant.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217371	7597-18-4	C7H5N3O2	25 g

• 6,7-Dihydroxyswainsonine
  This is a Swainsonine analogue which inhibits a-mannosidase with 20-to 100-fold less activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217387	144367-16-8	C8H15NO5	1 mg

• 6,7-Dimethyltetrahydropterin (hydrochloride)
  A noncompetitive inhibitor of GTP cyclohydrolase I exhibiting an IC₅₀ of 76-112 µM.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205161	167423-51-0	C8H14N5OCl	10 mg/50 mg

• 6'-Carboxy Simvastatin
  A HMG-COA reductase inhibitor. Useful as anticholesteramic.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207136	125206-31-7	C25H36O7	2.5 mg

• (-)-(6S)-2,6-Diamino-4,5,6,7-tetrahydrobenzothiazole
  A (S)-Pramipexole intermediate. Acts as a dopamine autoreceptor agonist.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217401	106092-09-5	C7H11N3S	100 mg

• 6-Bromoandrostenedione
  Androstenedione analog, an aromatase inhibitor

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207138	38632-00-7	C19H25BrO2	10 mg

• 7-(Trifluoromethyl)1H-indole-2,3-dione
  An indole derivative. Acts as an inhibitor of COX-1, COX-2, and Œ≤-catenin. Useful in the treatment of diseases such as lung cancer, diabetes and Alzheimerís disease.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217411	391-12-8	C9H4F3NO2	100 mg

• 7-Epi 10-Desacetyl Paclitaxel
  Paclitaxel impurity and Paclitaxel related compound B. The compound has been isolated from Taxus yunnanensis and shown to have potential growth inhibitory activities against human cancer cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207169	78454-17-8	C45H49NO13	2.5 mg

• 7-O-[2-(1,3-Dioxanyl)ethyl]daidzein
  A potent inhibitor of aldehyde dehydrogenase isozyme (ALDH2) and MOA.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217465	N/A	C21H20O6	10 mg

• 7-O-Ethyldaidzein
  A potent inhibitor of aldehyde dehydrogenase isozyme (ALDH2) and MOA,

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207181	146698-96-6	C17H14O4	10 mg

• 7-O-w-Bromopropyldaidzein
  Potent MOA and aldehyde dehydrogenase isozyme (ALDH2) inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207182	309252-38-8	C18H15BrO4	10 mg

• 9-Cyclopentyladenine monomethanesulfonate
  A stable, cell-permeable, non-competitive adenylyl cyclase inhibitor that targets the P-site domain. In detergent-dispersed rat brain preparation, IC₅₀ = 100 µM

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214435	189639-09-6	C11H17N5O3S	5 mg/25 mg

• A 205804
  Selective inhibitor of E-selectin and ICAM-1 expression (IC₅₀ values are 20, 25 and > 1000 nM for TNF-α-induced E-selectin, ICAM-1 and VCAM-1 expression respectively). Effective inhibitor of cell-cell adhesion in an in vitro flow experiment.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203484	251992-66-2	C15H12N2OS2	10 mg/50 mg

• 10-DEBC hydrochloride
  Selective inhibitor of Akt/PKB. Inhibits IGF-1-stimulated phosphorylation and activation of Akt (complete inhibition at 2.5 μM), suppressing downstream activation of mTOR, p70 S6 kinase and S6 ribosomal protein. Shows no activity at PDK1, SGK1 or PI 3-kinase. Inhibits cell growth (IC₅₀ ~ 2-6 μM) and induces apoptosis in rhabdomyosarcoma cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203459	201788-90-1	C20H25ClN2O ·HCl	10 mg/50 mg

• 10Z-Hymenialdisine

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-360987	82005-12-7	C11H10BrN5O2	500 µg

• A 286982

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-362705	280749-17-9	C24H27N3O4S	10 mg/50 mg

• 13-cis-Retinoic acid
  A vitamin A analog that inhibits cell proliferation and induces cell differentiation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205568	4759-48-2	C20H28O2	100 mg/250 mg

• A 839977

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-362707	870061-27-1	C19H14Cl2N6O	10 mg/50 mg

• 17-AAG
  17-AAG is a less toxic and more stable analog of geldanamycin. It is an HSP90 inhibitor that displays a 100-fold higher affinity for HSP90 derived from tumor cells compared to HSP90 from normal cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200641	75747-14-7	C31H43N3O8	1 mg

• 17β-hydroxy Wortmannin

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-358740	N/A	C23H26O8	500 µg/1mg

• 19,20-Epoxycytochalasin C
  19,20-Epoxycytochalasin C was identified in fungal extracts and like other cytochalasins is cytotoxic.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202006	189351-79-9	C30H37NO7	1 mg

• 19,20-Epoxycytochalasin D
  Data suggests the presence of the epoxide renders this metabolite more active than cytochalasin D in inhibition of tumor cell growth in vitro.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202007	191349-10-7	C30H37NO7	1 mg

• A 922500
  Diacyl glycerolacyltransferase 1 (DGAT-1) inhibitor (IC₅₀ values are 7 and 24 nM at human and mouse DGAT-1 respectively) that is devoid of activity at DGAT-2, ACAT1 or ACAT2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203793	959122-11-3	C26H24N2O4	10 mg

• A-803467
  A-803467 is a potent and selective inhibitor of the TTX-resistant voltage-gated sodium channel Nav1.8 which is preferentially expressed on sensory neurons.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201068	944261-79-4	C19H16ClNO4	10 mg/50 mg

• AAF-CMK
  Serine protease inhibitor which irreversibly inhibits tripeptidyl peptidase II (TPPII), a giant protease which may substitute for some proteasome functions1, nd reversibly inhibits TPPI2. Shows only marginal inhibition of the chymotrypsin-like activity of the proteasome.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205591	184901-82-4	C16H22ClN3O3•C2HF3O2	5 mg/25 mg

• Abacavir hydrochloride

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-358732	136470-78-5 (non-salt)	C14H18N6O•HCl	1 g/5 g

• Abacavir Sulfate
  A nucleoside reverse transcriptase inhibitor (NRTI).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207238	188062-50-2	C28H38N12O6S	5 mg/25 mg

• Abiraterone Acetate
  Abiraterone acetate has seen to be a novel steroidal inhibitor of C17,20 lyase. It has been observed to decrease the DHEA, androstenedione and testosterone.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207240	154229-18-2	C26H33NO2	5 mg

• AC 45594
  Selective inverse agonist at the orphan nuclear receptor steroidogenic factor-1 (SF-1) (IC₅₀= 50-100 nM). Displays no activity at estrogen, LRH-1, ROR, ERR or Nurr receptors. Inhibits SFRE-mediated transcription.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203798	13037-86-0	C13H20O2	1 g/5 g

• Acenaphthenequinone
  A quinoid polycyclic aromatic hydrocarbon, which acts as a redox-active compound. This compound is used to study ROS induced damage to lung tissue.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-239180	82-86-0	C12H6O2	25 g

• Acetazolamide
  Carbonic anhydrase inhibitor that increases cerebral blood flow.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214461	59-66-5	C4H6N4O3S2	10 g/25 g

• Acetildenafil
  A designer drug which acts as a phosphodiesterase inhibitor. Also a structural analog of Sidenafil (Viagra).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207250	831217-01-7	C25H34N6O3	2.5 mg

• Acetohydroxamic Acid
  A inhibitor of urease.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207251	546-88-3	C2H5NO2	10 g

• AdaAhx3L3VS
  A potent, covalent, cell-permeable, irreversible inhibitor of chymotrypsin-like, trypsin-like, and PGPH activities of the 20S proteasome.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221211	389064-25-9	C50H88N6O8S	250 µg

• ADAMTS-5 Inhibitor
  A thioxothiazolidinone compound that possesses a Zn²⁺-chelating structural motif and acts as an ADAMTS-5 (aggrecanase-2) inhibitor (IC₅₀ = 1.1 µM) with ~40-fold selectivity over ADAMTS-4 (aggrecanase-1).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221212	N/A	C16H11ClF3N3OS3	5 mg

• Adenylyl Cyclase Type V Inhibitor, NKY80
  A cell-permeable quinazolinone containing a non-nucleoside compound that acts as a potent, selective inhibitor of adenylyl cyclase (AC) type V isoform (IC₅₀ = 8.3 µM, 132 µM and 1.7 mM for type V, III and II, respectively) in the presence of Gsα GTPγS-Forskolin. Displays ~210-fold greater selectivity for type V over the type II isoform. The inhibition is non-competitive with respect to ATP and Forskolin. Regulates the AC catalytic activity in heart and lung tissues.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221217	N/A	C12H11N3O2	5 mg/25 mg

• AG 1433 HCl
  A specific and potent inhibitor of PDGF-β receptor kinase (IC5₅₀ = 5.0 µM) and of KDR/Flk-1/VEGF Receptor 2 (IC₅₀ = 9.3 µM). Acts also as angiogenesis inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221220	N/A	C16H14N2O2··HCl	5 mg

• Agistatine B
  A tricyclic analog of agistatine A, which has been described as an inhibitor of cholesterol biosynthesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202918	144096-46-8	C11H18O4	1 mg/5 mg

• Agistatine D
  Analog of agistatine A, which has been described as an inhibitor of cholesterol biosynthesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202919	144096-47-9	C11H14O4	1 mg/5 mg

• AICAR-Tri-O-Acetate

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217591	23274-21-7	C15H20N4O8	10 mg

• Akt Inhibitor VIII, Isozyme-Selective, Akti-1/2
  A cell-permeable quinoxaline compound that potently and selectively inhibits Akt1, Akt2 and Akt3 activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202048	612847-09-3	C34H29N7O	1 mg/5 mg

• Aloeresin A
  An inhibitor of α-glucosidase that can be converted to p-couramic and aloesin.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202922	74545-79-2	C28H28O11	1 mg

• ALX 5407 hydrochloride

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361102	571147-18-7	C24H24FNO3.HCl	10 mg

• AM 1172
  Potent and selective inhibitor of anandamide uptake, resistant to fatty acid amide hydrolase (FAAH) hydrolysis. Metabolically stable “reversed” isomer of AM 404

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202456	251908-92-6	C27H39NO2	1 mg/5 mg

• Amastatin hydrochloride
  A slow, tight binding competitive inhibitor of human serum aminopeptidase A, human serum aminopeptidase M, pig kidney leucine aminopeptidase, leucine aminopeptidase and tyrosine aminopeptidase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202051	100938-10-1	C21H38N4O8 ·HCl	1 mg/5 mg

• AMD3100 octahydrochloride hydrate
  A selective bicyclam derivative which functions as a stem cell mobiliser via blocking the CXCR4 chemokine receptor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-252367	155148-31-5 (anhydrous)	C28H54N8•8HCl•xH2O	5 mg

• Aminoglutethimide
  Inhibits aromatase and adrenal steroidogenesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207280	125-84-8	C13H16N2O2	1 g

• Aminophylline
  A non-selective phosphodiesterase (PDE) inhibitor which is commonly used as an antiepileptic drug.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-252368	317-34-0	C7H8N4O2•0.5C2H8N2	25 g

• Aminopterin
  Folic acid antagonist. Potent dihydrofolate reductase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202461	54-62-6	C19H20N8O5	10 mg/50 mg

• Anacardic Acid
  An effective inhibitor of the activities of p300 and p300/CBP associated factor histone acetyltransferase, HAT-dependent transcription, and SUMOylation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202463	16611-84-0	C22H36O3	5 mg/25 mg

• Anastrozole
  An aromatase inhibitor. Used as an antineoplastic.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217647	120511-73-1	C17H19N5	10 mg

• Androst-4-ene-3,6,17-trione
  An aromatase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207292	2243-06-3	C19H24O3	10 mg

• Anisindione

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-291902	117-37-3	C16H12O3	1 g/25 g

• Anisomycin
  Inhibits peptidyl transferase activity; activates JNK/SAPK and MAP Kinase pathways including phosphorylation of c-Jun, p54, ATF-2, ERK, caldesmon, IRS-1, and IRS-2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-3524	22862-76-6	C14H19NO4	5 mg/50 mg

• Antibiotic LL Z1640-2
  A signal-specific inhibitor of the JNK/p38 pathways and a member of the resorcylic acid lactone (RAL) family that also irreversibly inhibits TAK1.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202055	66018-38-0	C19H22O7	1 mg/5 mg

• ARL 67156 trisodium salt
  A newly synthesized analogue of ATP which functions as a selective ecto-ATPase inhibitor. In addition, studies suggest that ARL 67156 trisodium salt also acts as a weak antagonist for the purinoceptors P2X and P2T and as an agonist for P2u.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203521	160928-38-1	C15H21Br2N5O12P3 ·3Na	10 mg

• AS 101
  Immunomodulator; inhibits IL-10 synthesis and potentiates IL-1a, IL-2 and TNFa release

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203825	106566-58-9	C2H4Cl3O2Te ·NH4	10 mg/50 mg

• (+)-AS 115
  A potent and selective inactivator of KIAA1363, displaying an IC₅₀n value of 150 nM when tested as a racemic mixture in the SK0V-3 cell line. The activities of the individual enantiomers have not been determined.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205216	926657-43-4	C21H32FNO4	100 µg/500 µg

• (−)-AS 115
  KIAA1363 is a 2-acetyl monoacylglyceryl ether (MAGE) hydrolase which is upregulated in aggressive cancers from an array of tissues. The enzyme catalyzes the hydrolysis of the 2-acetyl MAGE to MAGE and serves as a central enzyme in the PAF and LPA signaling network. AS 115 is a potent and selective inactivator of KIAA1363, displaying an IC₅₀ value of 150 nM when tested as a racemic mixture in the invasive ovarian cancer cell line SK0V-3.2 Treatment of SKOV-3 cells with 10 µM AS-115 for 4 hours significantly reduced the formation of MAGE, alkyl-lysophosphatidylcholine, and alkyl-lysophosphatidic acid. The activity of the individual enantiomers of AS 115, i.e. (+)-AS 115 and (−)-AS 115, has not been determined.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221270	926657-43-4	C21H32FNO4	100 µg/500 µg

• Atazanavir
  An azapeptide protease inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207305	198904-31-3	C38H52N6O7	5 mg

• Atomoxetine-d3, Hydrochloride
  A labeled analogue of Tomoxetine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217670	N/A	C17H18D3NO.HCl	1 mg

• Aurintricarboxylic acid ammonium salt
  Aluminum reagent that readily polymerizes in solution (aq), producing a free radical that inhibits protein-nucleic acid interactions. Inhibits ribonuclease and topoisomerase Il2 through the prevention of enzyme-nucleic acid binding. Stimulates tyrosine phosphorylation and inhibits apoptosis in many cell types.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-210849	569-58-4	C22H14O9 ·3NH3	25 g/100 g

• Autophagy Inhibitor, 3-MA
  Cell-permeable autophagic sequestration blocker that protects cerebellar granule cells from apoptosis post serum/potassium deprivation. Displays distinctly different properties from LY 294002 (sc-201426) and Wortmannin (sc-3505).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205596	5142-23-4	C6H7N5	50 mg

• AX 048
  A PLA₂ and PGE₂ inhibitor.Contains a specific affinity for group IVA cPLA₂ which moderates antihyperalgesia effects.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-358797	873079-69-7	C22H41NO4	500 µg/1mg

• Axitinib
  A tyrosine kinase inhibitor that is used in cancer therapy.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217679	319460-85-0	C22H18N4OS	10 mg

• Azamulin
  A highly selective human CYP3A4 inhibitor and a mutilin derivative.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207310	76530-44-4	C24H38N4O4S	5 mg

• B-3530
  Inhibits cathepsins B, L, and S with similar kinetics. The diiodinated compound reacts irreversibly with cathepsins B and L, but not with cathepsin S and is able to penetrate cells and react with active enzymes within the cells. Often abbreviated DMK. Peptidyl diazomethyl ketones are specific inactivators of thiol proteinases.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-291922	N/A	C28H26N4O5	10 mg/50 mg

• AT-56
  A selective, competitive, and highly bioavailable inhibitor of L-PGDS with a K_i value of 75 µM.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-344899	162640-98-4	C25H27N5	1mg/5mg

• Bafilomycin A1
  A potent and selective inhibitor of vacuolar-type (v-type) H⁺ ATPase and belongs to a class of membrane ATPase inhibitors.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201550	88899-55-2	C35H58O9	100 µg/1 mg

• Bafilomycin D
  Shares the same mode of action as bafilomycin A1. Bafilomycin D contains the ring opened side chain and is a much more stable analogue of bafilomycin A1.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202074	98813-13-9	C35H56O8	1 mg

• BAG 956
  A dual PDK1 and class I PI3K inhibitor (IC50 values are 245, 56, 446, 35 and 117 nM for PDK1 and PI3K p110 -α, -β, -δ, and -γ respectively). Has been shown to inhibit cellular AKT phosphorylation at Thr308. Also blocks cell proliferation, causing arrest in G1 phase of the cell cycle. Slows tumor progression in mouse xenograft models.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-291923	853910-02-8	C28H21N5•xH2O	10 mg/50 mg

• Bambuterol Hydrochloride
  A bronchodilator. It inhibits plasma cholinesterase during metabolism prolongs suxamethonium-induced neuromuscular blockade.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205598	81732-46-9	C18H29N3O5 ·HCl	500 mg/1 g

• Bax channel blocker
  Potent inhibitor of Bax-mediated mitochondrial cytochrome c release (IC₅₀ = 0.52 μM). Suggested to inhibit Bax channel formation/activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203524	335165-68-9	C19H21Br2N3O ·2HCl	10 mg/50 mg

• BAY 73-6691
  Characterized in vitro as the first potent and selective inhibitor of phosphodiesterase 9 (PDE9).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-252407	794568-92-6	C15H12ClF3N4O	5 mg

• BAY 61-3606 hydrochloride hydrate

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-360240	N/A	C20H18N6O3•xHCl•yH2O	5 mg/25 mg

• BAY-60-7550
  Antagonizes oxidative stress-induced anxiety-like behavioral effects in mice by increasing cGMP signaling.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205219	439083-90-6	C27H32N4O4	500 µg/1 mg

• BBMP
  A mitochondrial permeability transition pore (PTP) inhibitor which is a potential therapeutic for neurodegenerative diseases.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214575	97120-13-3	C12H11BrN2O3S	5 mg/25 mg

• Benazepril Free base

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-337551	86541-75-5	C24H28N2O5	1 g

• Benazepril hydrochloride
  Angiotensin-converting enzyme (ACE) inhibitor. Reduces myocardial hypertrophy and blood pressure in spontaneous hypertensive rats.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203526	86541-74-4	C24H28N2O5 ·HCl	50 mg

• Benzamidine HCl hydrate
  A reversible inhibitor of serine proteases, trypsin and trypsin-like enzymes. It has also been shown to be a strong inhibitor of plasma and thrombin.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207323	206752-36-5	C7H80N2 ·HCl ·H2O	5 g/25 g

• Benzisoxazole Hsp90 Inhibitor
  Binds the N-terminal domain of Hsp90, efficiently displacing geldanamycin from the ATP binding site; inhibits the proliferation of several cancer cell lines.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-223790	1012788-65-6	C19H20ClN3O4	1 mg /5 mg

• Benzyl isothiocyanate
  An inhibitor of methylazoxymethanol acetate-induced intestinal carcinogenesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204641	622-78-6	C8H7NS	5 g/25 g

• Benzyl thiocyanate
  Effective against methylazoxymethanol acetate-induced intestinal carcinogenesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204643	3012-37-1	C7H5NS	10 g/50 g

• Benzyl-2-acetamido-2-deoxy-a-D-galactopyranoside
  Inhibitor of O-linked glycosylation in a variety of cell lines. Inhibits 2,3(O)-sialyltransferase and disrupts glycoprotein targeting in HT-29 cells. Substrate for N-acetyl-b-D-glucosaminyltransferase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203427	3554-93-6	C15H21NO6	100 mg

• Berberine

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204645	633-65-8	C20H18ClNO4	1 g/5 g

• BI-6C9
  A tBid inhibitor that possesses antiapoptotic properties.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-210915	791835-21-7	C23H25N3O4S2	1 mg/5 mg

• BIBB 515
  An important enzyme in the biosynthesis of animal, fungal and plant sterols; a selective and potent inhibitor of 2,3-Oxidosqualene cyclase (OSC) in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205221	156635-05-1	C22H21ClN2O2	1 mg/5 mg

• BIBR 1532
  A compound suggested to act as a selective and specific telomerase inhibitor. Shown to inhibit hTERT and cell proliferation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203843	321674-73-1	C21H17NO3	10 mg/50 mg

• Bifemelane hydrochloride
  MAO-A and MAO-B inhibitor. Increases locomotor activity in MPTP-treated marmosets and reverses catalepsy induced by tetrabenazine in mice.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203529	62232-46-6	C18H23NO ·HCl	10 mg/50 mg

