AR Activators

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For functional analysis of AR Activators, see our complete listing of AR Antibodies.

PRODUCT NAME	CATALOG #	DESCRIPTION	CITATIONS	RANKING
Andarine	sc-364405	Andarine stimulates AR-mediated transcription to 93% of that observed for 1 nM DHT at a concentration of 10 nM. CAS # 401900-40-1
A 61603 HYDROBROMIDE	sc-203789	Potent α-adrenoceptor agonist, at least 35-fold more potent at α1A than at α1B or α1D sites. CAS # 107756-30-9
CGP 12177 hydrochloride	sc-203878	CGP 12177 hydrochloride is a β1-AR and β2-AR adrenoreceptor antagonist. Also behaves non-conventionally as a β3-AR partial agonist. CAS # 81047-99-6
B-HT 920	sc-203523	B-HT 920 is a dopamine D2 receptor agonist, SR-3 antagonist and α2-adrenoceptor agonist. It also displays antiparkinsonian activity. CAS # 36085-73-1
Carvedilol	sc-200157	Carvedilol is an α1 and β-adrenergic receptor (AR) agonist selective towards α1D-AR and α1B-AR and possesses antioxidant properties. CAS # 72956-09-3
Cimaterol	sc-203549	Cimaterol is a β-AR adrenergic agonist. β-AR agonists in general have opposite activities as beta-blockers. CAS # 54239-37-1
Cirazoline hydrochloride	sc-203550	Selective a1 agonist CAS # 40600-13-3
CL 316243 disodium salt	sc-203895	CL 316243 disodium salt is a highly selective β3-AR adrenoceptor agonist that has been shown to increase adipose tissue thermogenesis. CAS # 151126-84-0
Clonidine hydrochloride	sc-203002	Clonidinie hydrochloride is an antihypertensive α2-AR adrenergic receptor agonist and I1 imidazoline receptor ligand. CAS # 4205-91-8	8
Dobutamine Hydrochloride	sc-203031	Dobutamine Hydrochloride is a derivative of dopamine and has exhibited usage as a β1-AR adrenergic agonist. CAS # 49745-95-1
Formoterol Fumarate	sc-203050	Formoterol Fumarate has been shown to be a potent agonist of β-AR adrenoceptor with selectivity for β2-AR than β1-AR receptors. CAS # 43229-80-7
Guanabenz acetate	sc-203590	Guanabenz acetate is an α2A-AR adrenergic agonist and IGRS (imidazoline I2 binding site) selective ligand. CAS # 23256-50-0
Guanfacine hydrochloride	sc-203988	Guanfacine hydrochloride is an anti-hypertensive agent that has been shown to be a specific α2A-AR adrenoceptor agonist. CAS # 29110-48-3
Isoproterenol Hydrochloride	sc-202188	Isoproterenol Hydrochloride is a phenethylamine derivative and selective β-AR adrenergic agonist shown to increase cytosolic cAMP. CAS # 51-30-9
L-(-)-Epinephrine-(+)-bitartrate	sc-204032	L-(-)-Epinephrine-(+)-bitartrate is an α,β-adrenergic receptor agonist. L-(-)-Epinephrine-(+)-bitartrate has positive chronotropic and inotropic effects. CAS # 51-42-3
L-(–)-Norepinephrine-(+)-bitartrate	sc-203093	L-(–)-Norepinephrine-(+)-bitartrate is a bitartrate preparation of the α,β-adrenoceptor agonist norepinephrine. CAS # 69815-49-2
L-755,507	sc-204045	L-755,507 is a very potent and selective β3-AR adrenergic receptor partial agonist, selective over both β1-AR and β2-AR adrenoceptor binding. CAS # 159182-43-1
Medetomidine hydrochloride	sc-204073	Medetomidine hydrochloride is a potent and highly selective α2-AR adrenoceptor agonist. CAS # 106807-72-1
Naphazoline Hydrochloride	sc-205764	Naphazoline hydrochloride produces ionotropic effects via α-adrenoceptor stimulation. CAS # 550-99-2
Octopamine Hydrochloride	sc-203168	Octopamine hydrochloride is an activator of β3-AR and α2A-AR adrenoceptors. CAS # 770-05-8
Oxymetazoline Hydrochloride	sc-203172	Oxymetazoline Hydrochloride is a direct sympathomimetic agent and a nonselective adrenomimetic of α1-AR and α2-AR adrenergic receptor agonists. CAS # 2315-02-8	1
(R)-(-)-Phenylephrine hydrochloride	sc-203677	Phenylephrine (PE) is an α1-adrenoceptor agonist that promotes hypertrophic growth in the ventricular myocytes, and activates several MAPK signaling pathways. CAS # 61-76-7
Ritodrine	sc-204882	Ritodrine is a β2-adrenoceptor agonist that acts as an adrenergic receptor stimulant. CAS # 23239-51-2
Salbutamol hemisulfate	sc-203373	Salbutamol hemisulfate is a non-selective, short-acting β2-AR adrenergic receptor agonist that displays more potency at β2 receptors than β1. CAS # 51022-70-9
Salmeterol	sc-224277	Salmeterol is a potent and selective β2-AR adrenoceptor agonist shown to bind to the exo-site domain of the receptor. CAS # 89365-50-4
Tizanidine • HCl	sc-200148	Tizanidine • HCl is a centrally acting α2-adrenergic (α2-AR). Displays affinity for the I1-imidazoline receptor and exhibits spasmolytic activity. CAS # 64461-82-1
(±)-Epinephrine	sc-252779	±)-Epinephrine is an adrenoceptor agonist. The L-form is a direct-acting sympathomimetic agent with pronounced effect on alpha- and beta-adrenergic receptors. CAS # 329-65-7
Xylazine	sc-253838	Xylazine (Rompun) is an α2 class of adrenergic receptor agonist. Xylazine is a clonidine analoque that acts on presynaptic and postsynaptic receptors of the central and peripheral nervous systems. CAS # 7361-61-7
Detomidine HCl	sc-357329	Detomidine HCl is a nonnarcotic, synthetic alpha-2 adrenoreceptor agonist. Detomidine HCl is a sedative with analgesic properties. CAS # 90038-01-0
Moxonidine hydrochloride	sc-204096	Centrally acting antihypertensive agent. Mixed I1 imidazoline receptor and α2-adrenergic agonist; displays 40-fold higher affinity for I1 receptors versus α2-adrenoceptors. CAS # 75438-57-2
DL-Isoproterenol Hemisulfate	sc-294398	This is a bronchodilator. CAS # 6078-56-4