• Binucleine 2
  Cell-permeable pyrazolo that inhibits the cytokinesis function of the Aurora B kinase pathway and Histone H3 Ser10 phosphorylation in mitotic Drosophila Kc167 cells. Inactive in mammalian systems.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202500	220088-42-6	C13H11ClFN5	5 mg

• Bioallethrin
  Though a type I pyrethroid, its effects on calcineurin (PP2B) resembles those of type II pyrethrins. Unlike most type I pyrethrins, which are very weak, bioallethrin is a potent calcineurin inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202501	22431-63-6	C19H26O3	25 mg/100 mg

• Bis[(4-chlorophenyl)thiomethylene]biphosphonic Acid, Tetraisopropyl Ester
  An intermediate in the synthesis of Tilduronic Acid, a biphosphonate bone resorption inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207374	887353-24-4	C25H36Cl2O6P2S2	100 mg

• Bistheonellide A
  A dimeric marine toxin that can inhibit actin polymerization and cell cycle progression in the G₁ phase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202081	105304-96-9	C74H128O20	100 µg

• (±)-Blebbistatin
  A selective inhibitor of nonmuscle myosin II ATPase and several striated muscle myosins, while reversibly blocking cell blebbing and disrupting cytokinesis via ubiquitin-mediated proteolysis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203532	674289-55-5	C18H16N2O2	10 mg

• BM 15766 sulfate
  A dehydrocholesterol reductase inhibitor that targets 7-dehydrocholesterol reductase. 7-dehydrocholesterol reductase catalyzes the last step of cholesterol synthesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-210953	86621-94-5	C22H25ClN2O2•H2SO4	1 mg/5 mg

• BML-244
  A highly potent, cell-permeable inhibitor of cathepsin K (IC₅₀=51 nM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221370	N/A	C11H21NO3	5 mg/25 mg

• BML-260
  A potent inhibitor of the dual specificity phosphatase JSP-1 (IC₅₀=18µM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-223822	101439-76-3	C17H11NO3S2	10 mg/50 mg

• BML-277
  This product is a checkpoint kinase 2 inhibitor. It protects T cells from apoptosis by controlling the response of p53 to radiation-induced DNA breaks.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200700	516480-79-8	C20H14ClN3O2	10 mg/50 mg

• BMS 453 hydrate
  Shown to be a retinoic acid receptor antagonist which causes a cell cycle arrest at G₁. Also shown to induce Rb hypophosphorylation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-311294	166977-43-1	C27H24O2•xH2O	10 mg

• Bortezomib
  A selective and robust 26S proteasome inhibitor, that is a boronic acid dipeptide derivative.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217785	179324-69-7	C19H25BN4O4	2.5 mg/25 mg

• Bourgeonal
  A potent agonist at hOR17-4 (a human testicular olfactory receptor) that acts as a strong chemoattractant in sperm behavioral assays.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-210959	18127-01-0	C13H18O	10 mg

• BPPA
  Inhibitor of human telomerase (IC₅₀=4.5 µM). Displays cytotoxic activity against human carcinoma cell lines (IC₅₀=1-6µM), an effect unrelated to telomerase inhibition.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200885	N/A	C30H36N4O4 ·2C2H4O2	5 mg/25 mg

• Brassinin
  Effective inhibitor of stage two skin carcinogenesis. Inducer of Phase II enzymes. Inhibitor of chemically induced carcinogenesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202978	105748-59-2	C11H12N2S2	50 mg/100 mg

• BTS
  Inhibitor of Ca²⁺-stimulated myosin S1 ATPase, reversibly blocks gliding motility. Weakens myosin interaction with F-actin. Has no effect on platelet myosin II.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202087	1576-37-0	C14H15NO2S	5 mg

• Bufotalin
  Less potent Na⁺/K⁺-ATPase inhibitor than other bufadienolides. Potent immunosuppressor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202509	471-95-4	C26H36O6	5 mg

• BX 513 hydrochloride
  Inhibits MIP-1α-induced intracellular calcium mobilization (IC₅₀ = 2.5 μM). Selective CCR1 receptor antagonist (K_i values are 0.04, > 10, > 10 and > 10 nM for CCR1, CCR5, CXCR2 and CXCR4 receptors respectively). A full inverse agonist at US28, a HCMV-encoded chemokine receptor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203861	193542-65-3	C28H29ClN2O.HCl	10 mg/50 mg

• BX 795
  A specific and potent inhibitor of IκKε and TBK1. Also has been shown to block nuclear translocation, phosphorylation, and transcriptional activity of interferon regulatory factor 3.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-281689	702675-74-9	C23H26IN7O2S	2 mg/5 mg

• BYK204165
  A potent and selective inhibitor of poly(ADP-ribose) polymerase 1 (PARP1); 100-fold selective for PARP-1 over PARP-2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214642	1104546-89-5	C15H12N2O2	5 mg

• β-cyano-L-Alanine
  A reversible inhibitor of the H2S-synthesizing enzyme cystathionine γ lyase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205546	6232-19-5	C4H6N2O2	10 mg/50 mg

• C 021 dihydrochloride
  A potent CCR4 chemokine receptor antagonist (IC50 values are 0.14 and 0.039 μM for inhibition of chemotaxis in human and mouse respectively)

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-293973	864289-85-0	C27H41N5O2.2HCl	10 mg/50 mg

• CA-074
  Potent and specific inhibitor of cathepsin B in vitro and in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202513	134448-10-5	C18H29N3O6	1 mg

• CA-074 methyl ester
  A Cathepsin B inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214647	147859-80-1	C19H31N3O6	5 mg

• Candesartan Celexetil Ester
  An ester analog of the angiotensin II antagonist Candesartan. Converted to Candesartan during gastrointestinal absorption.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204666	145040-37-5	C33H34N6O6	100 mg/250 mg

• Canrenone
  An active metabolite of spironolactone which inhibits aldosterone biosynthesis, as well as block ouabin effects.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205616	976-71-6	C22H28O3	1 g/5 g

• Carbenoxolone disodium
  Glucocorticoid that inhibits 11 β-hydroxysteroid dehydrogenase (11-HSD) and blocks gap juntion communication.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203868	7421-40-1	C34H48Na2O7	50 mg

• Carbimazole

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205620	22232-54-8	C7H10N2O2S	1 g/5 g

• Carbonyl Cyanide m-Chlorophenylhydrazone
  Reported to be a protonophore, and an inhibitor of ER-Goligi protein transport. Also shown to bind Cytochrome C oxidase with a high affinity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202984	555-60-2	C9H5ClN4	250 mg

• Carboxy-PTIO
  A water soluble derivative of PTIO, reacts with and extinguishes NO without affecting NOS activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200352	148819-93-6	C14H17N2O4	10 mg

• Carboxyatractyloside potassium salt
  A highly selective inhibitor of cytosolic side-specific mitochondrial ADP/ATP carriers. For example, adenine nucleotide translocase (ANT) causes stabilization of the c conformation of ANT leading to permeability transition pore (PTP) opening, loss of mitochondrial membrane potential, and eventually apoptosis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214665	35988-42-2 (non-salt)	C31H44O18S2•xK+	2 mg

• Cathepsin/Subtilisin Inhibitor
  Inhibits members of the cysteine protease family including cathepsin L, and members of the serine protease family including subtilisin Carlsberg and thermitase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221400	N/A	C26H32N3O6Cl	1 mg

• CAY10581
  The enzyme indoleamine 2,3-dioxygenase (IDO) has been implicated in mediating pathological immunosuppression associated with certain diseases, including cancer. Several naphthoquinones inhibit IDO in cells and in vitro, but at low (μM) potency. Importantly, naphthoquinones reduce tumor growth in wild type mice but not in IDO-deficient mice. CAY10581 is a naphthoquinone derivative that potently inhibits IDO (IC₅₀ = 55 nM). It is a more potent inhibitor of IDO than 1-methyl-d-tryptophan (1MT) or annulin B. CAY10581 acts as a reversible uncompetitive inhibitor of IDO and demonstrates minimal impact on cell viability at 100 μM after 24 hours.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-223871	1018340-07-2	C22H21NO4	1 mg/5 mg

• CAY10589
  Microsomal Prostaglandin E2 Synthase-1 (mPGES-1), with cyclooxygenase-2 (COX-2), synthesizes PGE2, which is directly involved in signaling during fever,inflammation and pain. 5-Lipoxygenase (5-LO) initiates the synthesis of leukotrienes (LTs), which are pro-inflammatory mediators. This chemical is a dual inhibitor of mPGES-1 (IC₅₀ = 1.3 μM) and 5-LO (IC₅₀ = 1.0 μM). It effectively inhibits LT and PGE2 synthesis in both cell free and intact cell assays and has minor effects on COX-1 and COX-2, inhibiting these enzymes 34% and 38.8%, respectively, at 10 μM.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-223872	1077626-52-8	C25H28ClN3O2S	1 mg/5 mg

• CAY10594
  A potent PLD2 inhibitor, both in vitro and in cells; strongly inhibits the invasive migration of breast cancer cells in transwell assays.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-223874	1130067-34-3	C26H28N4O2	1 mg/5 mg

• CAY10626

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-358741	1202884-94-3	C31H35F3N8O3	1mg/5mg

• CCG 2046
  Inhibits RGS4.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204676	13017-69-1	C11H10N4	10 mg/50 mg

• CCG-1423
  CCG-1423 is a specific inhibitor of Rho pathway-mediated signalling and activation of serum response factor (SRF) transcription.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205241	285986-88-1	C18H13ClF6N2O3	1 mg/5 mg

• CCR2 Antagonist
  A highly potent CKR-2B (CCR2) receptor antagonist which prevents MCP-1 binding to CKR-2B. Potently antagonizes calcium flux and chemotaxis with selectivity over CKR-3 (CCR3).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202525	445479-97-0	C28H34F3N5O4S	5 mg

• CCR4 Antagonist
  A cell-permeable diaminoquinazoline compound that acts as a potent antagonist against the G-protein-coupled chemokine receptor CCR4. Shown to inhibit CCL22/CCR4-mediated chemotaxis in both murine and human cultures.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221406	N/A	C27H41N5O2 ·0.5 ·H2O	5 mg

• CCT 018159
  Cell-permeable pyrazoloresorcinol compound. Inhibits HSP90 ATPase activity by targeting the N-terminal ATP binding site. Shows no detectable effects against human Hsp70 or topoisomerase II.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202526	171009-07-7	C20H20N2O4	5 mg

• Celocoxib
  A selective cyclooxygenase-2 (COX-2) inhibitor. An anti-inflammatory used in the treatment of familial adenomatous polyposis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-217869	169590-42-5	C17H14F3N3O2S	100 mg/1 g

• Cerivastatin, Sodium Salt
  This compound is a competitive inhibitor of HMG-CoA reductase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207418	143201-11-0	C26H33FNNaO5	2.5 mg

• Cetaben
  The peroxisome proliferator has hypolipidemic activity, can act independent of PPARα, and inhibit ACAT and cholesterol production in human hepatoma Hep-G2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203185	55986-43-1	C23H39NO2	10 mg

• CFM 1571 hydrochloride
  Soluble guanylyl cyclase (sGC) activator (EC₅₀ = 5.49 μM). Does not activate adenylyl cyclase, shows no significant inhibition of phosphodiesterases and displays minimal inhibition of iNOS (25%) and nNOS (17%). Inhibits collagen-stimulated platelet aggregation in vitro (IC₅₀ = 2.84 μM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203540	268725-86-6	C23H28N4O3 ·HCl	10 mg

• cFMS Receptor Inhibitor II
  A cell-permeable anilinoquinoline compound that acts as a strong, active site-targeting inhibitor of MCSF receptor/cFMS. This inhibitor is much more selective against cFMS-independent growth of NSO cells than cFMS Receptor Inhibitor III. They are both equally potent in inhibiting the cFMS-dependent growth of M-NSF-60 cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221415	N/A	C23H20N4O	1 mg

• cFMS Receptor Inhibitor III
  A cell-permeable anilinoquinoline compound that acts as a strong, active site-targeting inhibitor of MCSF receptor/cFMS. This compound is 100-fold more potent in inhibiting the cFMS-dependent growth of M-NSF-60 cells than the cFMS-independent growth of NSO cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221416	N/A	C25H23N3O3S	1 mg

• cFMS Receptor Inhibitor IV
  A cell-permeable furan carboxamide compound that acts as a potent, reversible, and ATP-competitive cFMS/CSF-1R inhibitor. It blocks cFMS autophosphorylation in cell-free in vitro kinase assays and in CSF-1/M-CSF-stimulated HEK-293 cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221417	959626-45-0	C22H26N4O2	5 mg

• CFTR Inhibitor-172
  A voltage-independent inhibitor of CFTR. Shown to block intestinal fluid secretion that is cholera toxin-induced.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204680	307510-92-5	C18H10F3NO3S2	10 mg/50 mg

• CGS 35066
  Potent endothelin-converting enzyme (ECE) inhibitor that displays > 100-fold selectivity over neutral endopeptidase 24.11 (IC₅₀ values are 22 and 2300 nM respectively). Blocks the hypertensive effects induced by big ET-1 in vitro and reduces the magnitude of cerebral vasospasm following subarachnoid hemorrhage (SAH).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203546	261619-50-5	C16H16NO6P	10 mg

• Chlorothiazide
  A carbonic anhydrase inhibitor that is slightly less potent than Acetazolamide (sc-214461), that has been shown to block renal reabsorption of sodium and chloride ions.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202536	58-94-6	C7H6N3ClO4S2	1 g

• CI 898 dihydrochloride
  Dihydrofolate reductase inhibitor, displaying antineoplastic and antiprotozoal properties. Affects G1/S phase cell cycle progression.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203890	82952-64-5	C19H23N5O3.2HCl	10 mg

• Cicaprost
  An analog of PGI₂ which causes IP activation. Activation of IP is associated with phosphorylation of transcription factor cAMP response element binding protein.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-358799	94079-80-8	C22H30O5	500 µg/1mg

• Ciclesonide
  A glucocorticoid microemulsion nasal preparation that acts as an allergy inhibitor and treats rhinitis

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207432	126544-47-6	C32H44O7	10 mg

• Cilazapril
  A monoethyl ester, which acts as an angiotensin-converting enzyme (ACE) inhibitor. The inhibitor functions by inhibiting the the ability of ACE to cleave bonds of angiotensin I and Hip-His-Leu.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207435	88768-40-5	C22H31N3O5	10 mg

• Cinobufagin
  Specific Na⁺/K⁺-ATPase inhibitor. About as active as ouabain

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202542	470-37-1	C26H34O6	5 mg

• Cinobufotalin
  Specific Na⁺/K⁺-ATPase inhibitor. Less active than ouabain.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202101	1108-68-5	C26H34O7	5 mg

• cis-4-Hydroxy-L-proline
  Proline antagonist in collagen synthesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-311305	618-27-9	C5H9NO3	250 mg/1 g

• Clavulanic Acid Potassium Salt
  A β-Lactamase inhibitor usually added to amoxicillin to increase its effectiveness.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207446	61177-45-5	C8H8KNO5	10 mg

• Collagenase Inhibitor I
  A potent and specific inhibitor of vertebrate collagenases with values in the micromolar range.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221432	123984-15-6	C22H32N4O6	5 mg

• Combrestatin A4
  A potent inhibitor of tubulin polymerization and displays strong inhibitory activity on tumor cell growth.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204697	117048-59-6	C18H20O5	1 mg/5 mg

• Conduritol A

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211126	526-87-4	C6H10O4	10 mg

• Conduritol D

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211128	4782-75-6	C6H10O4	10 mg

• Coumestrol
  A plant estrogen and highly potent inhibitor of 17-β-hydroxysteroid oxidoreductase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205638	479-13-0	C15H8O5	10 mg/25 mg

• CP 100356 hydrochloride

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361154	142716-85-6	C31H36N4O6•HCl	10 mg/50 mg

• CP 316 819
  Glycogen phosphorylase inhibitor and potential treatment for glycemic control in diabetes, type 2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207456	186392-43-8	C21H22ClN3O4	10 mg

• Cupferron
  A water soluble free radical polymerization inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214782	135-20-6	C6H9N3O2	25 g

• Curcumin (Synthetic)
  Major curcumoid isolated from tumeric with antioxidant, anticancer and anti-inflammatory activities. Reported to supress NF-κB, COX-1, COX-2 and TNF-α. Upregulates PPARγ, p53 and Nrf2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-294110	458-37-7	C21H20O6	5 g/25 g

• CV-6209
  A competitive PAF receptor antagonist. Inhibits PAF induced human platelet aggregation and PAF induced hypotension and lethality.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207461	100488-87-7	C34H60ClN3O6	2.5 mg

• Cyclic Pifithrin-α hydrobromide

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361164	511296-88-1	C16H16N2S.HBr	10 mg/50 mg

• Cyclosporin H
  An immunologically inactive cyclosporine H that is shown to be a potent inhibitor of phorbol ester.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203013	83602-39-5	C62H111N11O12	1 mg/5 mg

• Cyclothiazide
  Potently inhibits the desensitization of AMPA receptors. Antihypertensive.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202560	2259-96-3	C14H16ClN3O4S2	10 mg/50 mg

• D-Amino Acid Oxidase Inhibitor
  A cell-permeable, potent inhibitor of cellular activity of transfected D-amino acid oxidase (DAO/DAAO/DAMOX/OXDA) in Chinese Hamster Ovary cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203909	39793-31-2	C7H5NO2S	50 mg

• D-Eritadenine
  A potent inhibitor of S-adenosyl-L-homocysteine hydrolase. It is a hypocholesterolemic that is isolated from shiitake mushrooms and affects phospholipid and linoleicacid metabolisms, decreasing total cholesterol levels in plasma.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207632	23918-98-1	C9H11N5O4	10 mg

• D-erythro-2-Tetradecanoylamino-1-phenyl-1-propanol

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-280655	143492-39-1	C23H39NO2	100 mg

• D-erythro-Dihydro-D-sphingosine-1-phosphate
  Used as a negative control for C2 Ceramide.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211174	108126-32-5	C18H40NO5P	5 mg

• D-erythro-N,N-Dimethylsphingosine
  A general modulator of protein kinases.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211175	119567-63-4	C20H41NO2	5 mg

• D-Limonene
  Monoterpene found to prevent mammary cancer by inducing hepatic glutathione-S- transferase and uridine diphosphoglucuronosyl transferase. Isoprenylation inhibitor of small G-proteins.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205283	5989-27-5	C10H16	100 ml/500 ml

• D,L-Benzylsuccinic Acid
  Effective carboxypeptidase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207490	36092-42-9	C11H12O4	5 g

• D,L-Venlafaxine
  An isomer of Venlafaxine, the reuptake inhibitor of neuroamines such as serotonin and norepinephrine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207501	93413-69-5	C17H27NO2	50 mg

• D(+)Galactosamine, Hydrochloride
  Powerful inhibitor of hepatic RNA synthesis. Increases the adherence of polymorphonuclear leukocytes to hepatic endothelial cells and induces superoxide production.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202568	1772-03-8	C6H13NO5 ·HCl	1 g/5 g

• D609
  D609 is a selective inhibitor of phosphatidylcholine-specific PLC.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201403	83373-60-8	C11H15OS2K	5 mg/25 mg

• Dabigatran etexilate
  Dabigatran etexilate is the prodrug of the active moiety dabigatran. Dabigatran etexilate has recently been in clinical trials for use as an anticoagulant drug. It has been shown to have slight, but significant drug-drug interactions when used in combination with strong P-glycoprotein inducers or inhibitors such as amiodarone (sc-291891) or rifampicin (sc-200910). It has also been associated with lower rates of stroke and systemic embolism than warfarin (sc-205888), a comparable anticoagulant.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-351724	211915-06-9	C34H41N7O5	10 mg

• Daidzin
  A kudzu isoflavone. Demonstrates chemopreventive activities by inhibiting the bioactivation of carcinogenic arylamines. Daidzin is also an inhibitor of human mitochondrial aldehye dehydrogenase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202123	552-66-9	C21H20O9	1 mg/5 mg

• Daltroban
  A selective thromboxane A2 receptor antagonist which exerts protective effects on brain infarction, heart cell injury due to hypoxia and hypoglycemia and lowers serum CPK activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214835	79094-20-5	C16H16ClNO4S	5 mg/25 mg

• Danazol
  A synthetic gonadotropin inhibitor which has a preventive effect on estrogen-related endometrial carcinogenesis in mice.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203021	17230-88-5	C22H27NO2	100 mg/250 mg

• Daunorubicinol (mixture of diastereomers)
  A Daunorubicin metabolite.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218089	28008-55-1	C27H31NO10	2.5 mg

• Decarestrictine D
  A 10-membered lactone which potently inhibits cholesterol biosynthesis and shows hypolipidemic activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202571	127393-89-9	C10H16O5	1 mg/5 mg

• Dechlorane 603
  A chlorinated polycyclic compound which is an antioxidant having prolonged thermal stability

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211216	13560-92-4	C17H8Cl12	25 mg

• Dechlorane A

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-363275	13560-89-9	C18H12Cl12	100 mg

• Dehydrocostus Lactone
  Inhibits NF-Kappa-B activiation by preventing TNF-alpha induced degradation and phosphorylation. Renders HL-60 cells susceptible to TNF-alpha induced apoptosis by enhancing caspase3 and caspase8 activities.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205643	477-43-0	C15H18O2	5 mg/10 mg

• Demecolceine
  An antimitotic agent that disrupts microtubles preventing tubulin polymerization. Stimulates the intrinsic GTPase activity of tubulin. Induces apoptosis in several normal and tumor cell lines and activates JNK/SAPK signaling.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218111	518-11-6	C20H23NO5	50 mg

• Demecolcine Hydrogen Bromide Salt
  An antimitotic agent that disrupts microtubles preventing tubulin polymerization. Stimulates the intrinsic GTPase activity of tubulin. Induces apoptosis in several normal and tumor cell lines and activates JNK/SAPK signaling.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218112	N/A	C21H26BrNO5	50 mg

• Deoxy Blebbistatin
  A Blebbistatin derivative, a compound that blocks myosin II-dependent cell processes.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218116	856925-72-9	C18H16N2O	25 mg

• Dermatan Sulfate
  Mucopolysaccharide containing iduronic acid. Abundant in skin, arterial walls, and heart valves. Shown to inhibit adenylate kinase from rat hepatic membranes and acts as a potent mediator of fibroblast growth factor-2 responsiveness.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203916	54328-33-5	N/A	250 mg

• Desmethyl Atomoxetine Hydrochloride
  A metabolite of Tomoxetine (Atomoxetine, LY 139603).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207537	881995-46-6	C16H20ClNO	1 mg

• Desmethyl Atomoxetine-d7 Hydrochloride Salt
  A labeled derivative of Tomoxetine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218148	N/A	C16H12D7NO.HCl	1 mg

• Diallyl sulfide
  A modulator of drug metabolizing enzyme P450 system and inducer of the phase II detoxifying enzyme GST. Inhibitor of chemical-induced carcinogenesis in many tissues.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204718	592-88-1	C6H10S	25g/100 g

• Dibenzazepine (Deshydroxy LY 411575)
  A dipeptidic (c)-secretase inhibitor and anti-Alzheimer agent.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207554	209984-56-5	C26H23F2N3O3	2 mg

• Diethylumbelliferyl phosphate
  A potent, selective cholesterol esterase inhibitor which blocks steroidogenesis primarily by preventing cholesterol transport into the mitochondria of steroidogenic cells. Inhibitors of cholesterol esterase are anticipated to limit the absorption of dietary cholesterol. IC₅₀= 11.6 µM.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211328	897-83-6	C13H15O6P	5 mg/25 mg

• Dihydrokainic acid
  An agonist of the glutamate-recognizing ionotropic kainate receptors. Employed as a tool for inducing excitotoxicity and producing seizures in neurotransmission models.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200442	52497-36-6	C10H17NO4	5 mg/25 mg

• Dimethyl-Bisphenol A
  A newly identified HIF-1α degradation promotor1.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205650	1568-83-8	C17H20O2	10 mg/50 mg

• Diminutol
  A cell-permeable 2,6,9-trisubstituted purine analog that blocks mitotic spindle assembly by competitively inhibiting NQO1, an NADP-dependent oxidoreductase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203923	361431-33-6	C19H26N6OS	5 mg

• Dipeptidylpeptidase II Inhibitor
  Aminoacylpiperidine compound that acts as a strong and very specific inhibitor of dipeptidylpeptidase II. Displays >7,700-fold selectivity for DPP II over DPP IV from human seminal fluid.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221546	N/A	C9H19N3O	10 mg

• Dipeptidylpeptidase IV Inhibitor II
  A new acylating inhibitor for the proline-specific peptidases dipeptidylpeptidase II and IV. Acts as a strong reversible inhibitor of human placenta dipeptidylpeptidase II and porcine kidney dipeptidylpeptidase IV. Combines the efficacy of aminoacyl pyrrolidides and the potential transacylating capability of diacylhydroxylamines.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221547	1258008-19-3	C16H21N3O4•HCl	1 mg

• Dipeptidylpeptidase IV Inhibitor III
  Orally bioavailable dicyanopyrrolidine compound. Slow-binding and active site-targeting inhibitor of DPP IV with little activity against DPP II, DPP III, DPP VIII, DPP IX, FAP, or APP.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202582	866396-34-1	C14H20N4O2 ·HCl	5 mg

• Dipeptidylpeptidase IV Inhibitor IV, K579
  An agent that acts as a low-binding DPP IV inhibitor. It is more potent and a slower binding inhibitor than NVP-DPP728.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202583	440100-64-1	C17H24N6O	5 mg

• Disodium Cycloheptylaminomethylene diphosphonate
  While used in the treatment of bone disorders, it inhibits squalene synthase and cholestrol biosynthesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204731	138330-18-4	C8H17NNa2O6P2	25 mg/100 mg

• DL-2-Mercaptomethyl-3-guanidinoethylthiopropanoic Acid
  A potent and reversible inhibitor of human plasma carboxypeptidase N. Reported to inhibit hydrolysis of bradykinin.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-311322	77102-28-4	C7H15N3O2S2	100 mg

• DL-Propargylglycine (hydrochloride)
  An irreversible inhibitor of cystathionine-γ-lyase (CSE), which is a H₂S synthesizing enzyme. This compound also inhibits methionine biosynthesis, causes growth inhibition and morphological changes.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221558	N/A	C5H7NO2 ·HCl	1 mg/5 mg

• DL-TBOA

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361170	N/A	C11H13NO5	10 mg/50 mg

• DMFO Hydrochloride
  A specific irreversible inhibitor of ornithine decarboxylase, which shows antiapoptotic, antiparasitic, and antiangiogenic activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203563	70052-12-9	C6H12F2N2O2 ·HCl	10 mg/50 mg

• DNA Base Excision Repair Pathway Inhibitor
  A potent, nontoxic, specific, and cell-permeable DNA repair enzyme inhibitor. Targets the Ref-1 (APE1) active site inhibiting its 3′-phosphodiesterase and 3′-phosphatase activities.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202588	6960-45-8	C9H6N2O4	100 mg

• Docetaxel Trihydrate
  This compound acts as an antineoplastic, as well as an antimitotic agent that promotes the assembly of microtublules which inhibits their depolymerization to free tubulin.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207594	148408-66-6	C43H59NO17	5 mg

• Dorzolamide Hydrochloride
  An inhibitor of carbonic anhydrase, as well as an antiglaucoma agent.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207596	130693-82-2	C10H17ClN2O4S3	10 mg

• Dutasteride

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207600	164656-23-9	C27H30F6N2O2	10 mg

• Dynamin Inhibitor I, Dynasore
  Cell-permeable semicarbazone compound. Inhibits the GTPase activities of dynamin1/2 and Drp1, while exhibiting no significant effect against two other small GTPases, Mx1 and Cdc42.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202592	304448-55-3	C18H14N2O4	10 mg

• Dynamin Inhibitor II
  A cell-permeable cationic surfactant that reversibly inhibits dynamin GTPase activity by targeting the PH domain and interfering with phospholipid binding.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203931	1119-97-7	C17H38NBr	500 mg

• Dynasore monohydrate
  A cell-permeable, reversible noncompetitive dynamin 1 and 2 GTPase activity inhibitor, where it also inhibits mitochondrial Drp1. Dynasore blocks dynamin-dependent endocytosis and scission of endocytic vesicles. it is profibrotic, induces PAI-1 in pleural mesothelial cells, and may be an effective pleurodesing agent. Dynasor blocks human papillomavirus type 16 (HPV16) and bovine papillomavirus type 1 (BPV1) (pseudovirions) infections.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-214953	304448-55-3 (anhydrous)	C18H14N2O4 ·H2O	5 mg/25 mg

• EBPC
  A potent aldose reductase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203572	57056-57-2	C14H15NO4	10 mg/50 mg

• Eg5 Inhibitor III, Dimethylenastron
  Cell-permeable quinazoline-thione compound that acts as a strong, specific, and reversible inhibitor of the microtubule-stimulated ATPase activity of the mitotic motor, Eg5. Shows little effect on the ATPase activity of kinesin-1, -4, -7 and -10. Also inhibits bipolar spindle formation in both HeLa cells and in Xenopus egg extracts and induces cell cycle arrest (~1 µM). Shown to induce mitotic arrest, apoptosis and upregulate Hsp70 in human multiple myeloma cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221576	863774-58-7	C16H18N2O2S	1 mg

• Eg5 Inhibitor IV, VS-83
  A cell-permeable Monastrol analog with enhanced potency and selectivity (over 8 other kinesins) in inhibiting mitotic kinesin Eg5-ATPase activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203933	909250-29-9	C14H11FN2OS	5 mg

• Eg5 Inhibitor VI
  Cell-permeable biphenylsulfamide compound that acts as a strong, reversible, and ATP-competitive inhibitor of Eg5/KSP ATPase activity with reactivity against both wild-type and the D130V mutant in cell-free assays. The inhibitor exhibits a much weaker antiproliferative activity against WT-expressing cells in cultures because of the higher ATP binding affinity of the WT enzyme, and its in vivo antitumor efficacy has only been demonstrated in HCT116 D130V xenografed mice, but not mice with WT KSP-bearing Colo205.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-281686	N/A	C13H11F3N2O2S	5 mg

• Eg5 Inhibitor VII
  Cell-permeable quinolinone compound that acts as a very potent and selective Eg5/KSP inhibitor by antagonizing ATP binding via an allosteric site. Effectively induces monopolar spindles in ovarian adenocarcinoma SKOV3 cells and inhibits the proliferation of colorectal carcinoma HCT116 cells. It is not competitive with respect to microtubule and exhibits minimal activity against a panel of 7 other mitotic kinesins.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221578	N/A	C16H12F3NO	5 mg

• eIF4E/eIF4G Interaction Inhibitor, 4EGI-1
  Reported to inhibit cap-dependent protein translation and also induce apoptosis in cells via down-regulations of FLIP_S/L and induction of DR5.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202597	315706-13-9	C18H12Cl2N4O4S	10 mg

• Elacridar
  A prototypical BCRP inhibitor which inhibits the Bcrp1-mediated transport.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207613	143664-11-3	C34H33N3O5	10 mg/5 mg

• Elacridar-d4
  A prototypical BCRP inhibitor. Inhibits the Bcrp1-mediated transport.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218297	143664-11-3 (unlabeled)	C34H29D4N3O5	1 mg

• Elasnin
  An inhibitor of human leukocyte elastase, different other elastases and chymotrypsin.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-280684	68112-21-0	C24H40O4	1 mg/5 mg

• Elastase Inhibitor II
  A strong irreversible inhibitor of human neutrophil elastase (HNE). The cross-linking of the catalytic residues His57 and Ser195 results in inhibition.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-294466	N/A	C20H31ClN4O7	5 mg/10 mg

• Elastase Inhibitor III
  Strong irreversible inhibitor of human leukocyte elastase (HLE). Protects against injury of the lungs induced by instillation of elastase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-294467	N/A	C22H35ClN4O7	5 mg

• Enalapril Maleate
  An angiotensin-converting enzyme inhibitor. Actively interferes with the renin-angiotensin- aldosterone system.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205666	76095-16-4	C24H32N2O9	1 g/5 g

• ent Atomoxetine-d3, Hydrochloride
  A labeled enantiomer of Tomoxetine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218309	N/A	C17H19D3ClNO	1 mg

• ent S-(+)-Atomoxetine Hydrochloride
  An enantiomer of Atomoxetine (Tomoxetine, LY 139603) which is less effective than Tomoxetine as a competitive and specific inhibitor of norepinephrine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211408	82857-39-4	C17H22ClNO	5 mg

• EO 1428
  Selective inhibitor of p38α and p38β2. Displays no activity at p38γ, p38δ, ERK1/2 and JNK1. Inhibits production of inflammatory cytokines including IL-8, TNF-α, IL-6, IL-1β and IL-10 (IC₅₀ values are 4, 5, 17, 30 and 74 nM respectively). Displays anti-inflammatory activity in murine models of acute and chronic dermatitis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203942	321351-00-2	C20H16BrClN2O	10 mg/50 mg

• Epostane
  A 3β-Hydroxysteroid dehydrogenase inhibitor and a derivative of trilostane. Interceptive.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207627	80471-63-2	C22H31NO3	1 mg

• Erastin
  Cell-permeable piperazinyl-quinazolinone compound that exhibits oncogene-selective lethality. Shown to bind mitochondrial volatage-dependent anion channels (VDAC) and alter its gating; rapidly induce an oxidative, non-apoptotic cell death in several human tumors harboring activating mutations in the RAS-RAF-MEK signaling.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205677	571203-78-6	C30H31ClN4O4	5 mg

• ErbB2 Inhibitor II
  Cell-permeable triazole compound that targets the ATP-binding site of erbB2/HER2. Reduces the phosphorylation of erbB2 in MDA-MB-453 cells, but not that of the over-expressed erbB1 in MDA-MB-468 cells even at concentrations as high as 100 µM. Has been shown to suppress MDA-MB-453 growth with an IC₅₀ of 30.9 µM.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221592	N/A	C15H10N4O	5 mg

• Esomeprazole Magnesium
  Omeprazole S-form and gastric proton pump inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207635	217087-09-7	C34H36MgN6O6S2	10 mg

• Estrone 3-O-Sulfamate
  A potent inhibitor of estrone sulfatase. This compound inhibits estrone sulfatase >99% at 0.1μM in intact MCF-7 cells, IC₅₀=65pM.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207641	148672-09-7	C18H23NO4S	1 mg

• Etidronate Disodium

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205687	7414-83-7	C2H6Na2O7P2	1 g/5 g

• Etoposide Phosphate

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-357357	117091-64-2	C29H33O16P	25 mg/100 mg

• Etravirine
  Novel HIV reverse transcriptase inhibitor useful in treatment of HIV infection.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207674	269055-15-4	C20H15BrN6O	5 mg

• Everolimus
  A macrolide derived from Rapamycin (sc-3504), shown to inhibit cell proliferation induced by growth factors.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218452	159351-69-6	C53H83NO14	5 mg/50 mg

• Exo 1
  A reversible inhibitor of exocytosis Golgi ARF 1 (ADP-Ribosylation Factor) GTPase activator.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215010	75541-83-2	C15H12NFO3	5 mg/25 mg

• Ezetimibe
  A cholesterol transport inhibitor that affects NPC1L1 and prevents its incorporation into membrane clathrin-coated vesicles.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205690	163222-33-1	C24H21F2NO3	25 mg/100 mg

• FAAH Inhibitor I
  A cell-permeable carbamate compound that acts as a strong, selective, and irreversible inhibitor of fatty acid amide hydrolase. Has been shown to block anandamide breakdown in cultured rat cortical neurons and inhibit brain FAAH activity and modulate anxiety in rats. Has no affect on activities of serine hydrolases , acetylcholinesterase butyrylcholinesterase, and monoglyceride lipase. Does not show any interaction with several ion-channels, neurotransmitter transporters, or affect the ligand binding of cannabinoid receptors, CB1 and CB2

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221605	N/A	C18H21NO3	10 mg

• FAAH Inhibitor II
  Cell-permeable carbamate compound. Potent, selective, and irreversible inhibitor of fatty acid amide hydrolase (FAAH). Block anandamide breakdown in rat cortical neurons.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202605	546141-08-6	C20H22N2O3	5 mg

• FABP4 Inhibitor
  A biphenylazolo-oxyacetate that is an effective inhibitor of adipocyte Fatty-Acid-Binding Protein.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202606	300657-03-8	C31H26N2O3	5 mg

• Farnesyl Thiosalicylic Acid Amide
  Association of Ras protein to the inner surface of the plasma membrane is required for Ras signaling activity. Farnesyl thiosalicylic acid (FTS) inhibits Ras-mediated signaling by dislodging Ras from the cell membrane thereby rendering it susceptible to proteolytic degradation. FTS amide is an FTS derivative with an amide added to the carboxyl group. FTS amide inhibits the growth of U87 and Panc-1 tumor cells with IC₅₀ values of 10 and 20 µM, respectively, a relatively higher potency compared to that of FTS (IC₅₀s = 50 and 35 µM, respectively) (2). Treatment of nude mice bearing either Panc-1 or U87 glioblastoma tumors with 100 mg/kg FTS-amide twice daily for four days inhibits tumor growth by at least 50% of controls.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-223986	1092521-74-8	C22H31NOS	1 mg/5 mg

• Fasentin
  A novel glucose uptake (GluT1) inhibitor. Evasion of death receptor ligand-induced apoptosis is an important contributor to cancer development and progression. Therefore, compounds that restore sensitivity to death receptor stimuli would be important tools to better understand this biological pathway and provide potential leads for therapeutic adjuncts. Sensitizes cells to FAS-induced cell death. Fasentin selectively sensitized to death ligands, but did not decrease FLIP expression. It alters gene expression associated with nutrient and glucose deprivation. Fasentin interacted with a unique site in the intracellular channel of the glucose transport protein GLUT1. It highlights a new mechanism to sensitize cells to death ligands. Dipyridamole (sc-200717), which is a weak GluT inhibitor which partially inhibits glucose uptake ane sensitize cells to FAS. Two glucose uptake inhibitor, phloretin & cytochalasin B, have been reported to be highly toxic and not sensitize cells to FAS.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215012	392721-37-8	C11H9ClF3NO2	5 mg/25 mg

• FBPase-1 Inhibitor
  A cell-permeable benzoxazolo-sulfonamide compound that inhibits hFBPase-1 enzymatic activity by competing at the AMP allosteric binding site. Has been shown to block glucose production in starved rat hepatoma cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221608	N/A	C13H7Cl3N2O3S	10 mg

• Febuxostat
  This compound inhibits xanthine oxidase and xanthine dehydrogenase, where it is used for the treatment of chronic gout and hyperuricemia.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207680	144060-53-7	C16H16N2O3S	10 mg

• Finasteride
  Orally active antiandrogen that inhibits type II 5α reductase (IC₅₀ = 65 nM). Suppresses the conversion of testosterone to dihydrotestosterone. Reduces prostatic dihydrotestosterone levels and prostate size in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203954	98319-26-7	C23H36N2O2	50 mg

• FK-506
  An agent that binds to the immunophilin FKBP12 and inhibits PP2B (calcineurin). The compound can also inhibit specific transduction pathways.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-24649	104987-11-3	C44H69NO12	1 mg/10 mg

• FK-866
  A non-competitive and specific inhibitor of nicotamide phosphrybosyltransferase that mediates NAD⁺ biosynthesis within cells and causes apoptosis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205325	658084-64-1	C24H29N3O2	5 mg/10 mg

• FKGK 11
  Phospholipase A2 (PLA2) catalyzes the hydrolysis of fatty acids at the sn-2 position of glycerophospholipids, yielding a lysophospholipid and a free fatty acid as products. There are three broad classes of PLA2, secretory (sPLA2), calcium-independent cytosolic (iPLA2), and calcium-dependent cytosolic (cPLA2), that have different functions. FKGK 11 is a selective inhibitor of iPLA2 that demonstrates an XI(50) value of 0.0073, where XI(50) equals the mole fraction of FKGK 11 in the total substrate interface required to inhibit iPLA2 by 50% . In comparison, mole fractions as high as 0.091 do not inhibit cPLA2 activity and cause only minute inhibition of sPLA2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-223989	1071000-98-0	C13H13F5O	500 µg/1 mg

• Flurofamide
  A bacterial urease inhibitor with a potency 1000 fold greater than Acetohydroxamic Acid.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203957	70788-28-2	C7H9FN3O2P	50 mg

• Fluvastatin, Sodium Salt
  A synthetic 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) reductase inhibitor that acts as an anti-hypercholesterolemic agent.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202613	93957-55-2	C24H25FNNaO4	25 mg

• Fluvoxamine
  A selective serotonin reuptake inhibitor (SSRI), which is used as an anti-depressant.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207697	54739-18-3	C15H21F3N2O2	25 mg

• Foroxymithine
  A potent chelator of the ferrous ion and specific inhibitor of angiotens.in I converting enzyme at an IC₅₀ of 7μg/ml

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202159	100157-28-6	C22H37N7O11	1 mg

• Fosinopril sodium
  An angiotensin-converting enzyme inhibitor shown to protect the organs in sinoaortic-denervated rats.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205702	88889-14-9	C30H45NNaO7P	25 mg/100 mg

• FTI 276

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361181	170006-72-1	C21H27N3O3S2.C2HF3O2	1 mg

• Fumitremorgin C
  A diketopiperazine, fungal toxin, isolated from Aspergillus fumigatus that acts as a strong and specific BRCP inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202162	118974-02-0	C22H25N3O3	250 µg

• Furosemide
  Loop diuretic inhibitor of Na+/2Cl-/K+ (NKCC) cotransporter. Acts as a non-competitive antagonist at GABA_A receptors with ~ 100-fold greater selectivity for α6-containing receptors than α1-containing receptors.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203961	54-31-9	C12H11ClN2O5S	50 mg

• Gadolinium (III) chloride hexahydrate
  Inhibits macrophages.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202617	13450-84-5	GdCl3•6H2O	100 mg/500 mg

• Galactostatin Bisulfite
  A β-galactosidase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218555	1196465-02-7	C6H13NO7S	1 mg

• Galiellalactone
  A hexaketide metabolite, which selectively inhibits IL-6 induced SEAP expression by blocking the binding of activated Stat3 dimers to DNA.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202165	133613-71-5	C11H14O3	500 µg

• Gamma-Secretase Inhibitor
  Reversible peptidomimetic inhibitor of Alzheimer's Gamma-Secretase activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221656	N/A	C33H57N5O9F2	1 mg

• Garcinol
  A potent inhibitor of p300 and PCAF histone acetyltransferases. Shown to down-regulate global gene expression in HeLa cells and to inhibit growth in two breast cancer cell lines. Also exhibits anti-carcinogenic and anti-inflammatory properties.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200891	78824-30-3	C38H50O6	10 mg/50 mg

• Gedunin
  Naturally occurring Hsp90 inhibitor. In vitro, induces Hsp90-dependent client protein degradation and displays antiproliferative activity (IC₅₀ values are 3.22, 8.84 and 16.8 μM in SKBr3, MCF-7 and CaCo-2 cancer cell lines respectively). Exhibits antimalarial activity against P. falciparum (IC₅₀ values are 0.14 and 3.1 μM in parasite development and [3H]-hypoxanthine uptake assays respectively).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203967	2753-30-2	C28H34O7	10 mg

• Gemfibrozil 1-O-β-D-Glucuronide Allyl Ester
  Gemfibrozil glucuronide derivative.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-280722	N/A	C24H34O9	1 mg

• GGACK
  A specific and potent factor Xa inhibitor, reported to decrease creatine kinase and amylase activity

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201314	65113-67-9	C14H25ClN6O5	5 mg

• Glucagon Receptor Antagonist I
  Potent and selective cell-permeable thienyl-amide compound that acts as a competitive antagonist of the glucagon receptor. Exhibits binding to hGCGR with high affinity and prevent its interaction with glucagon (IC₅₀ = 181 nM, KDB = 81 nM, and pA2 = 7.1 in membranes prepared from CHO-hGCGR). Also suppresses glucagon-induced glycogenolysis in human primary hepatocytes and in mice (50 mg/kg, ip).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203972	438618-32-7	C20H30N2OS	1 mg/5 mg

• Glucagon Receptor Antagonist, Control
  Cell-permeable thienyl-amide compound that serves as an inactive control for Glucagon Receptor Antagonist.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203973	362482-00-6	C21H23BrN2OS	1 mg/5 mg

• (±)-Lisofylline
  A synthetic methylxanthine metabolite of Pentoxifylline. Inhibits phosphatidic acid generation. Suppresses release of IL-12 and blocks IL-12-mediated STAT4 activation. Protects against autoimmune pancreatic β cell destruction.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201055	6493-06-7	C13H20N4O3	10 mg/50 mg

• Glutaryl-leu-OH
  Potent and highly specific enkephalinase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-285863	209127-97-9	C16H21NO5	25 mg/100 mg

• Glycogen Phosphorylase Inhibitor
  A cell-permeable urea compound that acts as a potent and AMP-competitive inhibitor of glycogen phosphorylase (GP; IC₅₀ = 53 nM). Inhibits glucagon-induced glyocgenolysis in both hepatocytes in vitro and in rats in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203975	648926-15-2	C17H15ClF2N4O4	1 mg

• Granisetron
  Used to successfully treat post operative nausea.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203983	109889-09-0	C18H24N4O	25 mg/100 mg

• GSK 264220A
  An endothelial lipase and a lipoprotein lipase inhibitor (IC50 values are 0.13 and 0.10 μM respectively).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295026	685506-42-7	C17H21N3O4S	10 mg/50 mg

• Guanosine 3',5'-cyclic Monophosphothioate, Rp-Isomer sodium salt
  Inhibitor of cGMP-dependent protein kinase (PKG) 1α (cGMP antagonist).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203063	86562-09-6 (non-salt)	C10H11N5O6SP ·Na	1 mg

• GW 9662
  A selective, irreversible, and effective PPARγ antagonist that also acts as a FXR and PXR agonist. Shown to block Rosiglitazone (sc-202795)-mediated activation of PPARγ.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202641	22978-25-2	C13H9ClN2O3	5 mg

• GW-441756
  A specific tropomyosin-related kinase A (TrkA) tyrosine kinase inhibitor, reported to block cell death induced by TrKA.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200683	504433-23-2	C17H13N3O	10 mg/50 mg

• GW2974
  A dual selective inhibitor of EGFR and Neu (ErbB-2) receptor tyrosine kinases. This compound inhibits cancer line PC-3 growth.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-252869	202272-68-2	C23H21N7	50 mg

• GW311616A
  A potent inhibitor of intracellular human neutrophil elastase (HNE, α-1-proteinase).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215120	197090-44-1	C19H32ClN3O4S	1 mg/5 mg

• HBDDE
  Inhibits PKCα (IC₅₀=43 µM) and PKCγ (IC₅₀=50 µM) without inhibiting the δ, βI and βII isotypes

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202174	154675-18-0	C16H18O8	1 mg/5 mg

• Hdm2 E3 Ligase Inhibitor
  A cell-permeable and reversible inhibitor of Hdm2 E3 ligase that selectively blocks Hdm2 E3-mediated ubiquitination. Has been shown to inhibit ubiquitination of p53 in vitro (IC₅₀ = 12.7 µM using Ub-Ubc as the donor substrate). The inhibition is non-competitive with respect to either the donor or acceptor substrate. Exhibits little effect towards other ubiquitin-using enzymes.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221707	N/A	C10H8F6N2O3S	5 mg

• HDS 029
  Potent inhibitor of ErbB receptor family (IC₅₀ values are 0.3, 0.5 and 1.1 nM for ErbB1 (EGFR), ErbB4 and ErbB2 respectively). EGF-induced erbB1 autophosphorylation inhibitor in NIH3T3 cells and heregulin-stimulated ErbB autophosphorylation in MDA-MB-453 human breast carcinoma cells (IC₅₀ values are 2.5 and 24 nM respectively).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203995	881001-19-0	C17H11ClFN5O	1 mg/10 mg

• Heat Shock Protein Inhibitor I
  A benzylidene lactam compound that blocks the induction of heat shock proteins HSP70, HSP72, and HSP105. Blocks the development of thermotolerance in a dose-dependent manner. Does not affect the thermosensitivity of nontolerant cells. Does not have an affect on the activities of PKA, PKC, or PTK.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221709	N/A	C13H11NO4	5 mg

• Hellebrin
  Cardiotonic glycoside with a bufadienolide-steroid structure. Extremely potent inhibitor of Na⁺/K⁺-ATPase and blocks efflux of Na⁺ and reuptake of K⁺ of this enzyme.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202645	13289-18-4	C36H52O15	1 mg/5 mg

• Heptakis(2,3-di-O-methyl-6-O-sulfo)-β-cyclodextrin Heptasodium Salt
  Anthrax lethal toxin inhibitor and β-Cyclodextrin derivative

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207730	201346-23-8	C56H91Na7O56S7	5 mg

• Hexestrol
  A carcinogenic synthetic estrogen that inhibits microtubule polymerization and the formation of ribbon structures, while also an inhibitor of lipid peroxidation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205713	84-16-2	C18H22O2	1 g/5 g

• HIF-1 Inhibitor
  Cell-permeable amidophenolic compound that inhibits hypoxia-induced HIF-1 transcription activity by selectively blocking the hypoxia-induced accumulation of cellular HIF-1α protein. Exhibits no apparent effect on the cellular level of HIF-1α mRNA nor HIF-1.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221724	N/A	C26H29NO5	10 mg

• Histone Lysine Methyltransferase Inhibitor
  An HMTase inhibitor, suppressing H3K9me2 generation by G9a. Does not compete with S-adenosyl-methionine cofactor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202651	935693-62-2	C28H38N6O2	5 mg

• HQNO
  A high affinity inhibitor of quinone oxidation and Zn(II), also described to inhibit proton channels needed to reduce oxygen and the activity of proton pumps.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202654	341-88-8	C16H21NO2	10 mg/50 mg

• HSD Inhibitor 23
  Selective, potent and cell permeable small molecule inhibitor of 11-β-hydroxysteroid dehydrogenase

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203076	868604-75-5	C24H33F3N4O2	1 mg

• HWY 5069
  An isoquinolinium derivative which inhibits the proliferation of wild-type and all mutants of Schizosaccharomyces pombe.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207737	914917-58-1	C31H45BrFN	5 mg

• Hydroxylamine hydrochloride
  A compound used as a catalyst, copolymerization inhibitor, and swelling agent that acts as a potent reducing agent, converting aldehydes and ketones to oximes. Also exhibits acitivity of converting acid chlorides to hydroxamic acids. Displays inhibitive activity as an MAO inhibitor for platelet aggregation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211616	5470-11-1	NH2OH ·HCl	5 g/100 g

• Ibandronic Acid
  A biphosphonate bone resorption inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207749	114084-78-5	C9H23NO7P2	100 mg

• Ibufenac
  Used as an analgesic and anti-inflammatory.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211624	1553-60-2	C12H16O2	50 mg

• ICI 192,605

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361209	117621-64-4	C22H23ClO5	10 mg/50 mg

• IDFP
  An organophosphorus compound that dually inhibits MAGL and FAAH with IC₅₀ values of 0.8 and 3 nM, respectively. At 10 mg/kg, IDFP elevates brain levels of 2-AG and AEA more than 10-fold, and decreases levels of arachidonic acid by 10-fold.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205348	615250-02-7	C15H32FO2P	500 µg/1 mg

• IDRA 21
  Analog of cyclothiazide. Inhibits AMPA receptor desensitization. Crosses the blood-brain barrier more readily than cyclothiazide and diazoxide and is a more potent cognitive enhancing drug.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202659	22503-72-6	C8H9ClN2O2S	5 mg/25 mg

• [Ile7]-Angiotensin III
  Angiotensin III inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295174	102029-49-2	N/A	1 mg/5 mg

• Imidapril Hydrochloride
  An inhibitor of angiotensin converting enzyme (ACE). Antihypertensive.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207751	89371-37-9	C20H28ClN3O6	10 mg

• IMS2186
  An anti-proliferative and anti-angiogenic compound. IMS2186 is a novel synthetic compound developed as an anti-CNV drug. The proposed mechanism of action under investigation, is blocking the cell cycle at G2 and inhibiting the production of PGE2/TNF-α. The latter contributing to anti-angiogenic and antiinflammatory effects. IMS2186 inhibits cell growth in vitro in tumor cells, non-transformed fibroblasts, and retinal pigment epithelial cells. IMS2186 inhibits angiogenesis (IC₅₀= 0.1 µM) and cell migration, which plays a role in many biological processes: inflammation, angiogenesis, and scar formation. The physicochemical structure of IMS2186 showed also that the free drug concentration in a physiological media (e.g., vitreous or saline) is 8-10 µM above the IC₅₀ for all these activities (0.1-3.0 µM). Intraocular injection of IMS2186 could be a long-lasting effective treatment for CNV (choroidal neovascularization) in AMD (age-related macular degeneration) with a reduction in scarring and related visual loss.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211638	1031206-36-6	C18H16O4	5 mg/25 mg

• Indibulin
  A microtubule destabilizer that blocks tubulin polymerization (IC50 = 0.3 μM). Blocks cell cycle progression at metaphase and displays antitumor activity against a variety of malignancies in vitro (IC50 values ranging from 0.036-0.285 μM). Has been shown to induce complete tumor remission in the Yoshida AH13 rat sarcoma model in vivo. Lacks neurotoxicity due to an ability to discriminate between posttranslationally modified tubulin in mature neuronal microtubules and less-modified tubulin present in immature neuronal or nonneuronal microtubules. Also displays oral availability and efficacy towards MDR tumor cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295179	204205-90-3	C22H16CIN3O2	10 mg/50 mg

• INH1
  Inhibitor that binds Hec1, inhibiting its association with Nek2 and kinetochores. Causes arrest of mitosis and inhibits proliferation in breast cancer cell lines (GI50= 10-20 μM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295181	313553-47-8	C18H16N2OS.HCl	10 mg/50 mg

• Inotilone
  A potent COX-2 inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207758	906366-79-8	C12H10O4	5 mg

• IP3K Inhibitor
  A cell-permeable 2,6-disubstituted purine compound that acts as a selective, ATP-competitive inhibitor of IP 3-K (IC50 = 10.2 µM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204015	519178-28-0	C20H16F3N7O2	5 mg

• Iripallidal, Iris pallida
  A bicyclic triterpenoid that exhibits anti-proliferative activity in a NCI 60 cell line screen with GI50 values from nanomolar to micromolar range. Binds to PKCα with high affinity. Also binds to RasGRP3. Induces phosphorylation of ERK1/2 in a RasGRP3-dependent manner.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221762	N/A	C31H50O4	1 mg/5 mg

• Isocarboxazid
  Monoamine oxidase inhibitor. Antidepressant.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218606	59-63-2	C12H13N3O2	100 mg

• Isodemecolcine
  An antimitotic agent that disrupts microtubles by binding to tubulin and preventing its polymerization. Stimulates the intrinsic GTPase activity of tubulin. Induces apoptosis in several normal and tumor cell lines and activates the JNK/SAPK signali

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-280855	4702-33-4	C21H25NO5	50 mg

• ITX 3
  A selective inhibitor of TrioN RhoGEF activity. Has been shown to inhibit TrioN-mediated GTP exchange on RhoG and Rac1, formation of TrioN-induced cellular structures in REF52 fibroblasts and NGF-mediated neurite outgrowth in PC12 cells in vitro.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295214	347323-96-0	C22H17N3OS	10 mg/50 mg

• IWR-1

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-252929	430429-02-0	C25H19N3O3	5 mg

• JAK2 Inhibitor III, SD-1029
  A cell-permeable xanthenedione compound that acts as a JAK2-selective inhibitor. Displays lower effect on the cellular phosphorylation levels of Jak1 and Src and shows little inhibition towards a panel of 49 other protein kinases in cell-free kinase assays. Effectively inhibits cell proliferation in JAK-activated BA/F3 cell lines as well as phosphorylation and nuclear translocation of cellular Stat3.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221773	N/A	C25H30Cl2N2O3 ·2HBr	10 mg

• JAK2 Inhibitor IV
  An aminoindazole compound that potently inhibits the activity of both the wild-type JAK2 and the constitutively active V617F mutant. Found in patients with clonal polycythemia vera, essential thrombocytosis, and chronic idiopathic myelofibrosis. Shows much reduced activity against JAK3.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221774	N/A	C17H20N4O2S	5 mg

• JAK2 Inhibitor V, Z3
  A cell-permeable pyridinylbutanone compound that inhibits cellular autophosphorylation of both Jak2 and the active V167F mutant.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221775	N/A	C23H24N2O	10 mg

• JAK3 Inhibitor V
  Inhibits STAT-5 phosphorylation and T-cell proliferation. A breakdown product of JAK3 Inhibitor-IV with similar inhibitory potency (pIC50 = 6.8 for JAK3; 5.0 for EGF-R; 4.7 for JAK1).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295218	4452-06-6	C13H10O	10 mg

• JLK 6
  Inhibitor of γ-secretase that selectively inhibits βAPP cleavage without affecting other γ-secretase-mediated pathways. Prevents recovery of Aβ40 and Aβ42 from HEK293 cell overexpressing wild-type or Swedish-mutated βAPP.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203612	62252-26-0	C10H8ClNO3	10 mg/50 mg

• JNJ 303

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361217	878489-28-2	C21H29ClN2O4S	10 mg/50 mg

• JTE 013

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203615	383150-41-2	C17H19N7OCl2	10 mg

• JZL 195

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-279248	N/A	C24H23N3O5	5 mg/10 mg

• Juglone
  Inhibits the transcription of RNA polymerase II by changing the sulfhydryl groups and blocking the assembly of the preinitiation complex.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202675	481-39-0	C10H6O3	1 g

• JZL184
  A strong and selective inhibitor of MAGL that displays IC₅₀ values of 8 nM and 4 µM for inhibition of MAGL and fatty acid amide hydrolase in murine brain membranes, respectively.1 JZL184 reduces MAGL activity by 85%, elevates brain 2-AG levels by 8-fold, and elicits analgesic activity in a variety of pain assays that qualitatively mimics direct central cannabinoid (CB1) agonists in mice.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-224031	1101854-58-3	C27H24N2O9	5 mg/10 mg

• K 858
  An ATP-uncompetitive mitotic kinesin Eg5 inhibitor, which does not effect microtubule dynamics.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-300856	72926-24-0	C13H15N3O2S	10 mg/50 mg

• KAD-1229 Calcium Hydrate
  Inhibitor of ATP-sensitive K⁺ channel activity in MIN 6 cells. Has also been shown to bind sulfonylurea receptors as well.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207776	207844-01-7	(C19H27NO4)2•Ca•2 ·H2O	10 mg

• Ketorolac

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-279250	74103-06-3	C15H13NO3	500 mg

• KF 38789
  Selective inhibitor of P-selectin-mediated cell adhesion (IC₅₀ = 1.97 μM) that displays no effects on L-selectin- and E-selectin-mediated adhesion. Blocks P-selectin-mediated binding in vitro and leukocyte accumulation in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203617	257292-29-8	C19H21NO5S	10 mg

• KM 11060
  Corrects F508del-CFTR trafficking; increases the amount of functional CFTR at the plasma membrane (~75%). Inhibits PDE5 activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204029	774549-97-2	C19H17Cl2N3O2S	10 mg/50 mg

• Ko 143
  Potent and selective breast cancer resistance protein multidrug transporter (BCRP) inhibitor (EC90 = 26 nM). Displays > 200-fold selectivity over P-gp and MRP-1 transporters. Increases intracellular drug accumulation and reverses BCRP-mediated multidrug resistance.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204030	461054-93-3	C26H35N3O5	1 mg/10 mg

• Kojic acid
  Tyrosinase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-255228	501-30-4	C6H6O4	5 g/10 g

• L-(-)-α-Methyldopa
  L-aromatic amino acid decarboxylase inhibitor. Antihypertensive.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203092	555-30-6	C10H13NO4	1 g

• L-4-Fluoro-phenyl-alanine
  Substrate for tyrosine hydroxylase that has been used to study the regulation of that enzyme. Substitution of p-fluorophenylalanine for phenylalanine in the culture medium inhibits mitosis and reversibly arrests HeLa cells in G2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207785	1132-68-9	C9H10FNO2	100 mg/500 mg

• L-5,5-Dimethylthiazolidine-4-carboxylic Acid
  Found to act on the cell membrane of tumor cells, possiblly causing a reverse transformation to normal cells through restoration of contact inhibition.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207786	72778-00-8	C6H11NO2S	500 mg

• L-690,330
  A bisphosphonate inhibitor of inositol monophosphate. Described to dose-dependently increase brain inositol(I)phosphate levels during cholinergic stimulation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202685	142523-38-4	C8H12O8P2	1 mg/5 mg

• L-Buthionine-(S,R)-Sulfoximine
  Potent and specific inhibitor of α-glutamylcysteine synthetase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218630	83730-53-4	C8H18N2O3S	1 g

• L-Phenylalaninol
  Inhibits ulcer formaiton by the reduction of gastric acid secretion.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204786	3182-95-4	C9H13NO	1 g/5 g

• L189
  A DNA ligase I, III and IV inhibitor (IC50 values are 5, 9 and 5 μM respectively) that blocks DNA binding (Ki = 5 μM for DNA ligase I). Shown to preferentially inhibits step 2 of the ligation reaction, and inhibits base excision repair (BER) and non-homologous end joining (NHEJ). Specifically sensitizes cancer cells to DNA damage and increases the cytotoxicity of DNA-damaging agents.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295349	64232-83-3	C11H10N4OS•xH2O	10 mg/50 mg

• Lansoprazole
  H⁺,K⁺-ATPase inhibitor that displays antisecretory and antiulcer activity. Inhibits gastric acid secretion.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203101	103577-45-3	C16H14F3N3O2S	250 mg/1 g

• (-)-Lentiginosine
  A selective and powerful amyloglucosidase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207824	125279-72-3	C8H15NO2	1 mg

• Leuhistin
  Inhibitor of aminopeptidase M.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202692	129085-76-3	C11H19N3O3	1 mg/5 mg

• Liarozole hydrochloride
  A hydrochloride salt preparation of Liarozole, which has been shown to inhibit cytochrome p-450-dependent metabolism of all-trans-retinoic-acid.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204055	145858-50-0	C17H13ClN4 ·HCl	10 mg/50 mg

• Limonin
  Bitter principle of citrus fruits. Chemically induced carcinogenesis inhibitor and HIV-1 replication inhibitor. Shows antinociceptive effect. Does not possess any inherent antioxidant activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204793	1180-71-8	C26H30O8	50 mg

• Lipase Inhibitor, THL
  A lipase inhibitor that interacts with the thioesterase domain of fatty acid synthase and results in cell apoptosis and a halt in cell proliferation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203108	96829-58-2	C29H53NO5	50 mg

• Liranaftate
  A squalene epoxidase inhibitor that is used as an antifungal agent.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207828	88678-31-3	C18H20N2O2S	10 mg

• Lisinopril
  A potent angiotensin-converting enzyme inhibitor that inhibits the formation of angiotensin I with an IC50 value of 1.2 nM (ovine).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205378	76547-98-3	C21H31N3O5	100 mg/500 mg

• Losartan Potassium
  A specific antagonist of the angiotensin II AT1 receptor. Blockade of angiotensin II-AT1 binding produces vasodilation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204796	124750-99-8	C22H22ClN6O.K	1 g/5 g

• Luffariellolide
  Structurally related to manoalide. Anti-inflammatory PLA₂ inhibitor. Less potent than manoalide, but partially reversible. Inhibits human recombinant sPLA₂ selectively over cPLA₂.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202212	111149-87-2	C25H38O3	1 mg

• LY 393558
  A dual 5-HT1B/1D receptor antagonist (pKB values are 9.05 and 8.98 respectively) and an 5-HT re-uptake inhibitor (pIC50 = 8.48). Has been shown to potently antagonize terminal autoreceptor activity in vitro and increase extracellular 5-HT levels above those evoked by fluoxetine in vivo. Also shown to act as an antagonist at 5-HT2A and 5-HT2B receptors (pKi values are 7.29 and 7.35 respectively).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295369	271780-64-4	C26H31FN4O4S2	10 mg/50 mg

• LY2183240
  A potent inhibitor of FAAH activity, and the uptake and enzymatic hydrolysis of anandamide (sc-205592).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200357	874902-19-9	C17H17N5O	10 mg/50 mg

• Lysyl Endopeptidase

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-360250	N/A	N/A	20 µg

• (+)-Madindoline A
  Madindolines are noncytotoxic indole alkaloids. (+)-Madindoline A (MadA; MDL-A) binds competitively but noncovalently to gp130 inhibiting downstream activation of the JAK/STAT pathway.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202702	184877-64-3	C22H27NO4	500 µg/1 mg

• MAZ51
  Inhibits vascular endothelial cell growth factor-C (VEGF-C)-induced intracellular phosphorylation of VEGFR-3 (Flt-4) (IC₅₀=1µM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202703	163655-37-6	C21H18N2O	2 mg

• MDL 72527
  A polyamine oxidase (POA) inhibitor. Does not inhibit monoamine oxidase or D-Amino acid oxidase. Has been shown to display anticancer and neuroprotective activity in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295375	93565-01-6	C12H20N2.2HCl	10 mg/50 mg

• MDM2 Inhibitor
  Cell-permeable boranyl-chalcone exhibiting strong binding to MDM2 and irreversibly disrupts MDM2/p53 protein complex. Expresses selective toxicity towards MDM2 overexpressing human breat cancer cell lines when compared to normal breast cell lines.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204072	562823-84-1	C15H12BIO3	10 mg

• MEDICA 16
  Hypolipidemic and antidiabetic agent. Inhibitor of citrate lyase and acetyl-CoA carboxylase, expected to disinhibit hepatic fatty acid oxidation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203131	87272-20-6	C20H38O4	5 mg

• MEK Inhibitor II
  A selectively potent MEK inhibitor, showing little effect on PKC and PKA. Inhibits Raf1 and ERK1, but only at much higher concentrations. Cell-permeable.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205745	623163-52-0	C14H8NO4Cl	5 mg

• Meloxicam sodium salt hydrate
  Has shown to abolish thymulin-induced increases of cytokines and NGF in the liver of rats and displays tumor growth suppression. May be capable of antagonizing cachexia in vitro. Non-steroidal anti-inflammatory drug (NSAID) that shows 300-fold selectivity for cyclooxygenase-2 (COX-2) vs cyclooxygenase-1 (COX-1).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215294	71125-39-8 (anhydrous)	C14H12N3NaO4S2•xH2O	100 mg

• Membrane Traffic Inhibitor, A5
  A piperazinyl compound which is cell-permeable, that has been reported to specifically block clathrin adaptor complex AP-1-dependent traffic between endosomes and trans-Golgi network (TGN) in budding yeast. Demonstrates little effect against other endosome and TGN trafficking pathways.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-353670	N/A	C17H24N2O•HCl	10 mg

• Metastin, Synthetic
  A KiSS-1 gene product with 54 amino-acid residues and a C-terminally amidated LRF-motif that acts as a metastasis inhibitor by G-protein-coupled receptors (GPCRs). It is reported to inhibit chemotaxis and invasion of hOT7T175-transfected CHO cells in vitro (IC50 = ₅₀ nM) and attenuates pulmonary metastasis of hOT7T175-transfected B16-BL6 melanomas in vivo. This is shown to be a potent and selective agonist of AXOR12 and hOT7T175 (a novel human GPCR). It induces an increase in intracellular Ca²⁺ levels in CHO/h175 and CHO/AXOR12:Gqi5 cells. It also binds to hOT7T175 with high affinity (K_ι = 340 pM, determined by competitive binding analysis).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221884	N/A	C258H401N79O78	250 µg

• Methantheline bromide

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-279310	53-46-3	C21H26BrNO3	10 mg

• Methyl α-Linolenyl Fluorophosphonate
  An analog of methyl arachidonyl fluorophosphonate (MAFP), which has been widely studied as an inhibitor of phospholipases, FAAH, and as a CB receptor ligand. The pharmacology of the α-linolenyl analog of MAFP has not been completely investigated.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221926	N/A	C19H34FO2P	1 mg/5 mg

• Methyl γ-Linolenyl Fluorophosphonate
  An analog of methyl arachidonyl fluozophosphonate (MAFP), which has been widely studied as an inhibitor of phospholipases, FAAH, and as a CB receptor ligand. The pharmacology of the γ-linolenyl analog of MAFP has not been completely investigated.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221932	N/A	C19H34FO2P	1 mg/5 mg

• Mildronate
  A pharmaceutical composition based on a reverse transcriptase inhibitor and meldonium.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207887	76144-81-5	C6H14N2O2	100 mg

• Moclobemide
  A reversible monoamine oxidase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207891	71320-77-9	C13H17ClN2O2	10 mg

• Moexipril hydrochloride
  Angiotensin-converting enzyme (ACE) inhibitor. Antihypertensive. Blocks degradation of bradykinin into inactive metabolites.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204095	82586-52-5	C27H34N2O7.HCl	10 mg/50 mg

• Moexiprilat Hydrate
  Analogue of Quinapril.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218866	103775-14-0	C25H30N2O7	5 mg

• Monastrol
  Cell permeable non-tubulin-interacting mitosis inhibitor. Blocks mitosis (IC₅₀=14µM) by binding to the mitotic kinesin Eg5.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202710	254753-54-3	C14H16N2O3S	1 mg/5 mg

• Monoacylglycerol Lipase Inhibitor, URB602
  Cell-permeable N-biphenyl carbamate that acts as a selective and non-competitive inhibitor of monoacylglycerol lipase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203141	565460-15-3	C19H21NO2	10 mg/50 mg

• MPP dihydrochloride
  Selective, high affinity silent antagonist at ERa receptors. Displays greater than 200-fold selectivity for ERa over ERb. Ki values are 2.7 and 1800 nM at ERa and ERb receptors respectively.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204098	289726-02-9	C29H31N3O3 ·2HCl	10 mg/50 mg

• MRK 560

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-363285	677772-84-8	C19H17ClF5NO4S2	10 mg/50 mg

• MRN-ATM Pathway Inhibitor, Mirin
  Shown to be a cell permeable compound that prevents MRN-dependent activation of ATM. Also reported to inhibit MRE11 which causes a reduction in the efficiency of nonhomologous end joining.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203144	299953-00-7	C10H8N2O2S	10 mg

• Mycalolide B
  A compound shown to inhibit actin polymerization (IC₅₀=10-50 nM), suppress actin-activated myosin Mg²⁺-ATPase activity and abolish both ADP and collagen-induced platelet aggregation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-358736	122752-21-0	C52H74N4O17	20 µg

• Myoseverin
  Microtubule-binding molecule that induces reversible fission of multinucleated myotubules into mononucleated fragments.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203146	267402-71-1	C24H28N6O2	1 mg

• Myoseverin B
  A new microtubule-binding molecule which acts reversibly on myoblast proliferation without the cytotoxic effects displayed by nonpurine-based microtubule-disrupting molecules, like taxol, vinblastine, nocodazole. It can be effectively used for inhibiting new vessel growth by inhibiting endothelial cell function and differentiation of progenitor cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215407	361431-27-8	C27H32N6O2	1 mg/5 mg

• N-([R,S]-2-Carboxy-3-Phenylropionyl)-L-Leucine
  Found to be a potent and specific inhibitor of enkephalinase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295509	102601-55-8	C16H21NO5	10 mg

• N-(1-Naphthalenylsulfonyl)-Ile-Trp-aldehyde
  Potent, reversible, and selective inhibitor of human cathepsin L (IC₅₀=1.9nM). Inhibits release of Ca²⁺and hydroxyproline from bone in vitro.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-221967	161709-56-4	C27H29N3O4S	1 mg/5 mg

• N-(2-Aminoethyl) Cyclopamine
  Cyclopamine derivative demonstrating teratogenic properties with reverse effects of oncogenic mutations.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207900	334616-31-8	C29H46N2O2	250 µg

• N-(2-Aminoethyl)-5-chloroisoquinoline-8-sulfonamide Dihydrochloride
  Found to have a potent inhibitory action against casein kinase 1 with respect to ATP and a much weaker effect on casein kinase 2 and other protein kinases.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218908	N/A	C11H14Cl3N3O2S	10 mg

• N-(2-Mercaptoethyl) Demecolcine
  An antimitotic agent which disrupts microtubles by binding to tubulin and preventing its polyerization. Stimulates the intrinsic GTPase activity of tubulin.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218920	1217746-74-1	C23H29NO5S	10 mg

• N-(2-Phenylethyl)indomethacin Amide
  An aromatic amide of indomethacin recently reported to be a potent and selective reversible inhibitor of COX-2. Inhibits human recombinant and ovine COX-2 with IC₅₀ of 0.06 μM and 0.125 μM, respectively.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218925	261766-32-9	C27H25ClN2O3	50 mg

• N-(3-Pyridyl)indomethacin Amide
  An aromatic amide of indomethacin recently reported to be a potent and selective reversible inhibitor of COX-2. Inhibits human recombinant COX-2 with IC₅₀ of 0.1 μM.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-218939	261755-29-4	C24H20ClN3O3	50 mg

• N-(4-Aminobutyl)-5-chloro-1-naphthalenesulfonamide Hydrochloride
  A neoplasm inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207913	78957-84-3	C14H18Cl2N2O2S	25 mg

• N-(4-Azidosalicyl)-6-amido-6-deoxy-glucopyranose
  Inhibits the labeling of the human erythrocyte monosaccharide transporter by [125I]IASA-glc more effectively that D-glucose.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207914	86979-66-0	C13H16N4O7	1 mg

• N-(4-Carboxy-3-hydroxyphenyl)maleimide
  Reported to be an irreversible inhibitor of LDH isoenzyme

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295580	19232-43-0	C11H7NO5	250 mg

• N-(6-Phenylhexyl)-5-chloro-1-naphthalenesulfonamide
  Activates protein kinase C in a Ca²⁺ -dependent manner via a mechanism similar to that of phosphatidylserine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-211996	102649-78-5	C22H24ClNO2S	25 mg

• N-(Methoxysuccinyl)-Ala-Ala-Pro-Val-chloromethyl ketone
  Inhibits human granulocyte elastase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215426	65144-34-5	C22H35ClN4O7	5 mg/10 mg

• N-[(4S)-4-amino-5-[(2-aminoethyl)amino]pentyl]-N'-nitroguanidine tris(trifluoroacetate) salt
  A potent and selective inhibitor of nNOS (neuronal nitric oxide synthase).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215427	357965-99-2	C14H24N7O8F9	5 mg/25 mg

• (+/-)-N-3-Benzylnirvanol
  A potent and selective human CYP2C19 inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-207943	93879-40-4	C18H18N2O2	10 mg

• N-Acetyl-2,3-dehydro-2-deoxyneuraminic Acid, Methyl Ester
  Bacterial, animal and viral sialidases inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219017	N/A	C12H19NO8	25 mg

• N-Acetyl-Asp-Glu-His-Asp-7-amido-4-methylcoumarin trifluoroacetate salt

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-301269	N/A	N/A	5 mg

• N-Acetyl-L-tyrosine ethyl ester monohydrate
  Widely employed substrate for the determination of the esterase activity of chymotrypsin

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-269703	36546-50-6	C13H17NO4•H2O	5 g

• N-Arachidonyl maleimide
  A highly potent and irreversible inhibitor of MAG lipase1 which covalently binds to a cysteine residue located near the fatty acid binding site2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205760	876305-42-9	C24H35NO2	5 mg/25 mg

• N-Carboxymethyl-Phe-Leu-OH
  A highly potent enkephalinase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-295684	81109-85-5	C17H24N2O5	100 mg/500 mg

• N-Deacetylcolchiceine
  Antimitotic agent disrupting microtubule action through the binding of tubulin and preventing polymerization. Has been shown to stimulate the intrinsic GTPase activity of tubulin. Induces apoptosis and activates the JNK/SAPK signals.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208016	3482-37-9	C19H21NO5	100 mg

• N-Deacetylcolchicine
  Antimitotic agent that intercepts microtubles by binding to tubulin and preventing its polymerization. Stimulates the intrinsic GTPase activity of tubulin. Induces apoptosis in several normal and tumor cell lines and activates the JNK/SAPK signal.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219099	3476-50-4	C20H23NO5	25 mg

• N-Desethyl Acetildenafil
  A pyrazolopyrimidinone derivative which acts as a cGMP phosphodiesterase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208022	147676-55-9	C23H30N6O3	2.5 mg

• N-Desmethyl Rosuvastatin Disodium Salt Monohydrate
  Inhibitor of the enzyme HMG-CoA reductase in vitro.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219129	N/A	C21H24FN3O6S ·2Na ·H2O	1 mg

• N-Ethyldeoxynojirimycin
  Inhibits HIV cytopathicity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222004	N/A	C8H17NO4··HCl	1 mg/5 mg

• N-Ethyldeoxynojirimycin Hydrochloride
  Thrombolytic derived from Moranoline wish activity as an HIV cytopathicity inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208035	210241-65-9	C8H17NO4•HCl	10 mg

• N-Ethylmaleimide
  An electrophilic small molecule, alkylates nucleophilic residues of proteins. Ablates the function of cysteine proteases and other enzymes employing active-site thiols.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202719	128-53-0	C6H7NO2	5 g

• N-Methyl Ritonavir Bicarbonate
  An analogue of the selective HIV protease inhibitor Ritonavir.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219181	N/A	C39H52N6O8S2	5 mg

• N-Methylaminogenistein

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-212240	359436-93-4	C16H13NO3	10 mg

• n-Octyl-Xanthate, Potassium Salt

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-212267	2720-80-1	C9H17KOS2	10 mg

• N-Oxalyl-D-alanine
  Cell permeable, potent competitive inhibitor of factor inhibiting HIF asparagine hydroxylase. But does not inhibit PHDs (prolyl hydroxylase domain-containing proteins; HIF-PHs).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222014	N/A	C5H9NO6	10 mg

• N-Oxalyl-L-alanine
  Cell permeable, competitive inhibitor of PHDs (prolyl hydroxylase domain-containing proteins; HIF-PHs). Less potent inhibitor of factor inhibiting HIF asparagine hydroxylase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205959	N/A	C5H7NO5•H2O	10 mg/50 mg

• N-Oxalylglycine
  A cell permeable α-ketoglutarate analogue that functions as a competitive inhibitor of prolyl 4-hydroxylase which hydroxylates proline-rich peptides in vitro.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202720	5262-39-5	C4H5NO5	10 mg/50 mg

• N-Trifluoroacetyl Deacetylcolchiceine
  An antimitotic agent that interrupts microtubles by binding to tubulin and preventing polymerization. Stimulates the intrinsic GTPase activity of tubulin. Apoptosis inducer in normal and tumor cell lines and activates the JNK/SAPK signaling.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219250	N/A	C21H20F3NO6	100 mg

• N-Trifluoroacetyl Deacetylcolchicine
  An antimitotic agent that interrupts microtubles by binding to tubulin and preventing polymerization. Stimulates the intrinsic GTPase activity of tubulin. Apoptosis inducer in normal and tumor cell lines and activates the JNK/SAPK signaling.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-358439	N/A	C22H22F3NO6	50 mg

• N-Trifluoroacetyl-N-methyl-deacetylcolchiceine
  An antimitotic agent that interrupts microtubles by binding to tubulin and preventing polymerization. Stimulates the intrinsic GTPase activity of tubulin. Apoptosis inducer in normal and tumor cell lines and activates the JNK/SAPK signaling.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219253	N/A	C22H22F3NO6	100 mg

• N-Trifluoroacetyl-N-methyl-deacetylcolchicine
  An antimitotic agent that interrupts microtubles by binding to tubulin and preventing polymerization. Stimulates the intrinsic GTPase activity of tubulin. Apoptosis inducer in normal and tumor cell lines and activates the JNK/SAPK signaling.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219254	N/A	C23H24F3NO6	250 mg

• MM 11253

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361255	345952-44-5	C28H30O2S2	10 mg/50 mg

• N-Trifluoroacetyliso Deacetylcolchicine
  An antimitotic agent that interrupts microtubles by binding to tubulin and preventing polymerization. Stimulates the intrinsic GTPase activity of tubulin. Apoptosis inducer in normal and tumor cell lines and activates the JNK/SAPK signaling.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219258	N/A	C22H22F3NO6	100 mg

• N1, N12-Diethylspermine·4HCl
  Antineoplastic activity. Inhibits polyamine synthesis1.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203442	113812-15-0	C14H34N4 ·4HCl	10 mg/50 mg

• N1,N11-Diethylnorspermine tetrahydrochloride
  Highly potent known inducer of the polyamine catabolic enzyme, spermidine/spermine N1-acetyltransferase (SSAT), able to increase enzyme activity 200-1000 fold.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204114	121749-39-1	C13H32N4.4HCl	10 mg/50 mg

• N2-Methyl-L-arginine
  Selective L-arginine uptake inhibitor (Ki = 500 μM). Inhibits uptake of arginine by the lysosomal system c in human fibroblast in vitro.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204115	2480-28-6	C7H16N4O2	10 mg/50 mg

• N744 tosylate
  An inhibitor of arachidonic acid-induced aggregation of tau proteins. N744 tosylate suppresses microsphere-mediated tau fibrillization via inhibiting the formation of filaments at the surface of microspheres.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215527	72616-22-9	C25H29N2O4S2 ·C7H7O3S	5 mg/25 mg

• Na+/H+ Exchanger Isoform-1 Inhibitor
  A cell-permeable acylguanidine compound that inhibits NHE-1-meidated pH recovery after acidosis in PS120 cells. Exhibits cardioprotective efficacy in both an isolated rat heart ischemia model in vitro and in a rat myocardial infarction model in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222035	N/A	C11H8N4OS ·CH3SO3H	5 mg

• MPEP hydrochloride

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-279454	96206-92-7	C14H11N ·HCl	50 mg/10 mg

• Nalidixic acid
  An inhibitor of bacterial DNA polymerase (DNA gyrase) and avian myeloblastoma virus reverse transcriptase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219324	389-08-2	C12H12N2O3	5 g/25 g

• Naltrindole Hydrochloride
  An apoptotic agent and a cell growth inhibitor. Also shown to be a highly potent and selective antagonist of δ opioids.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202236	111469-81-9	C26H26N2O3 ·HCl	5 mg

• Naphthofluorescein
  Inhibits the invasion of Matrigel by the human fibrosarcoma cell line, HT1080.1 The effects of this furin inhibitor on other furin-mediated processes, in vivo or in vitro, are still unknown.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205413	61419-02-1	C28H16O5	1 mg/5 mg

• Naringenin
  A flavonoid commonly found in grapefruits which functions as an antioxidant, free radical scavenger, anti-inflammatory compound, carbohydrate metabolism promoter, and immune system modulator.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219338	480-41-1	C15H12O5	25 g

• NBI-31772
  An insulin-like growth factor-1 binding proteins (IGFBPs) inhibitor; IGF-1 potentiator. NBI-31772 is an air/DMSO DOPA oxidation product, which inhibits IGF binding to IFGFB's by displacing IGF-1 from IGF1:IGFBP complex. Thus, it increases circulating level of IGF-1. NBI-31772 does not bind to IGFR.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-253181	374620-70-9	C17H11NO7	5 mg

• Nebularine
  A naturally occurring nucleoside, which inhibits mouse Sarcoma 180 and mycobacteria. This universal base can bind to all four of the nucleosides of DNA.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208087	550-33-4	C10H12N4O4	250 mg

• Neridronate
  A bone resorption inhibitor. It is used to treat Osteogenesis Imperfecta.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-253184	79778-41-9	C6H17NO7P2	10 mg

• Neridronate, Sodium Salt
  A biphosphonate bone resorption inhibitor. Used as a treatment for osteogenesis imperfecta.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219351	N/A	C6H16NNaO7P2	10 mg

• NF 340

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361274	N/A	C37H26N4Na4O15S4	10 mg/50 mg

• NF 449
  A selective Gsα-subunit G-protein antagonist which reduces the association rate of guanosine 5'-[γ-thio]triphosphate ([35S]GTP[γS]) binding to G_{α s} -s (Gs&alpha-s) and inhibits the stimulation of adenylyl cyclase activity in S49 cyc- membranes.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203159	389142-38-5	C41H24N6O29S8 ·8Na	10 mg

• NF007
  "Half-molecule" of NF023. Essentially inactive as a G-protein inhibitor and therefore can be used as a negative control.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222064	N/A	C17H12N2O12S3	10 mg

• NFAT Activation Inhibitor III
  A potent and selective inhibitor of calcineurin-NFAT signaling that does not effect calcineurin activity or calcineurin’s downstream signaling,

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203160	3519-82-2	C20H12O2	5 mg

• NFPS
  Non-transportable inhibitor of GlyT1. Displays no activity on GlyT2 or the transport of GABA, Glu, or Pro. Enhances amplitude of NMDA component of glutamatergic EPSCs.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204126	405225-21-0	C24H24FNO3	10 mg/50 mg

• Nilvadipine
  Antianginal and antihypertensive compound.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215567	75530-68-6	C19H19N3O6	50 mg

• Nisoldipine
  A dihydropyridine calcium channel blocker. Antihypertensive and antianginal.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-212396	63675-72-9	C20H24N2O6	250 mg

• Nitrogenistein

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208101	39679-60-2	C15H9NO5	10 mg

• Nomilin
  a natural product isolated from grapefruit seed and varying Citrus fruits with activity as an inducer of Phase II detoxifying enzymes and inhibitor of chemically induced carcinogenesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203163	1063-77-0	C28H34O9	25 mg/100 mg

• NPC-15437 dihydrochloride hydrate
  A selective inhibitor of protein kinase C.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215587	141774-20-1 (anhydrous)	C25H50N4O2•2HCl•xH2O	5 mg/25 mg

• NPS 2143 hydrochloride

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361280	284035-33-2	C24H25ClNO2.HCl	10 mg/50 mg

• NS 2028
  Potent, specific, and irreversible inhibitor of soluble guanylyl cyclase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202743	204326-43-2	C9H5BrN2O3	5 mg

• NSC 109555 ditosylate
  Reversible ATP-competitive Chk2 inhibitor, displaying no effect on a range of other kindases, including Chk1. Inhibits H1 phosphorylation, attenuates mitochondrial ATP synthesis. Displays antiproliferative activity in numeral leukemias in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204137	15427-93-7	C33H40N10O7S2	10 mg/50 mg

• NSC 632839 hydrochloride
  Inhibitor of ubiquitin isopeptidase activity that displays no effect on the proteolytic activity of the proteasome. Induces apoptosis via a Bcl-2-dependent and apoptosome-independent pathway of caspase activation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204138	157654-67-6	C21H21NO.HCl	10 mg/50 mg

• NSC 66811
  A potent MDM2 inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-311507	6964-62-1	C23H20N2O	10 mg/50 mg

• NSCI
  A selective inhibitor of nonpeptide caspase 3.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215590	872254-32-5	C26H25N3O6S	5 mg/25 mg

• NVP DPP 728 dihydrochloride
  Orally active DPP-IV inhibitor. Displays >15,000 fold selectivity over DPP-II anda range of Pro-cleaving proteases. Displays antidiabetic activity in vivo. Shown to improve Glc tolerance, increase GLP-1 and Insuling levels, augments insulin secretion and GLUT-2 levels, and preserves islet size.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204141	247016-69-9	C15H18N6O•2HCl	10 mg/50 mg

• O-Methylviridicatin
  3-O- methylviridicatin is a strong inhibitor of TNFα-induced replication of HIV.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202255	6152-51-4	C16H13NO2	1 mg

• o-Phenanthroline
  Metal chelating agent that prevents induction of chromosomal aberrations in streptozotocin-treated cells. Acts as a general matrix metalloproteinase inhibitor. Can be used as a photometric reagent for iron.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202256	5144-89-8	C12H8N2 ·H2O	500 mg

• Okadaol
  An analogue of okadaic acid (carboxyl group reduced to an alcohol). Has protein phosphatase inhibitory activity approximately 40% that of okadaic acid.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215623	131959-12-1	C44H70O12	25 µg/50 µg

• Oligomycin A
  An inhibitor of mitochondrial ATPases (F₁F₀) bound to the cell membrane.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201551	579-13-5	C45H74O11	5 mg/25 mg

• OMDM-2
  Metabolically stable, potent inhibitor of cellular anandamide uptake (neuronal (C6 glioma cells): IC₅₀=3.2µM; non-neuronal (rat RBL-2H3 cells): IC₅₀=17µM) with negligible effects on CB1 receptor (CB1: K_i=5.1µM; CB2: K_i>10µM), TRPV1 (EC₅₀=10µM) and FAAH (IC₅₀>100µM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204145	N/A	C27H45NO3	5 mg

• Omeprazole
  Cell-permeable, selective proton pump inhibitor. Acts as prodrug by undergoing acid-catalyzed rearrangement to a thiol-reactive cationic sulfenamide that inhibits (H⁺-K⁺)-ATPase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202265	73590-58-6	C17H19N3O3S	50 mg

• Ophiobolin C
  A phytotoxic metabolite from the ophiobolin class produced by many species of the genus Bipolaris. Studies suggest that Ophiobolin C inhibits CCR5 binding to the envelop protein gp120 and CD4, which is responsible for mediating the entry of HIV-1 into cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202268	19022-51-6	C25H38O3	1 mg

• OR-486
  Catechol-O-methyl transferase inhibitor

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204149	7659-29-2	C6H4N2O6	50 mg

• Oxcarbazepine
  A second-generation antiepileptic drug. Inhibits CYP2C19 and induces CYP3A4 and CYP3A5 systems. Studies suggest that the anticonvulsant activity of oxcarbazepine is mediated via the blocking of neuronal ion channels.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204826	28721-07-5	C15H12N2O2	10 mg

• Oxybutynin Chloride
  This compound inhibits proliferation and supresses gene expression in bladder smooth muscle cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208141	1508-65-2	C22H32ClNO3	2.5 g

• Ozagrel hydrochloride hydrate
  An selective inhibitor of thromboxane A2 synthase (TXA2).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215645	78712-43-3	C13H12N2O2•HCl•xH2O	5 mg/25 mg

• P32/98
  A specific, competitive transition-state substrate analog inhibitor of CD26 (dipeptidyl peptidase IV, DPPIV).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201305	136259-20-6	C9H18N2OS ·1/2C4H4O4	10 mg/50 mg

• Pamidronic Acid
  A biphosphonate bone resorption inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219549	40391-99-9	C3H11NO7P2	100 mg

• Paraoxon
  Cholinesterase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208151	311-45-5	C10H14NO6P	1 g

• Patulin
  A mycotoxin that has been reported to contain antibiotic characteristics. Also shown to specifically inhibit Na⁺-K⁺ ATPase activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204833	149-29-1	C7H6O4	1 mg/5 mg

• PD 123319 ditrifluoroacetate
  Potent, selective non-peptide angiotensin AT2 receptor antagonist. Tested on rat adrenal tissue and brain.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204835	130663-39-7	C31H32N4O3 ·2CF3CO2H	10 mg/50 mg

• Pemetrexed Disodium
  An antineoplastic, multitargeted antifolate which inhibits thymidylate synthase as well as other folate dependent enzymes.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219564	150399-23-8	C20H19N5Na2O6	10 mg

• Pentostatin
  Adenosine deaminase inhibitor. Anticancer agent.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204177	53910-25-1	C11H16N4O4	10 mg/50 mg

• Perindopril
  A potent angiotensin converting enzyme inhibitor used for antihypertensive therapy.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205799	82834-16-0	C19H32N2O5	100 mg/250 mg

• Perindopril t-Butylamine Salt
  An angiotensin-converting enzyme (ACE) inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208159	107133-36-8	C23H43N3O5	10 mg

• Perindoprilat
  An active metabolite of Perindopril, an angiotensin converting enzyme (ACE) inhibitor, which modulates the activity of Low density lipoprotein receptor-related protein (LRP).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208160	95153-31-4	C17H28N2O5	5 mg

• PF 915275
  Potent and selective 11β-hydroxysteroid dehydrogenase type 1 (11βHSD1) inhibitor (K_i = 2.3 nM) that displays little activity at 11βHSD2 (1.5% inhibition at 10 μM). Inhibits the conversion of prednisone to prednisolone in human hepatocytes in vitro (EC₅₀ = 15 nM). Orally active and has antidiabetic activity in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204182	857290-04-1	C18H14N4O2S	10 mg/50 mg

• Phalloidin Oleate
  A semi-synthetic derivative of Phalloidin (sc-202763) that is about 100-fold more cell-permeable than Phalloidin with similar acting binding properties.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222153	N/A	C53H80N8O12S	200 µg

• Phenoxymethylpenilloic Acid
  A reversible competitive inhibitor of Penicillinase, β-Lactamase 1.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208165	4847-29-4	C15H20N2O4S	10 mg

• Phosphoramidon, Disodium Salt
  Inhibits some metalloendopeptidases. Highly specific inhibitor of thermolysin. Inhibits the conversion of big endothelin-1 to endothelin (IC₅₀ = 4.6 µM). Effective concentration: 1-10 µM.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222168	N/A	C23H32N3O10P•2Na	5 mg

• Pimprinine
  Indole alkaloid produced by many species of Streptomyces. Inhibitor of monoamine oxidase and has shown antiepileptic effects. Inhibited tremorine-induced tremors and analgesia in mice.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202288	13640-26-1	C12H10N2O	1 mg

• Pirlindole mesylate
  A highly selective reversible inhibitor of monoamine oxidase type A.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203664	60762-57-4	C15H18N2•CH3SO3H	10 mg/50 mg

• Plumbagin from Plumbago indica
  Exhibits cytotoxicity in rodent models of carcinogenesis and carcinoma; has antifungal, antiviral, and antibacterial action.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-253283	481-42-5	C11H8O3	100 mg/250 mg

• Polydatin
  The glycoside of Resveratrol (sc-200808) originally isolated from the Chinese herb Polygonum cuspidatum. The compound has been shown to inhibit platelet aggregation and elevate the ratios of LDL-C/HDL-C and TC/HDL-C.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203203	65914-17-2	C20H22O8	10 mg

• Polyglutamine Aggregation Inhibitor III, C2-8
  Cell-permeable amidosulfonamide inhibitor of polyglutamine (polyQ)-aggregation in Huntington's disease (HD). Suggested to block the polymerization step of the polyQ aggregation

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202766	300670-16-0	C19H14Br2N2O3S	10 mg

• Polyglutamine Aggregation Inhibitor, PGL-135
  A cell-permeable benzothiazole compound that binds to polyglutamine (polyQ)-containing β-sheet structures and prevents polyQ-aggregation, a pathological hallmark of Huntington's disease (HD) and related glutamine repeat disorders.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204207	26278-83-1	C9H10N2OS ·HCl	10 mg

• Polyglutamine Aggregation Inhibitor, PGL-137
  A cell-permeable benzothiazole compound that binds to polyglutamine (polyQ)-containing β-sheet structures and acts as a polyQ-aggregation inhibitor of Huntington's disease (HD). Shown to be non-toxic and prevent HDQ51 (flag-tagged HD exon 1 protein with 51 glutamines)-aggregation in 293 Tet-Off (293 tetracycline-off) cells with an IC₅₀ of ~ 100 µM.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204208	943-04-4	C9H10N2OS	10 mg

• POM 1
  A polyoxotungstate that inhibits CD39, CD39L1, CD39L3 (nucleoside-triphosphate-diphosphohydrolases) and blocks the breakdown of ATP activated by IP.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203205	12141-67-2	Na6O39W12 ·H2O	50 g

• PPACK
  A potent and irreversible inhibitor of thrombin; reported to inhibit thrombin activation of progelatinase A.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201291	71142-71-7	C21H31ClN6O3	5 mg/25 mg

• PPARg Antagonist III, G3335
  A cell-permeable dipeptide that acts as a selective and reversible PPARγ antagonist. Shown to inhibit the agonist activity of Rosiglitazone in a dose-dependent manner in transfected COS-7 cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202771	36099-95-3	C16H19N3O5	50 mg

• Pravastatin 1,1,3,3-Tetramethylbutylamine
  A new salt of HMG-CoA reductase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208182	151006-14-3	C31H55NO7	25 mg

• Pravastatin, Sodium Salt
  A water-soluble, competitive 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) reductase inhibitor that potently blocks in vivo cholesterol synthesis (K_i ~1 nM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203218	81131-70-6	C23H35O7.Na	25 mg

• Probenecid
  Inhibitor of several ABC-transporters of the subfamily ABCC or MRP (multidrug resistant associated protein).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202773	57-66-9	C13H19NO4S	1 g/5 g

• Propentofylline
  A c-AMP phosphodiesterase inhibitor, a nerve growth factor stimulator, an adenosine transport inhibitor and a non-selective adenosine receptor antagonist. Nootropic.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208188	55242-55-2	C15H22N4O3	25 mg

• Proscillaridin A
  A cardiac glycoside which functions as a specific Na⁺/K⁺-ATPase inhibitor. It is reported that at high concentrations, above 300nM, Proscillaridin A can increase intracellular Ca²⁺ concentration, activate caspase-3 and induce apoptosis in human fibroblasts.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202775	466-06-8	C30H42O8	5 mg

• Protein Arginine N-Methyltransferase Inhibitor, AMI-1
  A cell-permeable, symmetrical sulfonated urea compound that acts as a potent, specific and non-AdoMet (S-adenosyl-L-methionine, SAM)-competitive inhibitor of protein arginine N-methyl transferases with minimal effect on lysine methyl transferases. Inhibits nuclear receptor reporter gene activation in MCF-7 cells, and HIV-1 RT polymerase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222202	N/A	C21H12N2Na4O9S2	5 mg

• Protein Synthesis Initiation Inhibitor, NSC 119889
  A cell-permeable, xanthenyl compound that prevents mRNA-ribosome interaction and inhibits 5'-mediated/cap-dependent initiation of protein synthesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222203	N/A	C20H8Br4O5	25 mg

• Protopanaxatriol
  May be an inhibitor of the uptake of glucose.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204866	34080-08-5	C30H52O4	5 mg/10 mg

• PSB 06126
  Nucleoside triphosphate diphosphohydrolase 3 (NTPDase 3) inhibitor. Reported to inhibit rat NTPDase 3 at low micromolar concentrations and display selectivity over NTPDase 1 and NTPDase 2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204215	N/A	C24H15N2NaO5S	10 mg/50 mg

• PSB 069
  Non-selective nucleoside triphosphate diphosphohydrolase (NTPDase) inhibitor. Reported to inhibit rat NTPDases 1, 2 and 3 with similar potencies.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204216	N/A	C20H12N2O5ClSNa	10 mg/50 mg

• PSC 833

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361298	121584-18-7	C63H111N11O12	1 mg

• Purpurin
  A xanthine oxidase inhibitor that inhibits azoxymethane-induced aberrant crypt foci in the rat.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205822	81-54-9	C14H8O5	5 g/25 g

• Pyridostigmine bromide
  An inhibitor of acetylcholinesterase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-212607	101-26-8	C9H13BrN2O2	1 g/5 g

• Pyripyropene A
  Highly specific inhibitor of acyl-coenzyme A:cholesterol acetyltransferase 2 (ACAT2)

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202302	147444-03-9	C31H37NO10	500 µg

• Pyrroloquinoline quinone
  A cofactor of microbial quinoprotein enzyme, and imidazopyrroline. A redox/cofactor found in a a class of enzymes called quinoproteins.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-210178	72909-34-3	C14H6N2O8	1 mg

• QS 11

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361301	944328-88-5	C36H33N5O2	10 mg/50 mg

• Quinapril Hydrochloride
  A firmly established and well tolerated angiotensin-converting enzyme inhibitor that attenuates the myocardial infarction induced rise in cardiac cytokine expression. Clinical trials show that quinapril prevents restenosis after coronary stenting in patients with angiotensin-coverting enzyme D allele.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205829	82586-55-8	C25H31ClN2O5	100 mg/500 mg

• R-(+)-Etomoxir
  An inhibitor of carnitine palmitoyltransferase A (CPT1), which is required for the oxidation of long-chain acyl CoA esters. Also a strong inhibitor of mitochondrial CPT1 and a candidate as an anti-diabetic drug.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208201	124083-20-1	C17H23ClO4	5 mg

• R-(+)-Etomoxir Carboxylate, Potassium Salt

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219696	132308-39-5	C15H8ClKO4	5 mg

• R-(+)-Tolterodine
  A muscarinic receptor antagonist which is used in the treatment of urinary incontinence.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-212626	124937-51-5	C22H31NO	5 mg

• (R,S)-Equol
  Flavonoid. Racemic mixture. Inhibits 12-O-tetradecanoylphorbol 13-acetate (TPA)-induced neoplastic cell transformation by targeting the MEK/ERK/p90RSK/activator protein-1 signaling pathway.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202307	94105-90-5	C15H14O3	5 mg/25 mg

• (R)-Lisinopril Sodium Salt
  R,S,S-Isomer of Lisinopril.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-212648	85955-59-5	C21H31N3NaO5	1 mg

• (R)-(-)-2,2-Dimethyl-1,3-dioxolane-4-methanol
  A MEK inhibitor

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219717	14347-78-5	C6H12O3	1 g

• (R)-(-)-Ibuprofen (S)-(+)-Lysinate
  A nonsteroidal anti-inflammatory drug (NSAID). Optically active, selective cyclooxygenase inhibitor (IC₅₀=14.9μM), that inhibits PGH synthase-1 and PGH synthase-2 with equal potency.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219722	N/A	C19H32N2O4	10 mg

• (R)-(-)-N-3-Benzylnirvanol
  A potent and selective human CYP2C19 inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208219	790676-41-4	C18H18N2O2	5 mg

• (R)-(+)-Acenocoumarol
  A short-lived oral anti-coagulant, which functions by inhibiting vitamin K epoxide reductase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205484	66556-77-2	C19H15NO6	1 mg/5 mg

• (R)-(+)-Blebbistatin
  Inactive enantiomer of the selective inhibitor of myosin II, (±)-blebbistatin.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204225	N/A	C18H16N2O2	1 mg

• (R)-(+)-Blebbistatin O-Benzoate
  Derivative of Blebbistatin, which is a compound that blockes myosin II-dependent cell processes.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219729	N/A	C25H20N2O3	5 mg

• (R)-2-Isopropyl-3,6-dimethoxy-2,5-dihydropyrazine
  An inhibitor with anti-tumor activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219735	109838-85-9	C9H16N2O2	100 mg

• (R)-Omeprazole Sodium Salt
  The R-Form of Omeprazole. Acts as a gastric proton-pump inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208250	161796-77-6	C17H19N3NaO3S	1 mg

• (R)-Oxybutynin Chloride
  The optically active inhibitor of proliferation and it also suppresses gene expression in bladder smooth muscle cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-219762	N/A	C22H32ClNO3	100 mg

• Rabeprazole Sodium Salt
  A partially reversible gastric proton pump inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208255	117976-90-6	C18H20N3NaO3S	10 mg

• rac Atomoxetine Hydrochloride
  A derivative of Tomoxetine.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-212721	82857-40-7	C17H22ClNO	5 mg

• rac Kainic Acid
  A neuroexcitatory chemical that is selective for the kainic acid receptor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-212731	73209-05-9	C10H15NO4	1 mg

• rac-Sitagliptin
  A trizolopyrazine dipeptidyl peptidase IV inhibitor (DPP-4). DPP-4 is an enzyme which breaks down incretins such as GLP-1, GIP, and gastrointestinal hormones.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208294	823817-56-7	C16H15F6N5O	1 mg

• Racecadotril
  A potent enkephalinase inhibitor which exhibits selective antisecretory activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205831	81110-73-8	C21H23NO4S	100 mg/500 mg

• Raltegravir Potassium Salt
  A potent human immunodeficiency virus (HIV) integrase inhibitor and a novel anti-AIDS drug.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208296	871038-72-1	C20H20FKN6O5	1 mg

• Ramipril
  An inhibitor of the angiotensin- converting enzyme (ACE) that is reported to quickly hydrolyze into the active metabolite Ramiprilat, after absorption.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205833	87333-19-5	C23H32N2O5	500 mg/1 g

• Ras/Rac Transformation Blocker, SCH 51344
  A cell-permeable pyrazoloquinoline compound that acts as an effective blocker of Ras-induced malignant transformation and inhibits Ras/Rac-dependent dissociation of EMS1 from the actin-myosin II complex and membrane ruffling. The effect of SCH 51344 is limited to Ras/Rac pathway(s) other than those involving ERK and JNK.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204231	171927-40-5	C16H20N4O3	10 mg

• Rasagiline Mesylate
  An antiparkinsonian. A selective irreversible MAO-B inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-206071	161735-79-1	C13H17NO3S	25 mg/100 mg

• Resibufogenin
  Specific Na⁺/K⁺-ATPase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202788	465-39-4	C24H32O4	10 mg

• Reversine
  Cell-permeable, 2,6-disubstituted purine analog that acts as a dedifferentiation-inducing agent.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203236	656820-32-5	C21H27N7O	5 mg

• Rhapontigenin
  A natural analog of resveratrol with antioxidant and anti-cancer activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-296263	500-65-2	C15H14O4	1 mg/5 mg

• Rho Kinase Inhibitor II
  A pyridyl urea compound that acts as a potent, selective, and ATP-competitive inhibitor of Rho-associated protein kinase (ROCK). Displays little activity towards Erk, PKA, PKC, PDGFR, or c-Kit/SCFR.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222253	N/A	C12H8Cl3N3O	5 mg

• Risedronate sodium
  A pyridinyl biphosphonate which inhibits osteoclast-mediated bone resorption.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204880	115436-72-1	C7H10NO7P2 • Na	100 mg

• Ro 08-2750
  Inhibitor of NGF-induced apoptosis. At submicromolar concentrations, inhibits binding selectively to p75NTR. At higher concentrations, inhibits binding selectively to P75NTR and TrkA. In SK-N-MC cells, prevents NGF-induced apoptosis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203682	37854-59-4	C13H10N4O3	1 mg/10 mg

• Ro 23-9358
  A Diacylglycerol lipase inhibitor which is an anti-obesity drug target.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215815	153125-17-8	C30H51NO6	5 mg/25 mg

• Ro 26-4550 trifluoroacetate
  Competitive reversible inhibitor of interleukin-2 (IL-2) binding to its receptor (IC₅₀ = 3 μM for inhibition of IL-2 interaction with IL-2R α-subunit). Appears to compete with IL-2Rα for its binding site on IL-2.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204888	193744-04-6	C28H31F3N4O5	10 mg

• Ro 41-1049 hydrochloride
  A selective, reversible, orally active inhibitor of MAO-A.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215816	127500-84-9	C12H12FN3OS•HCl	100 mg

• Ro 61-8048
  Potent and competitive kynurenine 3-hydroxylase inhibitor (K_i = 4.8 nM, IC₅₀ = 37 nM). Increases kynurenic acid levels to concentrations that antagonize the glycine site of NMDA receptors. Brain penetrant and exhibits antidystonic, anticonvulsant and neuroprotective activities.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204240	199666-03-0	C17H15N3O6S2 ·xH2O	10 mg/50 mg

• Ro 64-5229

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361308	N/A	C17H19Cl2N3O	10 mg/50 mg

• Roflumilast
  An antiasthmatic in treatment of chronic obstructive pulmonary disease. Selective phosphodiesterase 4 (PDE4) inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208313	162401-32-3	C17H14Cl2F2N2O3	5 mg

• Rotenone
  A mitochondrial electron transport inhibitor, which specifically inhibits NAD-linked substrate oxidation of NADH dehydrogenase with an EC50=10pmol/mg.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203242	83-79-4	C23H22O6	1 g

• RS 102895
  CCR2-selective chemokine receptor antagonist (IC50 values are 0.36 and 17.8 μM for inhibition of human recombinant CCR2b and CCR1 receptors respectively). Blocks MCP-1-stimulated calcium influx and chemotaxis with IC₅₀ values of 32 nM and 1.7 μM respectively. Inhibits α1A, α1D and 5-HT1A receptors.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204243	300815-41-2	C21H21F3N2O2 ·HCl	10 mg/50 mg

• RS 504393
  A CCR2 chemokine receptor antagonist, shown to also inhibit MCP-1 chemotaxis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204245	300816-15-3	C25H27N3O3•xH2O	10 mg

• RU 28318, potassium salt
  Potent, selective mineralocorticoid receptor antagonist. Selectively decreases ex-vivo MR binding in hippocampi of adrenalectomised rats. Inhibits aldosterone production and secretion. Induces hypotensive nature in female rats following central administration in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204250	76676-34-1	C25H37O4K•xH2O	10 mg/50 mg

• RSC-3388
  A pyrrolidine derivative which functions as an inhibitor of cytosolic phospholipase A2α. Useful in suppressing the production of prostaglandin E₂ in the human acute monocytic leukemia cell line THP-1.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-296281	337307-06-9	N/A	500 µg/1 mg

• RWJ 50271

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-362792	162112-37-0	C18H17F3N4O2S	10 mg/50 mg

• S-(-)-Tolterodine
  A muscarinic receptor antagonist which is used in the treatment of urinary incontinence.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-212799	124937-53-7	C22H31NO	5 mg

• S-(+)-Etomoxir
  An inhibitor of carnitine palmitoyltransferase A (CPT1), which is required for the oexidation of long-chain acyl CoA esters. A strong inhibitor of mitochondrial CPT1 and is a candidate as an anti-diabetic drug.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220002	828934-40-3	C17H23ClO4	5 mg

• (S)-(-)-Blebbistatin
  Selective inhibitor of myosin II. Active enantiomer. Inhibits contraction of cleavage furrow sans disruption of mitosis or of the contractile ring assembly. Rapid and reversible blocking of cell blebbing, as well as disruption of directed cell migration and of cytokinesis in vertebrate cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204253	856925-71-8	C18H16N2O2	1 mg

• (S)-(-)-Blebbistatin O-Benzoate
  A derivative of Blebbistatin, a compound that blockes myosin II-dependent cell processes.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220036	N/A	C25H20N2O3	10 mg

• (S)-(+)-Ibuprofen (S)-(+)-Lysinate
  A nonsteroidal anti-inflammatory drug (NSAID). Optically active, selective cyclooxygenase inhibitor (IC₅₀=14.9μM). Inhibits PGH synthase-1 and PGH synthase-2 with comparable potency.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220042	N/A	C19H32N2O4	10 mg

• (S)-(+)-N-3-Benzylnirvanol
  Potent and selective human CYP2C19 inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220043	790676-40-3	C18H18N2O2	5 mg

• (S)-(+)-α-Fluoromethylhistidine Dihydrochloride
  A histidine carboxylase inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220045	N/A	C7H12Cl2FN3O2	500 µg

• (S)-(−)-Acenocoumarol
  Acenocoumarol is a short-lived oral anti-coagulant, which functions by inhibiting vitamin K epoxide reductase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205501	66556-78-3	C19H15NO6	1 mg/5 mg

• (S)-N-[1-(4-Cyclopropylmethyl-3,4-dihydro-2H-benzo[1,4]oxazin-6-yl)-ethyl]-3-(2-fluoro-phenyl)acrylamide
  A potent and efficacious KCNQ2 opener that inhibits induced hyperexcitability of rat, hippocampal neurons.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-212889	697287-41-5	C23H25FN2O2	1 mg

• (S)-Oxybutynin Chloride
  The optically avtice inhibitor of proliferation and supresses gene expression in bladder smooth muscle cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220080	N/A	C22H32ClNO3	100 mg

• Sandoz 58-035
  An inhibitor of Acyl-CoA cholesterol acyltransferase (ACAT).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215839	78934-83-5	C30H47NOSi	5 mg/25 mg

• Sanguinarine chloride
  Na⁺/K⁺-and Mg²⁺-ATPase inhibitor. Antimicrobial, anti-inflammatory and antioxidant properties. Induces apoptosis. Modulates the Bcl-2 family.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202800	5578-73-4	C20H14NO4Cl	5 mg

• (Sar1,Gly8)-Angiotensin II
  Part peptide (Sar-Arg-Val-Tyr-Ile-His-Pro-Gly) Acetate Salt Inhibitor of Angiotensin II.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-296370	100900-29-6	C44H69N13O12	1 mg/5 mg

• SB 218078
  Phosphorylation product of inositol-trisphosphate (Ins P3). A potent inhibitor of Ins P3 5-phosphatase (IC₅₀ ~150 nM); facilitates Ca²⁺ influx by sensitising Ins P3-mediated activation of ICRAC. At higher concentrations, it acts as an inhibitor of Ins P3 receptors.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203692	135897-06-2	C24H15N3O3	1 mg

• SB 225002
  A selective non-peptide CXCR2 inhibitor which suppresses IL-8 induced neutrophil chemotaxis and margination.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202803	182498-32-4	C13H10BrN3O4	1 mg/5 mg

• SB 242084

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361338	181632-25-7	C21H19ClN4O2.2HCl	10 mg/50 mg

• SB 258719 hydrochloride

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361340	195199-95-2	C18H30N2O2S.HCl	10 mg/50 mg

• SB 265610

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361341	211096-49-0	C14H9BrN6O	1 mg/10 mg

• SB 271046 hydrochloride

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361343	209481-20-9	C20H22CIN3O3S2.HCl	10 mg/50 mg

• SB 328437
  A highly potent and selective CC chemokine receptor-3 (CCR3) antagonist. Inhibits calcium mobilization induced by eotaxin, eotaxin-2, or MCP-4. Also inhibits eotaxin, eotaxin-2, and MCP-4-mediated chemotaxis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222292	247580-43-4	C21H18N2O5	1 mg

• SB 431542
  A small molecule that acts as a specific and selective inhibitor of TGF-β superfamily type I ALK receptors ALK4, 5, and 7.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204265	301836-41-9	C22H16N4O3	1 mg/10 mg

• SB 612111 hydrochloride
  A piperidine derivative shown to act as a selective NOP receptor antagonist

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361347	371980-98-2	C24H29Cl2NO•HCl	10 mg/50 mg

• SB 657510

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361348	474960-44-6	C19H22BrCIN2O5S	10 mg/50 mg

• SB-415286
  Active enantiomer of ketoprofen1. Inhibits cyclooxygenase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204901	264218-23-7	C16H10ClN3O5	1 mg/5 mg

• SC 57461A
  Potent and selective inhibitor of LTA4 hydrolase. Does not inhibit other enzymes of the arachidonic acid cascade including COX-1, COX-2, LTC4 synthase and 5-lipoxygenase. Potently inhibits LTB4 production in whole blood (IC₅₀ = 49 nM). Orally active.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204266	423169-68-0	C20H25NO3.HCl	10 mg/50 mg

• SCH 28080
  Potent inhibitor of H⁺,K⁺-ATPase (IC₅₀ = 20 nM); binds to the K⁺ recognition site and is competitive with respect to K⁺. Inhibits gastric acid secretion in vitro and in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204269	76081-98-6	C17H15N3O	10 mg/50 mg

• Sch 58053
  Ezetimibe analog and intestinal lymphatic cholesterol transporter inhibitor (potent, rapid, and selective)

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208384	194423-53-5	C26H23ClFNO3	2.5 mg

• SCH-202676 hydrobromide
  This product is a G protein-coupled receptor allosteric modulator shown to inhibit agonist and antagonist binding to G protein-coupled receptors.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200835	70375-43-8	C15H13N3S··HBr	10 mg/50 mg

• Sclerotiorin
  Inhibits soybean lipoxygenase-1, cholesterol ester transfer protein, Grb2-Shc interaction and antagonism of endothelin receptors.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205505	549-23-5	C21H23ClO5	500 µg/1 mg

• SecinH3
  A cell-permeable triazolo compound that acts as a Sec7 domain-binding selective antagonist against cytohesin family of small GEFs

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203260	853625-60-2	C24H20N4O4S	5 mg

• sFRP-1 Inhibitor
  A cell-permeable diphenylsulfone-sulfonamide compound that acts as a selective and reversible inhibitor of sFRP-1, and potently activates canonical Wnt pathway. Shows a desirable aqueous solubility and in-vitro microsomal stability-human. Marginally affects cytochrome p450 isozymes.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222310	915754-88-0	C19H26N2O4S2	5 mg

• Siastatin B microbial
  A broad spectrum inhibitor of sialidase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215851	54795-58-3	C8H14N2O5	5 mg

• SID 7969543
  Selective steroidogenic factor-1 (SF-1, NR5A1) inhibitor (IC₅₀ values are 0.76, >33 and >33 μM at SF-1, RORα and VP16 respectively). Inhibits SF-1-dependent luciferase expression in HEK 293T cells in vitro (IC₅₀ = 30 nM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204278	868224-64-0	C24H24N2O7	10 mg/50 mg

• Sildenafil, Citrate
  A citrate form of Sildenafil and a selective inhibitor of the type 5 cGMP phosphodiesterase (PDE5 inhibitor). Additionally reported to enhance neuro-, synapto- and angiogenesis in rat models of stroke.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208388	171599-83-0	C22H30N6O4S•C6H8O7	50 mg

• Simvastatin
  A HMG-CoA reductase inhibitor with anti-proliferative properties. Shown to modulate purified bovine pituitary 20 S proteasome.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200829	79902-63-9	C25H38O5	50 mg/250 mg

• Sitagliptin Phosphate
  A trizolopyrazine dipeptidyl peptidase IV inhibitor that has recently been approved for type II diabetes therapy.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208391	654671-78-0	C16H15F6N5O ·H3PO4	1 mg

• Sivelestat
  A cell-permeable, potent, substrate-competitive, and highly specific inhibitor of neutrophil elastase (IC50 = 19-49 nM in rat, rabbit, hamster, human, and mouse leukocyte elastase).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203938	127373-66-4	C20H22N2O7S	1 mg

• Sivelestat sodium salt hydrate
  A competitive inhibitor of human neutrophil elastase (HNE), that has also been shown to inhibit leukocyte elastase obtained from several animal donors.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215858	201677-61-4	C20H29N2NaO11S	5 mg/25 mg

• SKF 91488 dihydrochloride
  This homologue of dimaprit is a strong inhibitor of histamine N-methyltransferase, with no histamine agonist activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203696	68643-23-2	C7H17N3S ·2HCl	10 mg/50 mg

• SM-19712
  A potent and selective nonpeptide endothelin converting enzyme inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215859	194542-56-8	C18H13ClN5NaO3S	5 mg/25 mg

• Sodium Copper Chlorophyllin
  A water soluble salt of chlorophyll which inhibits activation and degradation of electrophyllic intermediates.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205628	28302-36-5	C34H31CuN4Na3O6	5 g/25 g

• Sodium Phenylacetate
  An aromatic fatty acid, which displays cell growth inhibition, malignant phenotype reduction and cell differentiation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-296401	114-70-5	C8H7O2 ·Na	500 mg

• SPHK 1 Inhibitor 5C
  The sphingosine kinases (SphK) phosphorylate sphingosine, producing the important lipid mediator sphingosine-1-phosphate (S1P). The two known kinases, SphK1 and SphK2, have different developmental and tissue expression patterns, suggesting that they have distinct physiological functions. Notably, SphK1 is overexpressed in several forms of cancer and inhibition of SphK1 inhibits tumor growth. A selective inhibitor of SphK1, both in vitro (IC50 = 3. μM) and in U937 cells overexpressing human SphK1 (70 % inhibition at 5 μM). It has no inhibitory effect on SphK2 either in vitro or in cells. Similarly, this chemical does not reduce the activity of protein kinase C (PKC) except at very high concentration (>75 μM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-288340	120005-55-2	C26H45NO4	1 mg/5 mg

• SSR 69071
  Potent, orally active human leukocyte elastase inhibitor. Exhibits species selectivity. Inhibits HLE-induced lung hemorrhage in mice in vivo. In an acute model of coronary ischemia-reperfusion injury, reduces infarct size in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203702	344930-95-6	C27H32N4O7S	10 mg

• Steroidogenic Factor-1 Inhibitor, SID7970631
  A cell-permeable isoquinolinone compound that inhibits SF-1 functional activity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-311539	868224-75-3	C24H24N2O7	10 mg

• Strontium Ranelate
  A bone metabolism modulator that inhibits bone resorption while maintaining bone formation. Commonly used as an antiosteoporotic.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208403	135459-87-9	C12H6N2O8SSr2	10 mg

• Sulbactam

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-272516	68373-14-8	C8H11NO5S	100 mg

• Suplatast tosylate
  Th2 cytokine inhibitor that attenuates IL-2, IL-5 and IL-13 production and has no effect on IFN-γ production. Acts as an immunoregulator that suppresses IgE production, eosinophil infiltration and histamine release. Shows antiasthmatic, anti-inflammatory and antifibrotic activity in vivo and is orally active.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204315	94055-76-2	C16H26NO4S ·C7H7O3S	10 mg/50 mg

• Syk Inhibitor
  Oxindole compound that acts as a potent Syk inhibitor. Shown to effectively inhibit FcεRI-mediated degranulation in RBL-2H3.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204316	622387-85-3	C18H15N3O3S	5 mg

• (+/-)-Synephrine
  A α-adrenergic receptor agonist, vasoconstrictor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220182	94-07-5	C9H13NO2	25 g

• t-Butylhydroquinone
  A phenolic antioxidant functioning as an inhibitor of endoplasmic reticulum Ca²⁺-ATPase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202825	1948-33-0	C10H14O2	10 g

• T0070907
  Cell-permeable. Potent, specific, irreversible, and high-affinity antagonist of PPARγ.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203287	313516-66-4	C12H8ClN3O3	5 mg

• Tadalafil
  A phosphodiesterase 5 inhibitor. Used for the treatment of erectile dysfunction.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208412	171596-29-5	C22H19N3O4	50 mg

• TAK 165

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361372	366017-09-6	C25H23F3N4O2	10 mg/50 mg

• Talsaclidine Hydrochloride
  A novel M1-receptor selective muscarinic agonist for cholinergic substitution used in the therapy for Alzheimer's disease. Treatment decreases cerebrospinal fluid levels of A beta 42 in patients.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220185	N/A	C10H16ClNO	5 mg

• TAPI-0
  Hydroxamate-based inhibitor of collagenase, gelatinase, and TACE. Blocks spontaneous and PMA-induced release of TNF-α.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203410	143457-40-3	C24H32N4O5	1 mg

• TAS-301
  Inhibits migration and proliferation in vascular smooth muscle cells and also inhibits restenosis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215942	193620-69-8	C23H19NO3	10 mg

• Taurine
  Inhibitor of lipid peroxidation. Inhibits diethylnitrosamine and phenobarbital-induced hepatocarcinogenesis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202354	107-35-7	C2H7NO3S	10 g

• TCS PrP Inhibitor 13
  Antiprion agent that potently inhibits protease-resistant prion protein (PrP-res) accumulation in two types of prion-infected mouse neuroblastoma (N2a) cell lines (IC₅₀= 3 nM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204331	34320-83-7	C15H11N3O3	10 mg/50 mg

• Teijin compound 1
  A potent chemokine CCR2b receptor antagonist (IC50 = 180 nM). Shown to potently inhibit cell chemotaxis induced by MCP-1 (EC50 = 24 nM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-301864	226226-39-7	C21H21CIF3O2.HCl	10 mg/50 mg

• Telmisartan
  Angiotensin II receptor antagonist that inhibits the angiotensin II AT1 receptor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204907	144701-48-4	C33H30N4O2	50 mg/100 mg

• Telomerase Inhibitor IX
  A synthetic compound that acts as a reversible telomerase inhibitor, described to be more potent than epigallocatechin gallate.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204333	368449-04-1	C20H16N2O6	10 mg

• Temocapril Hydrochloride
  An ACE inhibitor (angiotensin converting enzyme). Pro-drug that is converted in vivo to treat hypertension.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204908	110221-44-8	C23H28N2O5S2•HCl	10 mg/25 mg

• Tetraisopropyl Dichloromethylene Diphosphonate
  An intermediate in the sythesis of Clodronic Acid, Disodium Salt, Tetrahydrate, which is a biphosphonate bone resorption inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220223	10596-22-2	C13H28Cl2O6P2	50 mg

• Tetraisopropyl pyrophosphoramide
  A selective inhibitor of butyrylcholinesterase.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215956	513-00-8	C12H32N4O3P2	100 mg/250 mg

• Tetramisole hydrochloride
  Suitable for inhibition of various mammalian alkaline phosphatase (i.e., liver, kidney, placenta, bone and tumor)(Intestinal alkaline phosphatases are only slightly inhibited.)

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215963	5086-74-8	C11H12N2S ·HCl	2 g/5 g

• Thielavin B
  A potent prostaglandin synthetase inhibitor derived from Thielavia terricola. Shown to inhibits the synthesis of prostaglandin E2 from endoperoxides.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202362	71950-67-9	C31H34O10	500 µg

• Thiolactomycin
  Inhibits bacterial myristate synthesis where it does not inhibit eukaryotic myristate synthesis. Exhibits antibiotic and antitrypanosomal activity. Recently it has been shown to be an effective agent against the human sleeping sickness parasite, Trypanosoma brucei, as well as malaria parasites and toxoplasmas.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-215970	82079-32-1	C11H14O2S	10 mg

• Tie-2 Inhibitor 13
  Shown to be a potent and cell permeable Tie-2 inhibitor (IC50=600nm).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-358703	857250-95-4	C17H13FO2S	1 mg

• Tie-2 Inhibitor 7
  A compound that can permeate the cell (IC₅₀= 1uM) and inhibit endothelial cell tube formation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202363	1020412-97-8	C31H29N3O5	1 mg

• Tin Protoporphyrin IX dichloride
  A potent inhibitor of heme oxygenase. Prevents hyperbilirubinemia in neonates.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203452	14325-05-4	C34H32N4O4Sn•2Cl	5 mg/25 mg

• Tipranavir
  Nonpeptidic HIV protease inhibitor (NPPI). Antiviral.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220260	174484-41-4	C31H33F3N2O5S	1 mg

• TJU103
  This is a non-peptidic organic compound that specifically blocks stable CD4-MHC class II binding. Exhibits significant inhibition of immune responses in animal models of autoimmune disease and allograft transplant rejection, which suggests that its potential as a novel immunosuppressant. It does not exhibit any toxic effects in vivo, with normal lymphocyte cellularity and subset composition in the spleen and lymph nodes of mice 24 h after injection.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222358	N/A	C15H12N4O	50 mg

• TMPyP4
  An aromatic cationic porphyrin ligand that binds and stabilizes the quadruplex structure of telomeric DNA. Inhibition of telomerase acitvity has been shown to cause cell growth arrest.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204346	36951-72-1	C44H38N8 ·C28H28O12S4	25 mg

• TMS
  Strong, selective and competitive inhibitor of cytochrome P450 1B1, an overexpressed enzyme in particular tumors (IC₅₀ = 6 nM). 50- and 520-fold selective over P450 1A1 and 1A2 respectively. Inhibits cancer cell growth in vitro.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203708	24144-92-1	C18H20O4	10 mg/50 mg

• TNP 470
  An analog of Fumagillin (sc-200377) that displays potent antiangiogenic activity in vitro and in vivo. Shown to inhibit methionine aminopeptidase type II (MetAP2).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-296547	129298-91-5	C19H28CINO6	5 mg

• TNP-AECM-FICOLL
  TNP (2,4,6-Trinitrophenyl) hapten is conjugated to AminoEthylCarboxyMethyl-FICOLL (AECM-FICOLL), a high molecular weight polysaccharide; useful as T-independent antigens for studying B lymphocyte activation.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-281696	N/A	N/A	10 mg/100 mg

• TNP(12)-BSA (Bovine Serum Albumin)
  A compound used to elicit an immune response in research animals. Contains a 2,4,6-Trinitrophenyl hapten, which is conjugated to bovine serum albumin. TNP to BSA molar ratio is approximately 12. For higher molar ratio, please see sc-360249 (molar ratio approximately 26).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-281697	N/A	C6H3N4O6-BSA	10 mg

• TNP(26)-BSA (Bovine Serum Albumin)
  A compound used to elicit an immune response in research animals. Contains a 2,4,6-Trinitrophenyl hapten, which is conjugated to bovine serum albumin. TNP to BSA molar ratio is approximately 26. For a lower molar ratio, please see sc-281697 (molar ratio approximately 12).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-362049	N/A	C6H3N4O6-BSA	10 mg

• Tolterodine L-Tartrate

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220271	124937-52-6	C26H37NO7	10 mg

• Torsemide
  Used as a diuretic.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-213059	56211-40-6	C16H20N4O3S	10 mg

• Trandolapril
  Angiotensin-converting enzyme (ACE) inhibitor with long biological half-life and a high degree of lipophilicity.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203299	87679-37-6	C24H34N2O5	10 mg/50 mg

• trans 2-Phenylcyclopropylamine Hydrochloride
  A non-selective MAO-A/B inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208452	1986-47-6	C9H12ClN	250 mg/1 g

• trans-HR22C16
  Cell permeable non-tubulin-interacting mitosis inhibitor. Blocks mitosis (IC₅₀=800nM) by binding to the mitotic kinesin Eg5.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202842	462630-41-7	C23H23N3O3	1 mg

• Triflumuron
  Chitin biosynthesis inhibitor. Has displayed to inhibit uridine incorporation into RNA.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205873	64628-44-0	C15H10ClF3N2O3	10 g/25 g

• Trilostane
  An inhibitor of isoforms 3β-HSD and 3β-HSD2 of 3β-hydroxysteroid dehydrogenase. A useful tool in steroid biosynthesis research.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208469	13647-35-3	C20H27NO3	10 mg/100 mg

• Triparanol
  An inhibitor of delta 24-reductase and an inhibitor of cholesterol biosynthesis. Described to inhibit Hedgehog pathway signaling and useful as a probe for studying the pathway.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208472	78-41-1	C27H32ClNO2	5 mg

• Tris DBA
  N-myristoyltransferase-1 (NMT-1) inhibitor that prevents activation of MAPK, PI 3-K and STAT3 signaling pathways. Used as a cyclization catalyst. Exhibits antiproliferative activity against melanoma cells in vitro and in vivo.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204355	52522-40-4	C52H43Cl3O3Pd2	10 mg/50 mg

• Tubulozole-T hydrochloride
  An anti-malarial agent that does not inhibit microtubule assemby. An inactive trans-isomer of tubulozole-C .

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216030	95480-32-3	C23H23Cl2N3O4S··HCl	50 mg

• U-73122 hydrate
  A phospholipase C inhibitor. This compound can inhibit the hydrolysis of phosphatidylinositol stimulated by cholecystokinin or carbachol.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216035	112648-68-7 (anhydrous)	C29H40N2O3 ·xH2O	5 mg

• U-73343
  An inactive structural analog of U-73122. Useful as a negative control for phospholipase C antagonism studies.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201422	142878-12-4	C29H42N2O3	5 mg/25 mg

• Ubiquinone-10
  Inhibitor of the mitochondrial permeability transition pore (MPTP). This inhibitory effect can be counteracted by ubiquinone-5

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202375	606-06-4	C19H26O4	2 mg

• Ubiquitin Isopeptidase Inhibitor II, F6
  Cell-permeable cross-conjugated alpha,beta-unsaturated dienone compound that induces caspase activation and apoptosis (IC50 = 15.65 and 16.23 µM in E1A and E1A/C9DN cells, respectively) via the apoptosome-independent mitochondrial pathway, selectively inhibiting ubiquitin isopeptidase activity. The cellular expression of Bax and Bak is essential for F6-activated apoptosis, while Bcl-2 appears to protect cells against the effect of F6.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-296678	157654-67-6 (HCl salt)	C21H21NO	10 mg

• UBP 310

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361389	N/A	C14H15N3O6S	10 mg/50 mg

• UCB 35625
  Potent chemokine CCR1 and CCR3 receptor antagonist. Inhibits MIP-1α-induced chemotaxis in CCR1 transfectants and eotaxin-induced chemotaxis in CCR3 transfectants (IC₅₀values are 9.57 and 93.8 nM respectively). Antagonizes CCR3-mediated entry of HIV-1 isolate 89.6 into NP-2 cells (IC₅₀ = 57 nM). Isomer of J 113863 (sc-203611).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204369	301648-08-8	C30H37Cl2IN2O2	1 mg/10 mg

• UCH-L3 Inhibitor
  1,3-indanedione compound that acts as a selective and potent inhibitor of UCH-L3 (IC₅₀ = 0.6 µM) with ~125-fold greater selectivity over UCH-L1 (IC₅₀ = 75 µM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204370	30675-13-9	C9H2Cl4O2	10 mg

• UCPH 101

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361391	1118460-77-7	C27H22N2O3	10 mg/50 mg

• V2R Antagonist, V2Rnh-02
  This is a pyrrolone compound that acts as a ligand-competitive vasopressin receptor antagonist with ~70-fold greater affinity for V2R than V1aR (IC₅₀ against arginine vasopression binding = 70 nM and 5 µM, respectively). It has shown to selectively inhibit cellular cAMP production mediated by V2R (IC₅₀ = 60 nM), but not β2-adrengergic receptor. It is reported to exhibit great aqueous solubility (377 µM in PBS) with a pKa of 4.76.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222408	N/A	C25H20FNO4	10 mg

• Vardenafil

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-362054	224785-90-4	C23H32N6O4S	100 mg/1 g

• Vatalanib Dihydrochloride
  Inhibits VEGFR-dependent tumor angiogenesis and EGFR- and RET-dependent tumor cell proliferation and survival. Is the active ingredient in the drug sold under the trade name Zactima™.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-202379	212141-51-0	C20H15ClN4 ·2HCl	5 mg/25 mg

• VER 155008

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-358808	1134156-31-2	C25H23Cl2N7O4	10 mg/50 mg

• VER-50589
  The heat shock proteins (Hsps) act as molecular chaperones. Hsp90 is an abundant protein with roles in protein folding, cell signaling, and cancer. VER-50589 is an isoxazole compound that inhibits Hsp90 with an IC50 value of 21 nM. It produces a mean cellular antiproliferative GI50 value of 78 nM when tested against a human cancer cell line panel. Consistent with inhibition of Hsp90, VER-50589 induces the expression of HSP27 and Hsp72 while reducing the client proteins C-RAF, B-RAF, survivin, and PRMT5, causing cell cycle arrest and apoptosis. VER-50589 shows favorable pharmacokinetics and impairs tumor growth in animals. Importantly, glioblastoma cells do not acquire resistance to VER-50589 and resistance to other Hsp90 inhibitors does not produce cross-resistance to VER-50589.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-296692	747413-08-7	C19H17ClN2O5	500 µg/1 mg

• VU0155069
  Phospholipase D (PLD) is an enzyme that cleaves the head group from phospholipids, producing the second messenger phosphatidic acid. Two mammalian isoforms of PLD (PLD1 and PLD2) have been identified, with multiple splice variants of each. Although the two isoforms share functional and structural features, they are regulated differently and apparently subserve distinct roles. VU0155069 is a selective and potent inhibitor of PLD1, both in vitro (IC₅₀ = 46 nM) and in cells (IC₅₀ = 11 nM). It is also effective as a PLD2 inhibitor at higher concentrations (IC₅₀ = 933 nM in vitro, 1,800 nM in cells). VU0155069 strongly inhibits the invasive migration of several breast cancer cell lines in transwell assays, suggesting that PLD might be a useful target in blocking tumor cell invasion.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-224371	1130067-06-9	C26H27ClN4O2	1 mg/5 mg

• VULM 1457
  Acyl-CoA: cholesterol acyltransferase (ACAT) inhibitor. Decreases cholesterol levels in the liver and plasma of diabetic-hypercholesterolaemic rats.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204390	228544-65-8	C25H27N3O3S	10 mg/50 mg

• W-5 Isomer hydrochloride
  Isomer of W-5 (sc-201500).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208488	35517-14-7	C15H20N2O2S•HCl	1 mg/5 mg

• W-7 Isomer hydrochloride
  Inhibitor of calmodulin. Isomer of W-7(sc-201501)

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203311	69762-85-2	C16H21ClN2O2S ·HCl	5 mg/25 mg

• W140 trifluoroacetate salt
  Sphingosine-1-phosphate (S1P) is a bioactive lipid that exhibits a broad spectrum of biological activities including cell proliferation, survival, migration, cytoskeletal organization, and morphogenesis. It exerts its activity by binding to five distinct G protein-coupled receptors, S1P1/EDG-1, S1P2/EDG-5, S1P3/EDG-3, S1P4/EDG-6, and S1P5/EDG-8. W140 (trifluoroacetate salt) is an inactive enantiomer of W146, a selective S1P1 antagonist (Ki = 77 nM), that binds to the S1P1 receptor with a Ki of 4.6 µM (2a = W146; 2b = W140 in supplemental material). It exhibits no biological activity in vivo and can therefore serve as an effective control compound for experiments involving W146.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-296699	N/A	C16H27N2O4P•C2F3HO2	500 µg/1 mg

• Wiskostatin
  A cell-permeable N-alkylated carbazole derivative that selectively blocks actin filament assembly. Acts as a selective, reversible inhibitor of N-WASP (neural Wiskott Aldrich syndrome protein), a signal integrating protein. Appears to bind to N-WASP, stabilize the autoinhibited conformation and prevent the activation of Arp2/3 (actin-related protein 2/3) complex.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204399	253449-04-6	C17H18Br2N2O	1 mg/5 mg

• Wnt Agonist
  A cell-permeable compound that acts as a potent and selective activator of Wnt signaling without inhibiting the activity of GSK-3β.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222416	N/A	C19H18N4O3	5 mg

• Wnt Synergist, QS11
  A cell-permeable purine compound that binds GTPase activating proteins of ADP-ribosylation factor and acts as a broad specificity ARFGAPs inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222417	N/A	C36H33N5O2	5 mg

• XR 9051 HCl

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-361409	180422-22-4	C39H38N4O5•HCl•xH2O	10 mg/50 mg

• Y-29794 oxalate
  Prolyl endopeptidase inhibitor, a serine peptidase that may be implicated in the biosynthesis of amyloid b-peptide. Potently inhibits rat brain prolyl endopeptidase (Ki = 0.95 nM) in vitro, and prevents amyloid b-peptide deposition in vivo. Orally active and brain penetrant.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204408	129184-48-1	C23H34N2OS2.C2H2O4	10 mg/50 mg

• YIC-C8-434
  Acyl-CoA:cholesterol acyltransferase (ACAT) inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-216068	214265-97-1	C31H44N2O4	5 mg

• YM-53601
  YM-53601 inhibits squalene synthase activity in rat hepatic microsomes and human HepG2 cells. Displaying an ED₅₀ value of 32 mg/kg of YM-53601, cholesterol biosynthesis is inhibited, causing a reduction in both cholesterol and triglyceride levels in plasma. Cholesterol-reducing HMG-CoA reductase inhibitors are often paired with fibrates, which can have adverse effects, to treat hyperlipidemia.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-205543	182959-33-7	C21H21FN2O•HCl	500 µg/1 mg

• γ-Secretase Inhibitor I
  An inhibitor of γ-secretase, a protease that cleaves the amyloid precursor protein (APP). The inhibition of this enzyme is believed to aid in the prevention of Alzheimer's disease.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-301796	133407-83-7	C26H41N3O5	1 mg

• γ-Secretase Inhibitor III
  A cell-permeable reversible inhibitor of Aβ and p3 secretion (Aβ40 IC50 = 2.3 µM; Aβ42 IC50 = 3 µM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-301797	N/A	C23H42N2O4	1 mg/5 mg

• Z-FA-FMK
  An irreversible inhibitor of cathepsins B, L, and S, cruzain and papain. Inhibits effector, but not initator, caspases in vitro, and suppresses some forms of caspase mediated apoptosis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201303	197855-65-5	C21H23FN2O4	1 mg/5 mg

• Z-Gly-Phe-NHO-Bz
  Z-Gly-Phe-NHO-Bz has been shown to Inhibit Cathepsin L, Cathepsin S, Cathepsin B.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-358593	N/A	C11H11N3O2	1 mg/5 mg

• Z-Guggulsterone

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204414	39025-23-5	C21H28O2	10 mg/25 mg

• Z-L-Abu-CONH-ethyl
  A cell-permeable dipeptidyl α-ketoamide that acts as a potent, reversible, and active site inhibitor of calpain-1 and calpain-2 (Ki ~ 250 nM). At 10-fold higher concentration it also inhibits cathepsin B (Ki = 2.4 µM). Has been shown to have a neuroprotective role in the central nervous system following focal ischemia.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-301995	N/A	C21H31N3O5	1 mg

• Z-L-Abu-CONH(CH2)3-morpholine
  A cell-permeable dipeptidyl α-ketoamide that acts as a potent, highly selective, reversible, and active site inhibitor of calpain-1 and calpain-2 (Ki = 140 nM and 41 nM, respectively). A weak inhibitor of cathepsin B (Ki = 6.9 µM). Has been shown to have a neuroprotective role in the central nervous system following focal ischemia. Also protects against virus-induced apoptotic myocardial injury in mice.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-301996	N/A	C26H40N4O6	1 mg/5 mg

• Z-Phe-Tyr(tBu)-diazomethylketone
  An irreversible inhibitor of cathepsin L.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-222423	N/A	C31H34N4O5	1 mg

• Z-Prolyl-prolinal
  Z-PP-CHO, a potent and specific, cell-permeable dipeptide aldehyde inhibitor of prolyl endopeptidase (PREP)

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-201285	86925-97-5	C18H22N2O4	5 mg/25 mg

• Z-VAD(OMe)-FMK
  An irreversible and cell permeable caspase inhibitor that has been shown to inhibit Fas-mediated apoptosis in Jurkat T-cells.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-311561	187389-52-2	C22H30FN3O7	1 mg

• Z-Val-Val-Nle-diazomethylketone
  An irreversible cathepsin inhibitor that is 380 times more effective in inactivating cathepsin S than L. Is often abbreviated as DMK. Peptidyl diazomethyl ketones are specific inactivators of thiol proteinases.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-301998	N/A	N/A	50 mg

• (Z)-Pugnac
  An inhibitor of O-GlcNAcase, an enzyme which removes the N-acetylglucosamine moieties from 2-acetamido-2-deoxy-&beta-D-glucopyranose (O-GlcNAc) bound to proteins that were modified by O-GlcNAc.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204415	132489-69-1	C15H19N3O7	10 mg/5 mg

• Zaragozic acid A trisodium salt
  This product is a potent inhibitor, in vivo and in vitro, of mammalian, fungal and Saccharomyces cervisiae squalene synthase. As a squalene synthase inhibitor, zaragozic acid has been shown to produce lower plasma cholesterol levels in primates.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-302001	144541-82-2	C35H46Na3O14	5 mg

• Zatebradine hydrochloride
  Bradycardic agent that creates use-dependent inhibition of hyperpolarization-activated current (If) in sinoatrial node cells (EC₅₀ = 480 nM) and Purkinje fibres. Displays negative chronotropic activity in isolated guinea pig atria (EC₅₀ of 13.4 μM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-203724	91940-87-3	C26H36N2O5•HCl	10 mg/50 mg

• ZM-447439
  A selective inhibitor of aurora kinases ARK-1, ARK-2, and ARK-3 (A, B, C), that can induce growth arrest, inhibit histone H3 phosphorylation and effectively activate apoptosis.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-200696	331771-20-1	C29H31N5O4	1 mg/10 mg

• Zofenopril Calcium Salt
  An antioxidant that acts as an angiotensin-converting enzyme inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208496	81938-43-4	C44H44CaN2O8S4	10 mg

• Zoledronic Acid, Disodium Salt, Tetrahydrate
  A biphosphonate bone resorption inhibitor.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-208497	165800-07-7	C5H8N2Na2O7P2•4H2O	50 mg

• Zolmitriptan
  A Serotonin 5HTID-receptor agonist.

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-220415	139264-17-8	C16H21N3O2	10 mg

• Zoniporide dihydrochloride
  Sodium-hydrogen exchanger isoform-1 (NHE-1) inhibitor that displays selectivity over other NHE isoforms (K_i values are 14, 2200 and 220000 nM for human NHE-1, human NHE-2 and rat NHE-3 respectively). Inhibits NHE-1 dependent 22Na⁺ uptake in vitro (IC₅₀ = 14 nM) and provides cardioprotection from myocardial ischemic injury in vivo (EC₅₀ = 0.25 nM).

  Catalog #	CAS Number	Molecular Formula	Unit
  sc-204423	241800-97-5	C17H16N6O ·2HCl	10 mg/50 mg